NO153430C - Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme 2-fenyl eller -pyridyl-pyrazolo(4,3-c)kinolin-3(1 og 5h)-on forbindelser. - Google Patents
Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme 2-fenyl eller -pyridyl-pyrazolo(4,3-c)kinolin-3(1 og 5h)-on forbindelser.Info
- Publication number
- NO153430C NO153430C NO801866A NO801866A NO153430C NO 153430 C NO153430 C NO 153430C NO 801866 A NO801866 A NO 801866A NO 801866 A NO801866 A NO 801866A NO 153430 C NO153430 C NO 153430C
- Authority
- NO
- Norway
- Prior art keywords
- hydroxy
- alkyl
- phenyl
- see diagramm
- hydrogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/56—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups bound to carbon atoms of six-membered aromatic rings and carboxyl groups bound to acyclic carbon atoms of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/28—Two oxygen or sulfur atoms
- C07D231/30—Two oxygen or sulfur atoms attached in positions 3 and 5
- C07D231/32—Oxygen atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Electrophonic Musical Instruments (AREA)
- Golf Clubs (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5071679A | 1979-06-21 | 1979-06-21 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO801866L NO801866L (no) | 1980-12-22 |
| NO153430B NO153430B (no) | 1985-12-09 |
| NO153430C true NO153430C (no) | 1986-03-19 |
Family
ID=21966959
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO801866A NO153430C (no) | 1979-06-21 | 1980-06-20 | Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme 2-fenyl eller -pyridyl-pyrazolo(4,3-c)kinolin-3(1 og 5h)-on forbindelser. |
Country Status (22)
| Country | Link |
|---|---|
| EP (1) | EP0022078B1 (da) |
| JP (1) | JPS5618980A (da) |
| KR (1) | KR840000421B1 (da) |
| AT (1) | ATE8629T1 (da) |
| AU (1) | AU538890B2 (da) |
| CA (1) | CA1148159A (da) |
| CY (1) | CY1357A (da) |
| DD (1) | DD151754A5 (da) |
| DE (1) | DE3068673D1 (da) |
| DK (1) | DK160762C (da) |
| FI (1) | FI68827C (da) |
| GR (1) | GR69282B (da) |
| HK (1) | HK47387A (da) |
| HU (1) | HU183156B (da) |
| IE (1) | IE49993B1 (da) |
| IL (1) | IL60357A (da) |
| MY (1) | MY8700556A (da) |
| NO (1) | NO153430C (da) |
| NZ (1) | NZ194102A (da) |
| PT (1) | PT71420A (da) |
| SG (1) | SG14387G (da) |
| ZA (1) | ZA803714B (da) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4459298A (en) * | 1982-09-28 | 1984-07-10 | Ciba-Geigy Corporation | Method of suppressing appetite |
| US4524146A (en) * | 1982-12-08 | 1985-06-18 | Ciba-Geigy Corporation | Certain -2-heterocycle substituted pyrazoloquinolines |
| US4479955A (en) * | 1983-01-10 | 1984-10-30 | Ciba-Geigy Corporation | Heterocycle-fused pyrazolo[3,4-d]pyridin-3-ones as benzodiazepine receptor modulators |
| EP0126970A3 (en) * | 1983-04-27 | 1985-11-06 | Beecham Group Plc | Anxiolytic and anti-depressant thienopyridine derivatives |
| FR2549833B1 (fr) * | 1983-07-26 | 1985-11-08 | Roussel Uclaf | Derives de la pyrazolo /4,3-c/ cinnolin-3-one, leurs sels, procede de preparation, application a titre de medicaments, compositions les renfermant et produits intermediaires |
| CA1263651A (en) * | 1984-07-09 | 1989-12-05 | Ciba-Geigy Ag | Certain ring-fused pyrazolo ¬3,4-d|-pyridin-3-one derivatives |
| PH21213A (en) * | 1984-10-26 | 1987-08-21 | Fujisawa Pharmaceutical Co | Benzene- and pyrazole- fused heterocyclic compound and pharmaceutical composition comprising the same |
| JPS61112075A (ja) * | 1984-11-05 | 1986-05-30 | Shionogi & Co Ltd | チエニルピラゾロキノリン誘導体 |
| DE3728278A1 (de) * | 1986-12-17 | 1988-06-23 | Bayer Ag | Herbizide und fungizide mittel auf basis von substituierten pyrazolin-5-on derivaten |
| US5243049A (en) * | 1992-01-22 | 1993-09-07 | Neurogen Corporation | Certain pyrroloquinolinones: a new class of GABA brain receptor ligands |
| GB9625398D0 (en) * | 1996-12-06 | 1997-01-22 | Merck Sharp & Dohme | Method of treatment,manufacture,compositions and compounds |
