MX340918B - Forma de cristal novedosa de compuesto de benzopirano triciclico y metodo de produccion de la misma. - Google Patents

Forma de cristal novedosa de compuesto de benzopirano triciclico y metodo de produccion de la misma.

Info

Publication number
MX340918B
MX340918B MX2011011329A MX2011011329A MX340918B MX 340918 B MX340918 B MX 340918B MX 2011011329 A MX2011011329 A MX 2011011329A MX 2011011329 A MX2011011329 A MX 2011011329A MX 340918 B MX340918 B MX 340918B
Authority
MX
Mexico
Prior art keywords
processes
crystal forms
producing same
novel crystal
benzopyran compound
Prior art date
Application number
MX2011011329A
Other languages
English (en)
Other versions
MX2011011329A (es
Inventor
Takada Yasutaka
Kamon Miyako
Kawahara Shiro
Umeda Yasuhiro
Original Assignee
Nissan Chemical Ind Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nissan Chemical Ind Ltd filed Critical Nissan Chemical Ind Ltd
Publication of MX2011011329A publication Critical patent/MX2011011329A/es
Publication of MX340918B publication Critical patent/MX340918B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/052—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4741—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having oxygen as a ring hetero atom, e.g. tubocuraran derivatives, noscapine, bicuculline
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/96—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings spiro-condensed with carbocyclic rings or ring systems

Abstract

Se describen formas de cristal de (3R, 4S)-7-hidroximetil-2,2,9-tr imetil-4-(fenetilamino)-3 4-dihidro-2H-pirano(2,3-g]quinolin-3-ol que es una excelente medicina, y un proceso para producir las formas de cristal. El método comprende cristalizar (3R, 4S)-7-hidroximetil-2,2,9-trimetil-4-(fenetilamino)-3,4-dihidro-2H -pirano[2,3-g]quinolin-3-ol a partir de un solvente de éster de ácido acético, un solvente de hidrocarburo alifático, un solvente de nitrilo, un solvente de hidrocarburo aromático, un solvente de cetona o un solvente de éter. Se obtienen las formas de cristal por los procesos.
MX2011011329A 2009-04-30 2010-04-30 Forma de cristal novedosa de compuesto de benzopirano triciclico y metodo de produccion de la misma. MX340918B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2009111281 2009-04-30
PCT/JP2010/057698 WO2010126138A1 (ja) 2009-04-30 2010-04-30 ３環性ベンゾピラン化合物の新規な結晶形態及びその製造方法

Publications (2)

Publication Number Publication Date
MX2011011329A MX2011011329A (es) 2011-11-18
MX340918B true MX340918B (es) 2016-07-20

Family

ID=43032280

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011011329A MX340918B (es) 2009-04-30 2010-04-30 Forma de cristal novedosa de compuesto de benzopirano triciclico y metodo de produccion de la misma.

Country Status (21)

Country Link
US (1) US9242992B2 (es)
EP (1) EP2426133B1 (es)
JP (1) JP5664870B2 (es)
KR (1) KR101703202B1 (es)
CN (1) CN102414213B (es)
AR (1) AR076524A1 (es)
AU (1) AU2010242339B2 (es)
BR (1) BRPI1007112A2 (es)
CA (1) CA2759073C (es)
ES (1) ES2562027T3 (es)
HK (1) HK1166501A1 (es)
IL (1) IL215930A (es)
MX (1) MX340918B (es)
NZ (1) NZ596060A (es)
PL (1) PL2426133T3 (es)
RU (1) RU2523279C2 (es)
SG (1) SG175377A1 (es)
TW (1) TWI480281B (es)
UA (1) UA105385C2 (es)
WO (1) WO2010126138A1 (es)
ZA (1) ZA201107662B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20220071951A1 (en) 2018-12-28 2022-03-10 Osaka University Therapeutic agent for inherited bradyarrhythmia
EP4173623A1 (en) * 2020-06-26 2023-05-03 Osaka University Therapeutic agent for drug-induced bradycardia and bradyarrhythmia

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446497A1 (de) * 1974-09-28 1976-04-08 Boehringer Sohn Ingelheim 4-oxo-4h-pyrano- eckige klammer auf 3,2-c eckige klammer zu -chinolin-2-carbonsaeuren und ihre salze
US5164509A (en) * 1990-11-26 1992-11-17 E. R. Squibb & Sons, Inc. Benzodiazolo analogs
GB9224169D0 (en) * 1992-11-18 1993-01-06 Lilly Industries Ltd Pharmaceutical compounds
US5919806A (en) * 1993-04-02 1999-07-06 Nissan Chemical Industries, Ltd. Medicines for cardiac insufficiency
EP0807629B1 (de) * 1996-05-15 2004-03-03 Aventis Pharma Deutschland GmbH Sulfonamid-substituierte Chromane, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
EP0918774B9 (en) * 1996-06-27 2002-04-10 Ligand Pharmaceuticals Incorporated Androgen receptor modulator compounds and methods
JP4840594B2 (ja) * 2004-03-23 2011-12-21 日産化学工業株式会社 抗不整脈薬としての３環性ベンゾピラン化合物

