JPS5673061A - 44*44alkyll44aroyll11piperidino*butyrophenone antipsychotic - Google Patents
44*44alkyll44aroyll11piperidino*butyrophenone antipsychoticInfo
- Publication number
- JPS5673061A JPS5673061A JP14952780A JP14952780A JPS5673061A JP S5673061 A JPS5673061 A JP S5673061A JP 14952780 A JP14952780 A JP 14952780A JP 14952780 A JP14952780 A JP 14952780A JP S5673061 A JPS5673061 A JP S5673061A
- Authority
- JP
- Japan
- Prior art keywords
- butyrophenone
- antipsychotic
- butyrophenone antipsychotic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8894279A | 1979-10-27 | 1979-10-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS5673061A true JPS5673061A (en) | 1981-06-17 |
Family
ID=22214421
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP14952780A Pending JPS5673061A (en) | 1979-10-27 | 1980-10-27 | 44*44alkyll44aroyll11piperidino*butyrophenone antipsychotic |
Country Status (12)
| Country | Link |
|---|---|
| JP (1) | JPS5673061A (en) |
| AU (1) | AU6369480A (en) |
| BE (1) | BE885894A (en) |
| CA (1) | CA1148162A (en) |
| DE (1) | DE3039974A1 (en) |
| ES (1) | ES496204A0 (en) |
| FR (1) | FR2468592A1 (en) |
| GB (1) | GB2061937A (en) |
| IL (1) | IL61340A0 (en) |
| IT (1) | IT1146198B (en) |
| NL (1) | NL8005890A (en) |
| ZA (1) | ZA806501B (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2009006334A (en) | 2006-12-19 | 2009-06-23 | Hoffmann La Roche | Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives. |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3852455A (en) * | 1970-11-27 | 1974-12-03 | Richardson Merrell Inc | 4-{8 4({60 hydroxybenzyl)piperidino{9 -4-fluorobutyrophenone derivatives as tranquilizers |
| US3888867A (en) * | 1972-05-03 | 1975-06-10 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)4'-fluorobutyrophenone derivatives |
| US4101662A (en) * | 1973-05-03 | 1978-07-18 | A. H. Robins Company, Incorporated | Method for inhibiting emesis and compositions therefor |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE713746C (en) * | 1939-03-31 | 1941-11-18 | I G Farbenindustrie Akt Ges | Process for the preparation of 4-arylpiperidyl-4-ketones |
| US3080372A (en) * | 1960-03-25 | 1963-03-05 | Res Lab Dr C Janssen | 1-aroylalkyl-4-arylpiperidine derivatives |
| CH492709A (en) * | 1968-01-11 | 1970-06-30 | Geigy Ag J R | Process for the preparation of new piperidine derivatives |
| CH498836A (en) * | 1968-12-20 | 1970-11-15 | Geigy Ag J R | Pharmaceutical piperidine derivs prodn |
| ZA717147B (en) * | 1970-11-27 | 1972-07-26 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)-4'-fluorobutyrophenone derivatives |
| SE7409245L (en) * | 1973-07-19 | 1975-01-20 | Robins Co Inc A H | |
| GB1535791A (en) * | 1975-05-07 | 1978-12-13 | Ferrosan Ab | Derivatives of 4-piperidinol |
| CH602642A5 (en) * | 1975-11-14 | 1978-07-31 | Orgamol Sa | |
| US4335127A (en) * | 1979-01-08 | 1982-06-15 | Janssen Pharmaceutica, N.V. | Piperidinylalkyl quinazoline compounds, composition and method of use |
-
1980
- 1980-10-22 ZA ZA00806501A patent/ZA806501B/en unknown
- 1980-10-23 ES ES496204A patent/ES496204A0/en active Granted
- 1980-10-23 DE DE19803039974 patent/DE3039974A1/en not_active Withdrawn
- 1980-10-24 AU AU63694/80A patent/AU6369480A/en not_active Abandoned
- 1980-10-24 FR FR8022862A patent/FR2468592A1/en active Granted
- 1980-10-24 GB GB8034418A patent/GB2061937A/en not_active Withdrawn
- 1980-10-24 IT IT49998/80A patent/IT1146198B/en active
- 1980-10-24 CA CA000363264A patent/CA1148162A/en not_active Expired
- 1980-10-24 IL IL61340A patent/IL61340A0/en unknown
- 1980-10-27 JP JP14952780A patent/JPS5673061A/en active Pending
- 1980-10-27 BE BE0/202608A patent/BE885894A/en not_active IP Right Cessation
- 1980-10-27 NL NL8005890A patent/NL8005890A/en not_active Application Discontinuation
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3852455A (en) * | 1970-11-27 | 1974-12-03 | Richardson Merrell Inc | 4-{8 4({60 hydroxybenzyl)piperidino{9 -4-fluorobutyrophenone derivatives as tranquilizers |
| US3888867A (en) * | 1972-05-03 | 1975-06-10 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)4'-fluorobutyrophenone derivatives |
| US4101662A (en) * | 1973-05-03 | 1978-07-18 | A. H. Robins Company, Incorporated | Method for inhibiting emesis and compositions therefor |
Also Published As
| Publication number | Publication date |
|---|---|
| IT8049998A0 (en) | 1980-10-24 |
| DE3039974A1 (en) | 1981-05-07 |
| AU6369480A (en) | 1981-04-30 |
| IL61340A0 (en) | 1980-12-31 |
| ES8201550A1 (en) | 1981-12-01 |
| BE885894A (en) | 1981-02-16 |
| CA1148162A (en) | 1983-06-14 |
| IT1146198B (en) | 1986-11-12 |
| ES496204A0 (en) | 1981-12-01 |
| GB2061937A (en) | 1981-05-20 |
| FR2468592B1 (en) | 1983-08-05 |
| NL8005890A (en) | 1981-04-29 |
| FR2468592A1 (en) | 1981-05-08 |
| ZA806501B (en) | 1981-10-28 |
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