MXPA05012110A - Procedimiento para sintetizar intermediarios inhibidores de beta-lactamasa. - Google Patents

Procedimiento para sintetizar intermediarios inhibidores de beta-lactamasa.

Info

Publication number
MXPA05012110A
MXPA05012110A MXPA05012110A MXPA05012110A MXPA05012110A MX PA05012110 A MXPA05012110 A MX PA05012110A MX PA05012110 A MXPA05012110 A MX PA05012110A MX PA05012110 A MXPA05012110 A MX PA05012110A MX PA05012110 A MXPA05012110 A MX PA05012110A
Authority
MX
Mexico
Prior art keywords
intermediates
lactamase inhibitor
synthesizing beta
beta
synthesizing
Prior art date
Application number
MXPA05012110A
Other languages
English (en)
Inventor
Anita Wai-Yin Chan
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of MXPA05012110A publication Critical patent/MXPA05012110A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Se proporciona un procedimiento para la preparacion de heteroaril carboxaldehidos biciclicos que tienen la formula estructural (I) (ver formula I) en donde X y Y se definen en la descripcion. Los heteroaril carboxaldehidos biciclicos son utiles como intermediarios en la preparacion de inhibidores de (-lactamasa.
MXPA05012110A 2003-05-16 2004-05-12 Procedimiento para sintetizar intermediarios inhibidores de beta-lactamasa. MXPA05012110A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47145803P 2003-05-16 2003-05-16
PCT/US2004/014834 WO2004104006A2 (en) 2003-05-16 2004-05-12 PROCESS FOR SYNTHESIZING β-LACTAMASE INHIBITOR IN INTERMEDIATES

Publications (1)

Publication Number Publication Date
MXPA05012110A true MXPA05012110A (es) 2006-02-08

Family

ID=33476847

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05012110A MXPA05012110A (es) 2003-05-16 2004-05-12 Procedimiento para sintetizar intermediarios inhibidores de beta-lactamasa.

Country Status (12)

Country Link
US (2) US7276611B2 (es)
EP (1) EP1626975A2 (es)
JP (1) JP2006528978A (es)
CN (1) CN1823074A (es)
AR (1) AR044341A1 (es)
AU (1) AU2004240925A1 (es)
BR (1) BRPI0410398A (es)
CA (1) CA2525504A1 (es)
CL (1) CL2004001038A1 (es)
MX (1) MXPA05012110A (es)
TW (1) TW200510430A (es)
WO (1) WO2004104006A2 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2002053566A1 (ja) * 2000-12-27 2004-05-13 住友製薬株式会社 新規なカルバペネム化合物
US7468364B2 (en) 2003-04-08 2008-12-23 Dainippon Sumitomo Pharma Co., Ltd. Carbapenem compounds
EP1626975A2 (en) * 2003-05-16 2006-02-22 Wyeth Holdings Corporation PROCESS FOR SYNTHESIZING ß-LACTAMASE INHIBITOR IN INTERMEDIATES
AU2004240924A1 (en) * 2003-05-16 2004-12-02 Wyeth Holdings Corporation Process for synthesizing beta-lactamase inhibitor intermediates
EP1660506A4 (en) * 2003-08-25 2009-02-25 Revaax Pharmaceuticals Llc ORAL NEUROTHERAPEUTIC CEFAZOLINE COMPOSITIONS
TW201245185A (en) 2011-04-01 2012-11-16 Lundbeck & Co As H New positive allosteric modulators of nicotinic acetylcholine receptor

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2118181B (en) 1982-04-08 1986-07-30 Erba Farmitalia Substituted penem derivatives and new process for their preparation
EP1626975A2 (en) * 2003-05-16 2006-02-22 Wyeth Holdings Corporation PROCESS FOR SYNTHESIZING ß-LACTAMASE INHIBITOR IN INTERMEDIATES
AU2004240924A1 (en) * 2003-05-16 2004-12-02 Wyeth Holdings Corporation Process for synthesizing beta-lactamase inhibitor intermediates

Also Published As

Publication number Publication date
BRPI0410398A (pt) 2006-07-04
AU2004240925A1 (en) 2004-12-02
US20040242874A1 (en) 2004-12-02
CL2004001038A1 (es) 2005-03-04
TW200510430A (en) 2005-03-16
WO2004104006A3 (en) 2005-01-27
WO2004104006A2 (en) 2004-12-02
US7276611B2 (en) 2007-10-02
US20080009634A1 (en) 2008-01-10
EP1626975A2 (en) 2006-02-22
CA2525504A1 (en) 2004-12-02
JP2006528978A (ja) 2006-12-28
CN1823074A (zh) 2006-08-23
AR044341A1 (es) 2005-09-07

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal