MXPA06003452A - Formulaciones de liberacion controlada que exhiben una velocidad de liberacion ascendente. - Google Patents
Formulaciones de liberacion controlada que exhiben una velocidad de liberacion ascendente.Info
- Publication number
- MXPA06003452A MXPA06003452A MXPA06003452A MXPA06003452A MXPA06003452A MX PA06003452 A MXPA06003452 A MX PA06003452A MX PA06003452 A MXPA06003452 A MX PA06003452A MX PA06003452 A MXPA06003452 A MX PA06003452A MX PA06003452 A MXPA06003452 A MX PA06003452A
- Authority
- MX
- Mexico
- Prior art keywords
- dosage form
- active agent
- pharmaceutically active
- drug
- sustained release
- Prior art date
Links
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- MIMJSJSRRDZIPW-UHFFFAOYSA-N tilmacoxib Chemical compound C=1C=C(S(N)(=O)=O)C(F)=CC=1C=1OC(C)=NC=1C1CCCCC1 MIMJSJSRRDZIPW-UHFFFAOYSA-N 0.000 description 1
- 229960004605 timolol Drugs 0.000 description 1
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- PHLBKPHSAVXXEF-UHFFFAOYSA-N trazodone Chemical compound ClC1=CC=CC(N2CCN(CCCN3C(N4C=CC=CC4=N3)=O)CC2)=C1 PHLBKPHSAVXXEF-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
Landscapes
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- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
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- Animal Behavior & Ethology (AREA)
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- Engineering & Computer Science (AREA)
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- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
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| US50619503P | 2003-09-26 | 2003-09-26 | |
| US57098104P | 2004-05-14 | 2004-05-14 | |
| PCT/US2004/031509 WO2005030182A1 (en) | 2003-09-26 | 2004-09-24 | Controlled release formulations exhibiting an ascending rate of release |
Publications (1)
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| MXPA06003452A true MXPA06003452A (es) | 2006-08-31 |
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| MXPA06003452A MXPA06003452A (es) | 2003-09-26 | 2004-09-24 | Formulaciones de liberacion controlada que exhiben una velocidad de liberacion ascendente. |
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| EP (1) | EP1677769A1 (enExample) |
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| NO (1) | NO20061863L (enExample) |
| NZ (1) | NZ546183A (enExample) |
| WO (1) | WO2005030182A1 (enExample) |
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| SI2218448T1 (sl) | 2002-12-13 | 2016-01-29 | Durect Corporation | Sistem za oralno dajanje zdravila, ki obsega tekoči nosilec materialov z visoko viskoznostjo |
| WO2005072079A2 (en) | 2003-09-26 | 2005-08-11 | Alza Coporation | Drug coating providing high drug loading and methods for providing the same |
| NZ546182A (en) * | 2003-09-26 | 2009-08-28 | Alza Corp | Controlled release formulations of opioid and nonopioid analgesics such as hydrocodone and acetaminophen |
| US7592326B2 (en) | 2004-03-15 | 2009-09-22 | Karaolis David K R | Method for stimulating the immune, inflammatory or neuroprotective response |
| US20050287214A1 (en) * | 2004-06-28 | 2005-12-29 | Ayer Atul D | Squeeze controlled oral dosage form |
| US8541026B2 (en) | 2004-09-24 | 2013-09-24 | Abbvie Inc. | Sustained release formulations of opioid and nonopioid analgesics |
| US20070042041A1 (en) * | 2005-08-17 | 2007-02-22 | Board Of Trustees Of The University Of Arkansas | Drug-surfactant complexes for sustained release |
| RU2433817C2 (ru) * | 2006-01-21 | 2011-11-20 | Эбботт Гмбх Унд Ко.Кг | Лекарственная форма и способ для доставки вызывающих зависимость лекарственных веществ |
| US9265732B2 (en) | 2006-03-06 | 2016-02-23 | Pozen Inc. | Dosage forms for administering combinations of drugs |
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| WO2009069151A2 (en) * | 2007-11-30 | 2009-06-04 | Matrix Laboratories Limited | Controlled release composition |
| AU2013202707C1 (en) * | 2007-12-06 | 2015-07-30 | Durect Corporation | Oral pharmaceutical dosage forms |
| CA2706658A1 (en) | 2007-12-06 | 2009-06-18 | Durect Corporation | Methods useful for the treatment of pain, arthritic conditions or inflammation associated with a chronic condition |
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| CN102026627B (zh) | 2008-03-11 | 2016-10-26 | 武田药品工业株式会社 | 口腔崩解固体制剂 |
