MX9701328A - Metodos de reduccion de la cicatrizacion en la curacion de heridas. - Google Patents

Metodos de reduccion de la cicatrizacion en la curacion de heridas.

Info

Publication number
MX9701328A
MX9701328A MX9701328A MX9701328A MX9701328A MX 9701328 A MX9701328 A MX 9701328A MX 9701328 A MX9701328 A MX 9701328A MX 9701328 A MX9701328 A MX 9701328A MX 9701328 A MX9701328 A MX 9701328A
Authority
MX
Mexico
Prior art keywords
methods
wound healing
reducing scarring
scarring
reducing
Prior art date
Application number
MX9701328A
Other languages
English (en)
Inventor
George Joseph Cullinan
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MX9701328A publication Critical patent/MX9701328A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4535Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Silicates, Zeolites, And Molecular Sieves (AREA)
  • Eye Examination Apparatus (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Un método de inhibicion de la cicatrizacion que comprende administrar a un ser humano en necesidad del mismo, una cantidad efectiva de un compuesto que tiene la formula (I) en donde R1 y R3 son independientemente hidrogeno, -CH3, (a) o (b), en donde Ar es fenilo opcionalmente sustituido; R2 se selecciona del grupo que consiste de pirrolidina, hexametilenimino y piperidino; o una sal de solvato farmaceuticamente aceptable del mismo.
MX9701328A 1994-08-22 1995-08-21 Metodos de reduccion de la cicatrizacion en la curacion de heridas. MX9701328A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/293,851 US5550151A (en) 1994-08-22 1994-08-22 Methods of reducing scarring in wound healing
PCT/US1995/010650 WO1996005826A1 (en) 1994-08-22 1995-08-21 Methods of reducing scarring in wound healing

Publications (1)

Publication Number Publication Date
MX9701328A true MX9701328A (es) 1997-05-31

Family

ID=23130857

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9701328A MX9701328A (es) 1994-08-22 1995-08-21 Metodos de reduccion de la cicatrizacion en la curacion de heridas.

Country Status (14)

Country Link
US (1) US5550151A (es)
EP (1) EP0772438B1 (es)
JP (1) JPH10504823A (es)
AT (1) ATE179890T1 (es)
AU (1) AU3411195A (es)
CA (1) CA2198011A1 (es)
DE (1) DE69509657T2 (es)
DK (1) DK0772438T3 (es)
ES (1) ES2131331T3 (es)
GR (1) GR3030255T3 (es)
IL (1) IL115023A0 (es)
MX (1) MX9701328A (es)
WO (1) WO1996005826A1 (es)
ZA (1) ZA956995B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4688046B2 (ja) * 2004-11-05 2011-05-25 株式会社ポーラファルマ 肥厚性瘢痕動物モデル

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133814A (en) * 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents
US4418068A (en) * 1981-04-03 1983-11-29 Eli Lilly And Company Antiestrogenic and antiandrugenic benzothiophenes
US4380635A (en) * 1981-04-03 1983-04-19 Eli Lilly And Company Synthesis of acylated benzothiophenes
US5075321A (en) * 1987-03-24 1991-12-24 University Of Pennsylvania Methods of treating diseases characterized by interactions of IgG-containing immune complexes with macrophage Fc receptors using antiestrogenic benzothiophenes
US5395842A (en) * 1988-10-31 1995-03-07 Endorecherche Inc. Anti-estrogenic compounds and compositions
JP3157882B2 (ja) * 1991-11-15 2001-04-16 帝国臓器製薬株式会社 新規なベンゾチオフエン誘導体

Also Published As

Publication number Publication date
JPH10504823A (ja) 1998-05-12
EP0772438B1 (en) 1999-05-12
IL115023A0 (en) 1995-12-08
GR3030255T3 (en) 1999-08-31
DE69509657T2 (de) 1999-09-30
AU3411195A (en) 1996-03-14
DK0772438T3 (da) 1999-11-01
EP0772438A1 (en) 1997-05-14
DE69509657D1 (de) 1999-06-17
CA2198011A1 (en) 1996-02-29
WO1996005826A1 (en) 1996-02-29
EP0772438A4 (en) 1997-09-03
ZA956995B (en) 1997-02-21
US5550151A (en) 1996-08-27
ATE179890T1 (de) 1999-05-15
ES2131331T3 (es) 1999-07-16

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