NL8005890A - 4,4 digesubstitueerde piperidinobutyrofenonen en zouten daarvan. - Google Patents
4,4 digesubstitueerde piperidinobutyrofenonen en zouten daarvan. Download PDFInfo
- Publication number
- NL8005890A NL8005890A NL8005890A NL8005890A NL8005890A NL 8005890 A NL8005890 A NL 8005890A NL 8005890 A NL8005890 A NL 8005890A NL 8005890 A NL8005890 A NL 8005890A NL 8005890 A NL8005890 A NL 8005890A
- Authority
- NL
- Netherlands
- Prior art keywords
- compound
- formula
- group
- cyano
- salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8894279A | 1979-10-27 | 1979-10-27 | |
US8894279 | 1979-10-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
NL8005890A true NL8005890A (nl) | 1981-04-29 |
Family
ID=22214421
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL8005890A NL8005890A (nl) | 1979-10-27 | 1980-10-27 | 4,4 digesubstitueerde piperidinobutyrofenonen en zouten daarvan. |
Country Status (12)
Country | Link |
---|---|
JP (1) | JPS5673061A (ja) |
AU (1) | AU6369480A (ja) |
BE (1) | BE885894A (ja) |
CA (1) | CA1148162A (ja) |
DE (1) | DE3039974A1 (ja) |
ES (1) | ES8201550A1 (ja) |
FR (1) | FR2468592A1 (ja) |
GB (1) | GB2061937A (ja) |
IL (1) | IL61340A0 (ja) |
IT (1) | IT1146198B (ja) |
NL (1) | NL8005890A (ja) |
ZA (1) | ZA806501B (ja) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ577114A (en) * | 2006-12-19 | 2011-12-22 | Hoffmann La Roche | Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE713746C (de) * | 1939-03-31 | 1941-11-18 | I G Farbenindustrie Akt Ges | Verfahren zur Darstellung von 4-Arylpiperidyl-4-ketonen |
US3080372A (en) * | 1960-03-25 | 1963-03-05 | Res Lab Dr C Janssen | 1-aroylalkyl-4-arylpiperidine derivatives |
CH492708A (de) * | 1968-01-11 | 1970-06-30 | Geigy Ag J R | Verfahren zur Herstellung von neuen Piperidinderivaten |
CH498836A (de) * | 1968-12-20 | 1970-11-15 | Geigy Ag J R | Verfahren zur Herstellung von neuen Piperidinderivaten |
US3852455A (en) * | 1970-11-27 | 1974-12-03 | Richardson Merrell Inc | 4-{8 4({60 hydroxybenzyl)piperidino{9 -4-fluorobutyrophenone derivatives as tranquilizers |
ZA717147B (en) * | 1970-11-27 | 1972-07-26 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)-4'-fluorobutyrophenone derivatives |
US3888867A (en) * | 1972-05-03 | 1975-06-10 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)4'-fluorobutyrophenone derivatives |
US4101662A (en) * | 1973-05-03 | 1978-07-18 | A. H. Robins Company, Incorporated | Method for inhibiting emesis and compositions therefor |
SE7409245L (ja) * | 1973-07-19 | 1975-01-20 | Robins Co Inc A H | |
GB1535791A (en) * | 1975-05-07 | 1978-12-13 | Ferrosan Ab | Derivatives of 4-piperidinol |
CH602642A5 (ja) * | 1975-11-14 | 1978-07-31 | Orgamol Sa | |
US4335127A (en) * | 1979-01-08 | 1982-06-15 | Janssen Pharmaceutica, N.V. | Piperidinylalkyl quinazoline compounds, composition and method of use |
-
1980
- 1980-10-22 ZA ZA00806501A patent/ZA806501B/xx unknown
- 1980-10-23 ES ES496204A patent/ES8201550A1/es not_active Expired
- 1980-10-23 DE DE19803039974 patent/DE3039974A1/de not_active Withdrawn
- 1980-10-24 GB GB8034418A patent/GB2061937A/en not_active Withdrawn
- 1980-10-24 IT IT49998/80A patent/IT1146198B/it active
- 1980-10-24 CA CA000363264A patent/CA1148162A/en not_active Expired
- 1980-10-24 AU AU63694/80A patent/AU6369480A/en not_active Abandoned
- 1980-10-24 IL IL61340A patent/IL61340A0/xx unknown
- 1980-10-24 FR FR8022862A patent/FR2468592A1/fr active Granted
- 1980-10-27 NL NL8005890A patent/NL8005890A/nl not_active Application Discontinuation
- 1980-10-27 JP JP14952780A patent/JPS5673061A/ja active Pending
- 1980-10-27 BE BE0/202608A patent/BE885894A/fr not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
BE885894A (fr) | 1981-02-16 |
IL61340A0 (en) | 1980-12-31 |
FR2468592A1 (fr) | 1981-05-08 |
ES496204A0 (es) | 1981-12-01 |
JPS5673061A (en) | 1981-06-17 |
DE3039974A1 (de) | 1981-05-07 |
ES8201550A1 (es) | 1981-12-01 |
FR2468592B1 (ja) | 1983-08-05 |
AU6369480A (en) | 1981-04-30 |
IT1146198B (it) | 1986-11-12 |
CA1148162A (en) | 1983-06-14 |
ZA806501B (en) | 1981-10-28 |
GB2061937A (en) | 1981-05-20 |
IT8049998A0 (it) | 1980-10-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
A85 | Still pending on 85-01-01 | ||
BA | A request for search or an international-type search has been filed | ||
BB | A search report has been drawn up | ||
BC | A request for examination has been filed | ||
BV | The patent application has lapsed |