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| CA2726917C (en) | 2008-06-04 | 2018-06-26 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders |
| WO2010009319A2 (en) | 2008-07-16 | 2010-01-21 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders |
| CA2731008A1 (en) * | 2008-07-18 | 2010-01-21 | Valeant Pharmaceuticals International | Modified release formulation and methods of use |
| US20100323016A1 (en) * | 2008-07-18 | 2010-12-23 | Biljana Nadjsombati | Modified release formulation and methods of use |
| US20100323015A1 (en) * | 2008-07-18 | 2010-12-23 | Biljana Nadjsombati | Modified release formulation and methods of use |
| US20100260844A1 (en) | 2008-11-03 | 2010-10-14 | Scicinski Jan J | Oral pharmaceutical dosage forms |
| CN101703488B (zh) * | 2008-12-16 | 2013-02-20 | 北京科信必成医药科技发展有限公司 | 具有润滑层结构的双层渗透泵控释片及其制备方法 |
| WO2010089132A1 (en) | 2009-02-06 | 2010-08-12 | Egalet A/S | Immediate release composition resistant to abuse by intake of alcohol |
| AU2010265213B2 (en) | 2009-06-24 | 2012-08-23 | Egalet Ltd. | Controlled release formulations |
| PL399450A1 (pl) * | 2009-08-31 | 2013-01-21 | Depomed, Inc | Utrzymujace sie w zoladku kompozycje farmaceutyczne do natychmiastowego i przedluzonego uwalniania acetaminofenu |
| US9198861B2 (en) | 2009-12-22 | 2015-12-01 | Mallinckrodt Llc | Methods of producing stabilized solid dosage pharmaceutical compositions containing morphinans |
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| US8597681B2 (en) | 2009-12-22 | 2013-12-03 | Mallinckrodt Llc | Methods of producing stabilized solid dosage pharmaceutical compositions containing morphinans |
| US20110150989A1 (en) * | 2009-12-22 | 2011-06-23 | Mallinkckrodt Inc. | Methods of Producing Stabilized Solid Dosage Pharmaceutical Compositions Containing Morphinans |
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| US8741885B1 (en) | 2011-05-17 | 2014-06-03 | Mallinckrodt Llc | Gastric retentive extended release pharmaceutical compositions |
| US9050335B1 (en) | 2011-05-17 | 2015-06-09 | Mallinckrodt Llc | Pharmaceutical compositions for extended release of oxycodone and acetaminophen resulting in a quick onset and prolonged period of analgesia |
| US8858963B1 (en) | 2011-05-17 | 2014-10-14 | Mallinckrodt Llc | Tamper resistant composition comprising hydrocodone and acetaminophen for rapid onset and extended duration of analgesia |
| PL395069A1 (pl) * | 2011-05-31 | 2012-12-03 | Warszawski Uniwersytet Medyczny | Przeciwbólowa kompozycja farmaceutyczna do podawania doustnego |
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-
2004
- 2004-09-24 CA CA2540059A patent/CA2540059C/en not_active Expired - Fee Related
- 2004-09-24 MX MXPA06003452A patent/MXPA06003452A/es active IP Right Grant
- 2004-09-24 US US10/949,687 patent/US20070259033A1/en not_active Abandoned
- 2004-09-24 WO PCT/US2004/031509 patent/WO2005030182A1/en not_active Ceased
- 2004-09-24 KR KR1020067008098A patent/KR101169614B1/ko not_active Expired - Fee Related
- 2004-09-24 JP JP2006528262A patent/JP2007506775A/ja active Pending
- 2004-09-24 NZ NZ546183A patent/NZ546183A/en not_active IP Right Cessation
- 2004-09-24 AU AU2004275835A patent/AU2004275835B2/en not_active Ceased
- 2004-09-24 EP EP04789047A patent/EP1677769A1/en not_active Withdrawn
-
2006
- 2006-03-26 IL IL174563A patent/IL174563A0/en unknown
- 2006-04-26 NO NO20061863A patent/NO20061863L/no not_active Application Discontinuation
-
2010
- 2010-06-22 US US12/820,436 patent/US20110159046A1/en not_active Abandoned
- 2010-11-23 US US12/953,247 patent/US20110129507A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1677769A1 (en) | 2006-07-12 |
| AU2004275835A1 (en) | 2005-04-07 |
| JP2007506775A (ja) | 2007-03-22 |
| CA2540059A1 (en) | 2005-04-07 |
| CA2540059C (en) | 2013-08-06 |
| IL174563A0 (en) | 2006-08-20 |
| US20070259033A1 (en) | 2007-11-08 |
| AU2004275835B2 (en) | 2011-06-23 |
| WO2005030182A1 (en) | 2005-04-07 |
| KR101169614B1 (ko) | 2012-08-03 |
| US20110159046A1 (en) | 2011-06-30 |
| KR20060120050A (ko) | 2006-11-24 |
| NO20061863L (no) | 2006-06-23 |
| NZ546183A (en) | 2011-04-29 |
| US20110129507A1 (en) | 2011-06-02 |
| HK1122728A1 (en) | 2009-05-29 |
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