NO150082C - Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme benzimidazol-2-derivater - Google Patents

Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme benzimidazol-2-derivater

Info

Publication number
NO150082C
NO150082C NO782615A NO782615A NO150082C NO 150082 C NO150082 C NO 150082C NO 782615 A NO782615 A NO 782615A NO 782615 A NO782615 A NO 782615A NO 150082 C NO150082 C NO 150082C
Authority
NO
Norway
Prior art keywords
derivatives
preparation
therapeutically effective
new therapeutically
analogy procedure
Prior art date
Application number
NO782615A
Other languages
English (en)
Norwegian (no)
Other versions
NO782615L (no
NO150082B (no
Inventor
Ernst Habicht
Pier Giorgio Ferrini
Alfred Sallmann
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from HU77CI1761A external-priority patent/HU180700B/hu
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of NO782615L publication Critical patent/NO782615L/no
Publication of NO150082B publication Critical patent/NO150082B/no
Publication of NO150082C publication Critical patent/NO150082C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/45Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46Friedel-Crafts reactions
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/12Radicals substituted by oxygen atoms
NO782615A 1977-08-01 1978-07-31 Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme benzimidazol-2-derivater NO150082C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU77CI1761A HU180700B (en) 1976-08-27 1977-08-01 Process for producing acylized benzimidasole derivatives
CH209478 1978-02-27

Publications (3)

Publication Number Publication Date
NO782615L NO782615L (no) 1979-02-02
NO150082B NO150082B (no) 1984-05-07
NO150082C true NO150082C (no) 1984-08-15

Family

ID=25689497

Family Applications (1)

Application Number Title Priority Date Filing Date
NO782615A NO150082C (no) 1977-08-01 1978-07-31 Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme benzimidazol-2-derivater

Country Status (19)

Country Link
US (1) US4323688A (es)
EP (1) EP0000574B1 (es)
JP (1) JPS5427565A (es)
AR (4) AR227125A1 (es)
AT (1) AT364830B (es)
AU (1) AU523324B2 (es)
CA (1) CA1109072A (es)
DD (1) DD138318A5 (es)
DE (1) DE2861987D1 (es)
DK (1) DK339578A (es)
ES (1) ES472208A1 (es)
FI (1) FI68231C (es)
GR (1) GR77614B (es)
IE (1) IE47285B1 (es)
IL (1) IL55253A (es)
NO (1) NO150082C (es)
NZ (1) NZ188006A (es)
PL (1) PL208772A1 (es)
PT (1) PT68365A (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2861987D1 (en) * 1977-08-01 1982-09-30 Ciba Geigy Ag Benzimidazole-2 derivatives, their preparation and their use for the preparation of medicaments
US4322431A (en) * 1979-02-09 1982-03-30 Ciba-Geigy Corporation Pharmaceutical preparations containing benzimidazole 2-derivatives
US4368201A (en) * 1981-07-20 1983-01-11 Usv Pharmaceutical Corporation Tetrahydronaphthoxazoles

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB243766A (en) * 1924-12-01 1926-07-29 Bayer Ag Process for the manufacture of benzimidazoles
US2053822A (en) * 1933-12-15 1936-09-08 Soc Of Chemical Ind Alkylated imidazoles of high molecular weight and process of making same
GB766749A (en) 1954-01-11 1957-01-23 Aschaffenburger Zellstoffwerke Benzimidazole cobalamines and process for their preparation and separation
US2876233A (en) * 1956-10-29 1959-03-03 Gruenenthal Chemie 1-(p-halobenzyl)-2-methyl benzimidazoles and salts
CH356460A (de) * 1956-10-30 1961-08-31 Gruenenthal Chemie Verfahren zur Herstellung von neuen Derivaten des Benzimidazols
CH356461A (de) * 1956-10-30 1961-08-31 Gruenenthal Chemie Verfahren zur Herstellung von neuen Derivaten des Benzimidazols
CH362411A (de) * 1956-10-30 1962-06-15 Gruenenthal Chemie Verfahren zur Herstellung von neuen Derivaten des Benzimidazols
US3325271A (en) * 1963-07-17 1967-06-13 United States Borax Chem Herbicidal composition and method employing substituted benzimidazoles
US3318889A (en) * 1963-10-14 1967-05-09 S B Penick & Company 2-benzimidazole carbamates
DE2014293A1 (de) * 1969-03-29 1970-10-08 Fisons Ltd., Felixstowe, Suffolk (Grossbritannien) Substituierte Benzimidazole und Verfahren zu ihrer Herstellung und Verwendung
CH528514A (de) * 1969-05-22 1972-09-30 Bayer Ag Verfahren zur Herstellung von Acylimidazolen
US3661925A (en) * 1970-05-15 1972-05-09 American Home Prod Process for the preparation of 2-benzimidazolecarboxamides
FR2115067B1 (es) * 1970-11-27 1974-03-22 Delalande Sa
DE2861987D1 (en) * 1977-08-01 1982-09-30 Ciba Geigy Ag Benzimidazole-2 derivatives, their preparation and their use for the preparation of medicaments