| US6835707B1 (en) | 1998-10-13 | 2004-12-28 | The Procter & Gamble Company | Laundry detergent compositions with a combination of cyclic amine based polymers and hydrophobically modified carboxy methyl cellulose |
| GB0305876D0 (en) * | 2003-03-14 | 2003-04-16 | Avidex Ltd | Immuno inhibitory heterocyclic compounds |
| JP2010529144A (ja) * | 2007-06-08 | 2010-08-26 | ヘリコン・セラピューティクス・インコーポレーテッド | 治療用ピラゾロキノリン尿素誘導体 |
| US8426438B2 (en) * | 2009-10-01 | 2013-04-23 | Merck Sharp & Dohme Corp. | Heterocyclic-fused pyrazolo[4,3-c]pyridin-3-one M1 receptor positive allosteric modulators |
| WO2011049731A1 (en) * | 2009-10-21 | 2011-04-28 | Merck Sharp & Dohme Corp. | Quinolinone-pyrazolone m1 receptor positive allosteric modulators |
| EP2699572B1 (en) | 2011-04-21 | 2016-08-10 | Origenis GmbH | Heterocyclic compounds as kinase inhibitors |
| WO2014060113A1 (en) | 2012-10-19 | 2014-04-24 | Origenis Gmbh | Novel kinase inhibitors |
| CN114891236B (zh) * | 2022-06-09 | 2023-04-28 | 安庆师范大学 | 一种三维Co-MOF化合物及其制备方法和应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3890324A (en) * | 1974-04-12 | 1975-06-17 | Lilly Co Eli | 1h-pyrazolo(4,3-)quinol-4(5h)-one-3-carboxylic acids |
| EP0005745B1 (en) * | 1978-05-26 | 1982-07-14 | Gruppo Lepetit S.P.A. | Pyrazolo (3,4-c) and thiazolo (5,4-c) isoquinolines, methods for preparing them, these compounds for use as antiinflammatory, cns-depressant and anti-anxiety agents and pharmaceutical compositions thereof |
-
1980
- 1980-06-16 CY CY135780A patent/CY1357A/xx unknown
- 1980-06-16 DE DE8080810200T patent/DE3068673D1/de not_active Expired
- 1980-06-16 EP EP80810200A patent/EP0022078B1/de not_active Expired
- 1980-06-16 AT AT80810200T patent/ATE8629T1/de not_active IP Right Cessation
- 1980-06-18 FI FI801964A patent/FI68827C/fi not_active IP Right Cessation
- 1980-06-19 GR GR62257A patent/GR69282B/el unknown
- 1980-06-19 PT PT71420A patent/PT71420A/pt unknown
- 1980-06-19 IL IL60357A patent/IL60357A/xx unknown
- 1980-06-19 CA CA000354349A patent/CA1148159A/en not_active Expired
- 1980-06-20 AU AU59455/80A patent/AU538890B2/en not_active Ceased
- 1980-06-20 NZ NZ194102A patent/NZ194102A/xx unknown
- 1980-06-20 ZA ZA00803714A patent/ZA803714B/xx unknown
- 1980-06-20 NO NO801866A patent/NO153430C/no unknown
- 1980-06-20 DK DK264880A patent/DK160762C/da not_active IP Right Cessation
- 1980-06-20 KR KR1019800002438A patent/KR840000421B1/ko active
- 1980-06-20 IE IE1279/80A patent/IE49993B1/en not_active IP Right Cessation
- 1980-06-21 JP JP8449380A patent/JPS5618980A/ja active Granted
- 1980-06-23 DD DD80222091A patent/DD151754A5/de unknown
- 1980-08-21 HU HU801539A patent/HU183156B/hu unknown
-
1987
- 1987-02-17 SG SG143/87A patent/SG14387G/en unknown
- 1987-06-18 HK HK473/87A patent/HK47387A/xx unknown
- 1987-12-30 MY MY556/87A patent/MY8700556A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI801964A (fi) | 1980-12-22 |
| ZA803714B (en) | 1981-06-24 |
| FI68827C (fi) | 1985-11-11 |
| ATE8629T1 (de) | 1984-08-15 |
| DE3068673D1 (en) | 1984-08-30 |
| AU5945580A (en) | 1981-01-08 |
| NZ194102A (en) | 1983-04-12 |
| JPH039114B2 (da) | 1991-02-07 |
| NO153430B (no) | 1985-12-09 |
| EP0022078A1 (de) | 1981-01-07 |
| IE801279L (en) | 1980-12-21 |
| HU183156B (en) | 1984-04-28 |
| DK264880A (da) | 1980-12-22 |
| SG14387G (en) | 1987-07-10 |
| AU538890B2 (en) | 1984-08-30 |
| CA1148159A (en) | 1983-06-14 |
| NO801866L (no) | 1980-12-22 |
| IE49993B1 (en) | 1986-01-22 |
| IL60357A (en) | 1984-05-31 |
| PT71420A (en) | 1980-07-01 |
| KR830002763A (ko) | 1983-05-30 |
| IL60357A0 (en) | 1980-09-16 |
| EP0022078B1 (de) | 1984-07-25 |
| KR840000421B1 (ko) | 1984-04-02 |
| HK47387A (en) | 1987-06-26 |
| MY8700556A (en) | 1987-12-31 |
| FI68827B (fi) | 1985-07-31 |
| DD151754A5 (de) | 1981-11-04 |
| JPS5618980A (en) | 1981-02-23 |
| CY1357A (en) | 1987-08-07 |
| GR69282B (da) | 1982-05-13 |
| DK160762C (da) | 1991-09-23 |
| DK160762B (da) | 1991-04-15 |
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