BE885894A - (ALKYL-4 AROYL-4 PIPERIDINO) -4 BUTYROPHENONES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND THERAPEUTIC COMPOSITIONS CONTAINING THEM - Google Patents

(ALKYL-4 AROYL-4 PIPERIDINO) -4 BUTYROPHENONES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND THERAPEUTIC COMPOSITIONS CONTAINING THEM

Info

Publication number
BE885894A
BE885894A BE0/202608A BE202608A BE885894A BE 885894 A BE885894 A BE 885894A BE 0/202608 A BE0/202608 A BE 0/202608A BE 202608 A BE202608 A BE 202608A BE 885894 A BE885894 A BE 885894A
Authority
BE
Belgium
Prior art keywords
butyrophenones
aroyl
piperidino
intermediates
alkyl
Prior art date
Application number
BE0/202608A
Other languages
French (fr)
Inventor
A Carr
R Farr
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of BE885894A publication Critical patent/BE885894A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/30Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
    • C07D211/32Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
BE0/202608A 1979-10-27 1980-10-27 (ALKYL-4 AROYL-4 PIPERIDINO) -4 BUTYROPHENONES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND THERAPEUTIC COMPOSITIONS CONTAINING THEM BE885894A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8894279A 1979-10-27 1979-10-27

Publications (1)

Publication Number Publication Date
BE885894A true BE885894A (en) 1981-02-16

Family

ID=22214421

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/202608A BE885894A (en) 1979-10-27 1980-10-27 (ALKYL-4 AROYL-4 PIPERIDINO) -4 BUTYROPHENONES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND THERAPEUTIC COMPOSITIONS CONTAINING THEM

Country Status (12)

Country Link
JP (1) JPS5673061A (en)
AU (1) AU6369480A (en)
BE (1) BE885894A (en)
CA (1) CA1148162A (en)
DE (1) DE3039974A1 (en)
ES (1) ES496204A0 (en)
FR (1) FR2468592A1 (en)
GB (1) GB2061937A (en)
IL (1) IL61340A0 (en)
IT (1) IT1146198B (en)
NL (1) NL8005890A (en)
ZA (1) ZA806501B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2354124T3 (en) * 2006-12-19 2013-07-31 Hoffmann La Roche Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE713746C (en) * 1939-03-31 1941-11-18 I G Farbenindustrie Akt Ges Process for the preparation of 4-arylpiperidyl-4-ketones
US3080372A (en) * 1960-03-25 1963-03-05 Res Lab Dr C Janssen 1-aroylalkyl-4-arylpiperidine derivatives
CH491917A (en) * 1968-01-11 1970-06-15 Geigy Ag J R Process for the preparation of new piperidine derivatives
CH498836A (en) * 1968-12-20 1970-11-15 Geigy Ag J R Pharmaceutical piperidine derivs prodn
US3852455A (en) * 1970-11-27 1974-12-03 Richardson Merrell Inc 4-{8 4({60 hydroxybenzyl)piperidino{9 -4-fluorobutyrophenone derivatives as tranquilizers
ZA717147B (en) * 1970-11-27 1972-07-26 Richardson Merrell Inc 4-(4-(alpha-hydroxybenzyl)piperidino)-4'-fluorobutyrophenone derivatives
US3888867A (en) * 1972-05-03 1975-06-10 Richardson Merrell Inc 4-(4-(alpha-hydroxybenzyl)piperidino)4'-fluorobutyrophenone derivatives
US4101662A (en) * 1973-05-03 1978-07-18 A. H. Robins Company, Incorporated Method for inhibiting emesis and compositions therefor
SE7409245L (en) * 1973-07-19 1975-01-20 Robins Co Inc A H
GB1535791A (en) * 1975-05-07 1978-12-13 Ferrosan Ab Derivatives of 4-piperidinol
CH602642A5 (en) * 1975-11-14 1978-07-31 Orgamol Sa
US4335127A (en) * 1979-01-08 1982-06-15 Janssen Pharmaceutica, N.V. Piperidinylalkyl quinazoline compounds, composition and method of use