Also Published As

Publication number Publication date
AU3847878A (en) 1980-02-07
AR227125A1 (es) 1982-09-30
IE781545L (en) 1979-02-01
DD138318A5 (de) 1979-10-24
AU523324B2 (en) 1982-07-22
IL55253A (en) 1982-04-30
ES472208A1 (es) 1979-03-16
GR77614B (es) 1984-09-25
ATA553978A (de) 1981-04-15
US4323688A (en) 1982-04-06
DE2861987D1 (en) 1982-09-30
EP0000574B1 (de) 1982-08-04
IL55253A0 (en) 1978-09-29
NO782615L (no) 1979-02-02
NZ188006A (en) 1981-11-19
AR231636A1 (es) 1985-01-31
FI68231B (fi) 1985-04-30
CA1109072A (en) 1981-09-15
IE47285B1 (en) 1984-02-08
NO150082B (no) 1984-05-07
AT364830B (de) 1981-11-25
FI68231C (fi) 1985-08-12
JPS5427565A (en) 1979-03-01
DK339578A (da) 1979-02-02
PL208772A1 (pl) 1979-06-04
AR228023A1 (es) 1983-01-14
FI782348A (fi) 1979-02-02
EP0000574A1 (de) 1979-02-07
PT68365A (de) 1978-08-01
AR223196A1 (es) 1981-07-31

Similar Documents

Publication Publication Date Title
NO160211C (no) Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme cefemderivater.
NO149174C (no) Analogifremgangsmaate ved fremstilling av nye terapeutisk virksomme tiazinderivater
NO147148C (no) Analogifremgangsmaate ved fremstilling av nye terapeutisk aktive fenyletanolaminderivater
NO145881C (no) Analogifremgangsmaate for fremstilling av nye terapeutisk virksomme acetohydroksamsyrer
NO148290C (no) Analogifremgangsmaate ved fremstilling av nye terapeutisk aktive polyenforbindelser
NO156611C (no) Analogifremgangsmaate for fremstilling av terapeutiske virksomme derivater av hydroksykarbonylfosfonsyre.
NO148813C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive karbostyrilderivater
NO147025C (no) Analogifremgangsmaate for fremstilling av terapeutisk virksomme pyridinyl-2(1h)-pyridinoner
NO148148C (no) Fremgangsmaate til fremstilling av terapeutisk aktive 4-hydroksy-2-pyrrolidinonderivater
SE431088B (sv) Forfarande for framstellning av terapeutiskt verksamma benshydrylsulfinylderivat
NO152651C (no) Analogifremgangsmaate for fremstilling av terapeutisk virksomme 0-substituerte derivater av (+)-cyanidan-3-ol
NO147562C (no) Analogifremgangsmaate for fremstilling av terapeutisk virksomme xantinderivater
NO145307C (no) Analogifremgangsmaate ved fremstilling av nye terapeutisk virksomme nucleosider
NO144848C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme 4-hydroksyfenylalkanolamin-derivater
NO148777C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive antrakinon-derivater
NO143796C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme piperazinyliminorifamyciner
NO148642C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive, nye prostacyclinderivater
NO152654C (no) Analogifremgangsmaate ved fremstilling av nye, terapeutisk aktive derivater av 7-acylamido-3-cephem-4-karboksylsyre
NO150081C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme derivater av perhydro-aza-heterocykler
NO149313C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive pyridobenzodiazepiner
NO146022C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme benzofenonderivater
NO149037C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive pyridobenzodiazepiner
NO150279C (no) Analogifremgangsmaate til fremstilling av nye terapeutisk virksomme benzopyranderivater
SE7803035L (sv) Forfarande for framstellning av tienopyridinderivat
NO148454C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive tiazolidin-dionderivater