Also Published As

Publication number Publication date
AU2010242339B2 (en) 2015-10-01
TW201111387A (en) 2011-04-01
KR20120024655A (ko) 2012-03-14
JP5664870B2 (ja) 2015-02-04
PL2426133T3 (pl) 2016-04-29
EP2426133A1 (en) 2012-03-07
EP2426133A4 (en) 2013-01-09
CA2759073A1 (en) 2010-11-04
MX2011011329A (es) 2011-11-18
CN102414213B (zh) 2014-12-24
CA2759073C (en) 2017-03-14
ES2562027T3 (es) 2016-03-02
SG175377A1 (en) 2011-12-29
HK1166501A1 (zh) 2012-11-02
RU2523279C2 (ru) 2014-07-20
IL215930A (en) 2016-09-29
UA105385C2 (uk) 2014-05-12
NZ596060A (en) 2012-12-21
US20120059169A1 (en) 2012-03-08
TWI480281B (zh) 2015-04-11
IL215930A0 (en) 2011-12-29
US9242992B2 (en) 2016-01-26
EP2426133B1 (en) 2015-12-16
BRPI1007112A2 (pt) 2015-08-18
CN102414213A (zh) 2012-04-11
AR076524A1 (es) 2011-06-15
RU2011148595A (ru) 2013-06-10
ZA201107662B (en) 2012-12-27
KR101703202B1 (ko) 2017-02-06
JPWO2010126138A1 (ja) 2012-11-01
WO2010126138A1 (ja) 2010-11-04
AU2010242339A1 (en) 2011-11-17

Similar Documents

Publication Publication Date Title
BR112012019413A2 (pt) processo para producao de uma corrente de alimentacao de ester para producao de esteres e coproducao de etanol
MX2012013922A (es) Procedimientos de baja energia para la recuperacion de alcohol.
EP3187589A3 (en) Baculovirus-based production of biopharmaceuticals free of contaminating baculoviral virions
WO2010122578A3 (en) Process for preparation of sitagliptin and its intermediates
NZ603268A (en) Process for synthesizing oxidized lactam compounds
WO2012038975A3 (en) Processes for the preparation of asenapine and intermediates thereof
WO2009116729A3 (en) Method for refining of high purity of tacrolimus
WO2012034648A9 (de) Spritzenkörper-kanülen-verbund und verfahren zu dessen herstellung
WO2007134846A3 (en) Process for purification of anastrozole
WO2011087316A3 (ko) 테트라졸 메탄설폰산 염의 제조방법 및 이에 사용되는 신규 화합물
TW200710076A (en) Process for producing aldehyde with 2-position branched long-chain alkyl
WO2011091131A3 (en) Eslicarbazepine acetate and its polymorphs
WO2008045185A3 (en) Process for the preparation of long-chain retinyl esters from short-chain retinyl esters and long-chain acids or long-chain esters employing lipases in organic solvents
MX340918B (es) Forma de cristal novedosa de compuesto de benzopirano triciclico y metodo de produccion de la misma.
WO2008000957A3 (fr) Procédé de préparation d'hydroquinone purifiée
WO2010004578A3 (en) Novel and improved processes for the preparation of paliperidone
WO2009124906A3 (en) A polymorph of argatroban monohydrate and a process for its synthesis
WO2013006099A3 (ru) 2,6-диизоборнилфенолы
EP2450337A3 (en) Process for making neo-enriched p-menthane compounds
BR112014000848A2 (pt) processo de separação
TW200616992A (en) Enantioselective separation method
WO2007143014A3 (en) Methods for preparing glutamic acid derivatives and intermediates thereof
WO2011097197A3 (en) Process for producing an ethyl acetate solvent and co-production of ethanol
WO2010064785A3 (en) Method for selectively crystallizing a z isomer of iopromide
WO2011045648A3 (en) Process for preparing (s)-(-)-10-acetoxy-10,11-dihydro-5h-dibenz[b,f]azepine-5-carboxamide and its esters thereof

Legal Events

Date Code Title Description
FG Grant or registration