Also Published As

Publication number Publication date
AU6369480A (en) 1981-04-30
IT8049998A0 (en) 1980-10-24
GB2061937A (en) 1981-05-20
ES8201550A1 (en) 1981-12-01
NL8005890A (en) 1981-04-29
JPS5673061A (en) 1981-06-17
DE3039974A1 (en) 1981-05-07
ES496204A0 (en) 1981-12-01
IL61340A0 (en) 1980-12-31
IT1146198B (en) 1986-11-12
FR2468592A1 (en) 1981-05-08
FR2468592B1 (en) 1983-08-05
CA1148162A (en) 1983-06-14
ZA806501B (en) 1981-10-28

Similar Documents

Publication Publication Date Title
FR2479208B1 (en) 2-CYANACRYLATES, PROCESS FOR THEIR PREPARATION AND CURABLE COMPOSITIONS CONTAINING THESE ESTERS
IT8149086A0 (en) INDOLIC HETEROCYCLIC COMPOUNDS PROCEDURE FOR PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
IT8149407A0 (en) AMINOALKYLFURAN DERIVATIVE PROCEDURE FOR PRODUCING IT AND PHARMACEUTICAL COMPOSITION CONTAINING IT
IT1142469B (en) SYRINGE FOR INJECTIONS OF MEDICAMENTS
BE871095A (en) COMPOSITIONS OF BATS FOR SYNANTHROPIC FLIES
FI811745L (en) PHARMACEUTICAL COMPOSITION FOR THE FRAMEWORK OF FRUIT
FR2326920A1 (en) AZETIDINONE COMPOUNDS AND METHODS FOR THEIR PREPARATION
BE893378A (en) CARBOXIMIDE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENT CONTAINING THEM
BE879263A (en) 2-METHYL-DIHYDROPYRIDINE COMPOUND, METHODS FOR OBTAINING SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME
IT8049022A0 (en) DEVICE FOR THE APPLICATION OF CIGARETTE FILTERS
FI790922A (en) 2,6-DIALKOXIBENZAMIDER MELLANPRODUKTER PHARMACEUTICAL COMPOSITION OF FOERFARANDE FOR BEHANDLING AV PSYCHOTIC SJUKDOMAR
BE887730A (en) NOVEL HETEROCYCLIC DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
BE885507A (en) HETEROCYCLIC COMPOUNDS, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
BE870576A (en) NEW DIALKYLAMINO-7 HALOGENO-6 OXO-4-DIHYDRO-1,4-QUINOLEINE-3-CARBOXYLIC ACIDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM
BE871857A (en) NEW DISUBSTITLED PIPERAZINES, THEIR METHODS OF PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FI812190L (en) NYA PENTAPEPTIDER FOERFARANDEN FOER DERAS FRAMSTAELLNING PHARMACEUTICAL COMPOSITION INNEHAOLLANDE NAEMNDA PENTAPEPTIDER OCH DERAS ANVAENDNING
BE885894A (en) (ALKYL-4 AROYL-4 PIPERIDINO) -4 BUTYROPHENONES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND THERAPEUTIC COMPOSITIONS CONTAINING THEM
BE884101A (en) SULFUR-CONTAINING ISOQUINOLEIN DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM
IT8148607A0 (en) HAYMAKING MACHINE FOR FORMATION OF SWANDS AND SPREADING
IT1171278B (en) ANTI-BREATHING COMPOSITION APPLICATOR TUBE FOR CAPILLARITY ACTION
FR2528829B1 (en) POLYPRENYLIC COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC COMPOSITION CONTAINING THEM
RO79428A2 (en) DRUG COMPOSITION FOR THE TREATMENT OF DERMATOSES
BE882443A (en) QUINOLONES AND THERAPEUTIC COMPOSITIONS CONTAINING THEM
IT8148776A0 (en) HETEROCYCLIC COMPOUNDS THEIR PHARMACEUTICAL PREPARATION AND COMPOSITION CONTAINING THESE COMPOUNDS
BE863588A (en) NEW 2,5-DIHYDRO-1,2-THIAZINO (5,6-) 1,1-DIOXIDES INDOLE-3-CARBOXAMIDES, METHODS FOR THEIR PREPARATION AND MEDICINAL PRODUCTS CONTAINING THEM

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: RICHARDSON-MERRELL INC.

Effective date: 19931031