MXPA06010793A - Compuestos composiciones, procesos de elaboracion, y metodos de uso relacionados a la inhibicion del factor inhibidor de migracion de macrofago. - Google Patents
Compuestos composiciones, procesos de elaboracion, y metodos de uso relacionados a la inhibicion del factor inhibidor de migracion de macrofago.Info
- Publication number
- MXPA06010793A MXPA06010793A MXPA06010793A MXPA06010793A MXPA06010793A MX PA06010793 A MXPA06010793 A MX PA06010793A MX PA06010793 A MXPA06010793 A MX PA06010793A MX PA06010793 A MXPA06010793 A MX PA06010793A MX PA06010793 A MXPA06010793 A MX PA06010793A
- Authority
- MX
- Mexico
- Prior art keywords
- group
- alkyl
- phenyl
- cycloalkyl
- heteroaryl
- Prior art date
Links
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55644004P | 2004-03-26 | 2004-03-26 | |
| PCT/US2005/010444 WO2005094329A2 (en) | 2004-03-26 | 2005-03-28 | Compouns, compositions, processes of making, and methods of use related to inhibiting macrophage migration inhibitory factor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA06010793A true MXPA06010793A (es) | 2006-12-19 |
Family
ID=35064296
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA06010793A MXPA06010793A (es) | 2004-03-26 | 2005-03-28 | Compuestos composiciones, procesos de elaboracion, y metodos de uso relacionados a la inhibicion del factor inhibidor de migracion de macrofago. |
Country Status (9)
| Country | Link |
|---|---|
| US (3) | US20050250826A1 (enExample) |
| EP (1) | EP1727542A4 (enExample) |
| JP (1) | JP2007530598A (enExample) |
| CN (1) | CN101098697B (enExample) |
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| CA (1) | CA2557166C (enExample) |
| MX (1) | MXPA06010793A (enExample) |
| WO (1) | WO2005094329A2 (enExample) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102558082B (zh) | 2004-03-05 | 2015-09-30 | 日产化学工业株式会社 | 异噁唑啉取代苯甲酰胺化合物的制备中间体 |
| TW200803740A (en) | 2005-12-16 | 2008-01-16 | Du Pont | 5-aryl isoxazolines for controlling invertebrate pests |
| TWI412322B (zh) | 2005-12-30 | 2013-10-21 | Du Pont | 控制無脊椎害蟲之異唑啉 |
| AU2007230948B2 (en) * | 2006-03-24 | 2012-06-28 | The Feinstein Institute For Medical Research | Modified macrophage migration inhibitory factor inhibitors |
| JP5473906B2 (ja) | 2007-06-13 | 2014-04-16 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | イソキサゾリン殺虫剤 |
| TWI430995B (zh) | 2007-06-26 | 2014-03-21 | Du Pont | 萘異唑啉無脊椎有害動物控制劑 |
| CA2971008A1 (en) | 2007-06-27 | 2008-12-31 | E. I. Du Pont De Nemours And Company | Animal pest control method |
| TWI461411B (zh) | 2007-08-17 | 2014-11-21 | Du Pont | 製備５－鹵烷基－４，５－二氫異唑衍生物之方法 |
| WO2009045999A1 (en) | 2007-10-03 | 2009-04-09 | E. I. Du Pont De Nemours And Company | Naphthalene isoxazoline compounds for control of invertebrate pests |
| TWI455919B (zh) | 2008-04-09 | 2014-10-11 | Du Pont | 製備３－三氟甲基查耳酮（ｃｈａｌｃｏｎｅ）之方法 |
| WO2010017132A1 (en) * | 2008-08-04 | 2010-02-11 | Chdi, Inc. | Certain kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof |
| US9149465B2 (en) | 2009-05-18 | 2015-10-06 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| US8927551B2 (en) | 2009-05-18 | 2015-01-06 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| US8765735B2 (en) | 2009-05-18 | 2014-07-01 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| WO2011066482A2 (en) * | 2009-11-25 | 2011-06-03 | Cytokine Pharmasciences, Inc. | Chiral synthesis of isoxazolines, isoxazoline compounds, and uses thereof |
| WO2011091040A1 (en) * | 2010-01-19 | 2011-07-28 | Cytokine Pharmasciences, Inc. | Use of isoxazoline compounds and compositions in bladder cancer |
| PH12012502333A1 (en) | 2010-05-27 | 2015-02-04 | Corteva Agriscience Llc | Crystalline form of 4- [5 - [3 -chloro-5 - (trifluoromethyl) phenyl] -4, 5 - dihydro - 5 - (trifluoromethyl) -3 - isoxazolyl] -n- [2-0x0-2- [ ( 2, 2, 2 - trifluoroethyl) amino] ethyl] -1- naphthalenecarboxamide |
| US9238689B2 (en) | 2011-07-15 | 2016-01-19 | Morpho Sys AG | Antibodies that are cross-reactive for macrophage migration inhibitory factor (MIF) and D-dopachrome tautomerase (D-DT) |
| EA201490279A1 (ru) | 2011-08-30 | 2014-08-29 | Схди Фаундейшн, Инк. | Ингибиторы кинуренин-3-монооксигеназы, фармацевтические композиции и способы их применения |
| EP3243515B1 (en) | 2011-08-30 | 2019-10-16 | CHDI Foundation, Inc. | Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof |
| WO2013161933A1 (ja) * | 2012-04-26 | 2013-10-31 | 富山化学工業株式会社 | 重水素化含窒素複素環カルボキサミド誘導体 |
| US11234918B2 (en) | 2012-06-06 | 2022-02-01 | Basf Corporation | Methods for botanical and/or algae extraction |
| EP2944310B1 (en) | 2014-05-16 | 2018-03-21 | Mifcare | MIF inhibitors for the acute or chronic treatment of pulmonary hypertension |
| PE20170770A1 (es) | 2014-07-17 | 2017-07-04 | Chdi Foundation Inc | Metodos y composiciones para tratar trastornos relacionados con vih |
| US11397182B2 (en) | 2014-10-07 | 2022-07-26 | Cornell University | Methods for prognosing and preventing metastatic liver disease |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4933464A (en) * | 1988-04-25 | 1990-06-12 | W. R. Grace & Co.-Conn. | Process for forming 3-phenylisoxazolines and 3-phenylisoxazoles |
| JP2787602B2 (ja) * | 1990-01-24 | 1998-08-20 | 大鵬薬品工業株式会社 | イソキサゾリン誘導体 |
| JP2738486B2 (ja) * | 1992-11-20 | 1998-04-08 | ファイザー製薬株式会社 | 抗炎症剤としての新規なイソオキサゾリン類 |
| JPH0741459A (ja) * | 1993-07-29 | 1995-02-10 | Sumitomo Pharmaceut Co Ltd | 新規エラスターゼ阻害剤 |
| US5849736A (en) * | 1993-11-24 | 1998-12-15 | The Dupont Merck Pharmaceutical Company | Isoxazoline and isoxazole fibrinogen receptor antagonists |
| ES2139754T3 (es) * | 1993-11-26 | 2000-02-16 | Pfizer | 3-fenil-2-isoxazolinas como agentes antiinflamatorios. |
| EP0730588B1 (en) * | 1993-11-26 | 1997-07-02 | Pfizer Inc. | Isoxazoline compounds as antiinflammatory agents |
| ATE169009T1 (de) * | 1994-03-09 | 1998-08-15 | Pfizer | Isoxazoline verbindung zur hemmung tnf-freigabe |
| US6420188B1 (en) * | 1996-02-16 | 2002-07-16 | The Picower Institute For Medical Research | Screening assay for the identification of inhibitors for macrophage migration inhibitory factor |
| US6492428B1 (en) * | 2000-07-26 | 2002-12-10 | The Picower Institute For Medical Research | Compounds having MIF antagonist activity |
| FR2764889B1 (fr) * | 1997-06-20 | 2000-09-01 | Sod Conseils Rech Applic | Nouveaux derives du 2-(iminomethyl)amino-phenyle, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant |
| US6335445B1 (en) * | 1997-03-24 | 2002-01-01 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them |
| EP1228037A4 (en) * | 1999-10-29 | 2004-06-02 | Picower Inst Med Res | COMPOUNDS HAVING ANTIAGONIST ACTIVITY OF MIF |
| EP1411930B1 (en) * | 2001-06-08 | 2013-01-16 | Cytokine Pharmasciences, Inc. | Isoxazoline compounds having mif antagonist activity |
| US20050202010A1 (en) * | 2003-08-29 | 2005-09-15 | Giroir Brett P. | Method of treatment and bioassay involving macrophage migration inhibitory factor (MIF) as cardiac-derived myocardial depressant factor |
| WO2005058845A2 (en) * | 2003-12-19 | 2005-06-30 | Novo Nordisk A/S | Novel glucagon antagonists/inverse agonists |
-
2005
- 2005-03-28 WO PCT/US2005/010444 patent/WO2005094329A2/en not_active Ceased
- 2005-03-28 CN CN2005800098795A patent/CN101098697B/zh not_active Expired - Fee Related
- 2005-03-28 CA CA2557166A patent/CA2557166C/en not_active Expired - Fee Related
- 2005-03-28 EP EP05742932A patent/EP1727542A4/en not_active Withdrawn
- 2005-03-28 US US11/090,128 patent/US20050250826A1/en not_active Abandoned
- 2005-03-28 MX MXPA06010793A patent/MXPA06010793A/es active IP Right Grant
- 2005-03-28 JP JP2007505270A patent/JP2007530598A/ja active Pending
- 2005-03-28 AU AU2005228417A patent/AU2005228417A1/en not_active Abandoned
- 2005-03-28 BR BRPI0507818-0A patent/BRPI0507818A/pt not_active IP Right Cessation
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2007
- 2007-05-01 US US11/742,978 patent/US20080113997A1/en not_active Abandoned
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2012
- 2012-09-25 US US13/626,816 patent/US20130225586A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN101098697B (zh) | 2010-11-10 |
| WO2005094329A8 (en) | 2006-01-05 |
| CN101098697A (zh) | 2008-01-02 |
| WO2005094329A2 (en) | 2005-10-13 |
| AU2005228417A1 (en) | 2005-10-13 |
| CA2557166A1 (en) | 2005-10-13 |
| JP2007530598A (ja) | 2007-11-01 |
| US20080113997A1 (en) | 2008-05-15 |
| EP1727542A4 (en) | 2009-08-05 |
| US20050250826A1 (en) | 2005-11-10 |
| US20130225586A1 (en) | 2013-08-29 |
| EP1727542A2 (en) | 2006-12-06 |
| BRPI0507818A (pt) | 2007-07-10 |
| WO2005094329A3 (en) | 2007-02-08 |
| CA2557166C (en) | 2015-06-30 |
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