MX381977B - Moduladores del receptor de péptido 1 tipo glucagón. - Google Patents

Moduladores del receptor de péptido 1 tipo glucagón.

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Publication number
MX381977B
MX381977B MX2017007494A MX2017007494A MX381977B MX 381977 B MX381977 B MX 381977B MX 2017007494 A MX2017007494 A MX 2017007494A MX 2017007494 A MX2017007494 A MX 2017007494A MX 381977 B MX381977 B MX 381977B
Authority
MX
Mexico
Prior art keywords
sub
peptide
glucagon
glp
receptor modulators
Prior art date
Application number
MX2017007494A
Other languages
English (en)
Spanish (es)
Other versions
MX2017007494A (es
Inventor
Adam R Yeager
Andrew Novak
Daniel Glynn
Enugurthi Brahmachary
Esther Martinborough
Junko Tamiya
Liming Huang
Manisha Moorjani
Marcus F Boehm
Mark Mills
Michael Knaggs
Premji Meghani
Thomas Fowler
Original Assignee
Receptos Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Receptos Llc filed Critical Receptos Llc
Publication of MX2017007494A publication Critical patent/MX2017007494A/es
Publication of MX381977B publication Critical patent/MX381977B/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/402—1-aryl substituted, e.g. piretanide
    • A—HUMAN NECESSITIES
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Pyrrole Compounds (AREA)
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