MXPA04007186A - Nuevos derivados de la piridazina, su utilizacion como medicamentos, composiciones farmaceuticas y su procedimiento de preparacion. - Google Patents
Nuevos derivados de la piridazina, su utilizacion como medicamentos, composiciones farmaceuticas y su procedimiento de preparacion.Info
- Publication number
- MXPA04007186A MXPA04007186A MXPA04007186A MXPA04007186A MXPA04007186A MX PA04007186 A MXPA04007186 A MX PA04007186A MX PA04007186 A MXPA04007186 A MX PA04007186A MX PA04007186 A MXPA04007186 A MX PA04007186A MX PA04007186 A MXPA04007186 A MX PA04007186A
- Authority
- MX
- Mexico
- Prior art keywords
- radical
- same
- medicaments
- producing
- pharmaceutical compositions
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000004892 pyridazines Chemical class 0.000 title 1
- 150000003254 radicals Chemical group 0.000 abstract 4
- -1 COOR Chemical group 0.000 abstract 3
- 102000004190 Enzymes Human genes 0.000 abstract 1
- 108090000790 Enzymes Proteins 0.000 abstract 1
- 102000035195 Peptidases Human genes 0.000 abstract 1
- 108091005804 Peptidases Proteins 0.000 abstract 1
- 108091000080 Phosphotransferase Proteins 0.000 abstract 1
- 239000004365 Protease Substances 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 150000005840 aryl radicals Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 230000002503 metabolic effect Effects 0.000 abstract 1
- 125000002950 monocyclic group Chemical group 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 102000020233 phosphotransferase Human genes 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/04—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Endocrinology (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Psychiatry (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0201632A FR2835835B1 (fr) | 2002-02-11 | 2002-02-11 | Nouveaux derives de la pyridazine, leur utilisation comme medicaments, compositions pharmaceutiques et leur procede de preparation |
| PCT/FR2003/000381 WO2003068140A2 (fr) | 2002-02-11 | 2003-02-07 | Derives de la pyridazine, leur utilisation comme medicaments, et leur procede de preparation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA04007186A true MXPA04007186A (es) | 2004-10-29 |
Family
ID=27620073
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA04007186A MXPA04007186A (es) | 2002-02-11 | 2003-02-07 | Nuevos derivados de la piridazina, su utilizacion como medicamentos, composiciones farmaceuticas y su procedimiento de preparacion. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7223758B2 (enExample) |
| EP (1) | EP1476434B1 (enExample) |
| JP (1) | JP4447324B2 (enExample) |
| AT (1) | ATE329907T1 (enExample) |
| AU (1) | AU2003222363A1 (enExample) |
| BR (1) | BR0307565A (enExample) |
| CA (1) | CA2475439A1 (enExample) |
| CY (1) | CY1107483T1 (enExample) |
| DE (1) | DE60306122T2 (enExample) |
| DK (1) | DK1476434T3 (enExample) |
| ES (1) | ES2266806T3 (enExample) |
| FR (1) | FR2835835B1 (enExample) |
| MX (1) | MXPA04007186A (enExample) |
| PT (1) | PT1476434E (enExample) |
| WO (1) | WO2003068140A2 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2839309B1 (fr) * | 2002-05-03 | 2004-07-23 | Aventis Pharma Sa | Nouveaux derives de l'acide hexahydro-pyridazine-3- carboxylique, chimiotheques les contenant, leur utilisation comme medicaments, compositions pharmaceutiques les contenant et leurs procedes de preparation |
| EP1851204A1 (en) * | 2005-02-23 | 2007-11-07 | SmithKline Beecham Corporation | Naphthalene derivatives as modulators of the glucocorticoid receptor |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE191713T1 (de) * | 1991-11-08 | 2000-04-15 | Sankyo Co | Piperazin derivate als collagenase inhibitoren |
-
2002
- 2002-02-11 FR FR0201632A patent/FR2835835B1/fr not_active Expired - Fee Related
-
2003
- 2003-02-07 ES ES03717380T patent/ES2266806T3/es not_active Expired - Lifetime
- 2003-02-07 DK DK03717380T patent/DK1476434T3/da active
- 2003-02-07 CA CA002475439A patent/CA2475439A1/fr not_active Abandoned
- 2003-02-07 EP EP03717380A patent/EP1476434B1/fr not_active Expired - Lifetime
- 2003-02-07 MX MXPA04007186A patent/MXPA04007186A/es unknown
- 2003-02-07 DE DE60306122T patent/DE60306122T2/de not_active Expired - Lifetime
- 2003-02-07 PT PT03717380T patent/PT1476434E/pt unknown
- 2003-02-07 AU AU2003222363A patent/AU2003222363A1/en not_active Abandoned
- 2003-02-07 WO PCT/FR2003/000381 patent/WO2003068140A2/fr not_active Ceased
- 2003-02-07 JP JP2003567325A patent/JP4447324B2/ja not_active Expired - Fee Related
- 2003-02-07 BR BR0307565-6A patent/BR0307565A/pt not_active IP Right Cessation
- 2003-02-07 AT AT03717380T patent/ATE329907T1/de active
-
2004
- 2004-08-11 US US10/916,175 patent/US7223758B2/en not_active Expired - Lifetime
-
2006
- 2006-09-07 CY CY20061101281T patent/CY1107483T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003068140A3 (fr) | 2004-04-08 |
| CY1107483T1 (el) | 2013-03-13 |
| EP1476434A2 (fr) | 2004-11-17 |
| AU2003222363A1 (en) | 2003-09-04 |
| CA2475439A1 (fr) | 2003-08-21 |
| DE60306122T2 (de) | 2007-06-06 |
| JP4447324B2 (ja) | 2010-04-07 |
| EP1476434B1 (fr) | 2006-06-14 |
| DE60306122D1 (de) | 2006-07-27 |
| US7223758B2 (en) | 2007-05-29 |
| US20050165017A1 (en) | 2005-07-28 |
| JP2005525334A (ja) | 2005-08-25 |
| WO2003068140A2 (fr) | 2003-08-21 |
| FR2835835A1 (fr) | 2003-08-15 |
| PT1476434E (pt) | 2006-10-31 |
| FR2835835B1 (fr) | 2004-04-16 |
| ATE329907T1 (de) | 2006-07-15 |
| BR0307565A (pt) | 2004-12-21 |
| ES2266806T3 (es) | 2007-03-01 |
| DK1476434T3 (da) | 2006-10-16 |
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