MX2021002474A - Administracion prolongada de lasmiditan por la noche para la prevencion de la migra?a. - Google Patents

Administracion prolongada de lasmiditan por la noche para la prevencion de la migra?a.

Info

Publication number
MX2021002474A
MX2021002474A MX2021002474A MX2021002474A MX2021002474A MX 2021002474 A MX2021002474 A MX 2021002474A MX 2021002474 A MX2021002474 A MX 2021002474A MX 2021002474 A MX2021002474 A MX 2021002474A MX 2021002474 A MX2021002474 A MX 2021002474A
Authority
MX
Mexico
Prior art keywords
lasmiditan
migraine
prevention
chronic nightly
migraine prevention
Prior art date
Application number
MX2021002474A
Other languages
English (en)
Inventor
Kirk Willis Johnson
Robert Russell Conley
Gudarz Davar
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MX2021002474A publication Critical patent/MX2021002474A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Saccharide Compounds (AREA)

Abstract

La presente invención se refiere al uso prolongado de lasmiditan por la noche para la prevención de la migraña, particularmente la migraña resistente al tratamiento que se define en el presente documento como migraña refractaria a dos o más esquemas de prevención o tratamiento previos de monoterapia y/o terapia doble.
MX2021002474A 2018-09-04 2019-09-03 Administracion prolongada de lasmiditan por la noche para la prevencion de la migra?a. MX2021002474A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862726585P 2018-09-04 2018-09-04
PCT/US2019/049340 WO2020051137A1 (en) 2018-09-04 2019-09-03 Chronic nightly dosing of lasmiditan for migraine prevention

Publications (1)

Publication Number Publication Date
MX2021002474A true MX2021002474A (es) 2021-08-24

Family

ID=68051892

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021002474A MX2021002474A (es) 2018-09-04 2019-09-03 Administracion prolongada de lasmiditan por la noche para la prevencion de la migra?a.

Country Status (35)

Country Link
US (1) US20210338655A1 (es)
EP (2) EP3846810B1 (es)
JP (2) JP7321256B2 (es)
KR (1) KR102649644B1 (es)
CN (1) CN112638383A (es)
AU (2) AU2019336667B2 (es)
BR (1) BR112021002945A2 (es)
CA (1) CA3111205A1 (es)
CL (1) CL2021000529A1 (es)
CO (1) CO2021002766A2 (es)
CR (1) CR20210126A (es)
DK (1) DK3846810T3 (es)
DO (1) DOP2021000039A (es)
EA (1) EA202190440A1 (es)
EC (1) ECSP21015491A (es)
ES (1) ES2967665T3 (es)
FI (1) FI3846810T3 (es)
HR (1) HRP20231587T1 (es)
HU (1) HUE064519T2 (es)
IL (1) IL281208A (es)
JO (1) JOP20210033A1 (es)
LT (1) LT3846810T (es)
MA (1) MA53551B1 (es)
MD (1) MD3846810T2 (es)
MX (1) MX2021002474A (es)
NZ (1) NZ774400A (es)
PE (1) PE20211599A1 (es)
PH (1) PH12021550448A1 (es)
PL (1) PL3846810T3 (es)
PT (1) PT3846810T (es)
RS (1) RS64857B1 (es)
SG (1) SG11202101530PA (es)
SI (1) SI3846810T1 (es)
TW (1) TWI826514B (es)
WO (1) WO2020051137A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2019123406A (ru) 2014-02-05 2019-10-03 Мерк Шарп И Доум Корп. Технология приготовления таблеток для cgrp-активных соединений
MX2023001071A (es) * 2020-07-29 2023-05-12 Allergan Pharmaceuticals Int Ltd Tratamiento de la migraña.
US11717515B2 (en) 2020-12-22 2023-08-08 Allergan Pharmaceuticals International Limited Treatment of migraine

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5698571A (en) * 1994-10-05 1997-12-16 Eli Lilly And Company 5-HT1F mediated inhibition of neurogenic meningeal extravasation: a method for the treatment of migraine
TWI263497B (en) * 2002-03-29 2006-10-11 Lilly Co Eli Pyridinoylpiperidines as 5-HT1F agonists
PT2413933T (pt) * 2009-04-02 2017-12-12 Colucid Pharmaceuticals Inc Composição de 2,4,6-trifluoro-n-[6-(1-metil-piperidin-4-ilcarbonil)-piridin-2-il]-benzamida
US8697876B2 (en) * 2010-04-02 2014-04-15 Colucid Pharmaceuticals, Inc. Compositions and methods of synthesis of pyridinolypiperidine 5-HT1F agonists

Also Published As

Publication number Publication date
FI3846810T3 (fi) 2023-12-15
CA3111205A1 (en) 2020-03-12
TW202033197A (zh) 2020-09-16
DK3846810T3 (da) 2023-12-04
EP3846810A1 (en) 2021-07-14
PL3846810T3 (pl) 2024-03-18
AU2019336667A1 (en) 2021-03-11
HRP20231587T1 (hr) 2024-03-15
PT3846810T (pt) 2023-12-14
ECSP21015491A (es) 2021-04-29
JOP20210033A1 (ar) 2021-02-25
JP2021535913A (ja) 2021-12-23
KR102649644B1 (ko) 2024-03-21
CO2021002766A2 (es) 2021-03-19
MD3846810T2 (ro) 2024-04-30
EA202190440A1 (ru) 2021-06-24
AU2019336667B2 (en) 2022-09-29
BR112021002945A2 (pt) 2021-05-11
NZ774400A (en) 2024-03-22
ES2967665T3 (es) 2024-05-03
WO2020051137A1 (en) 2020-03-12
EP4279132A2 (en) 2023-11-22
JP7321256B2 (ja) 2023-08-04
EP4279132A3 (en) 2024-03-06
SG11202101530PA (en) 2021-03-30
IL281208A (en) 2021-04-29
RS64857B1 (sr) 2023-12-29
JP2023156344A (ja) 2023-10-24
TWI826514B (zh) 2023-12-21
US20210338655A1 (en) 2021-11-04
EP3846810B1 (en) 2023-10-18
CL2021000529A1 (es) 2021-08-13
DOP2021000039A (es) 2021-03-31
CR20210126A (es) 2021-04-22
PH12021550448A1 (en) 2021-09-27
HUE064519T2 (hu) 2024-03-28
PE20211599A1 (es) 2021-08-18
KR20210039419A (ko) 2021-04-09
MA53551A (fr) 2022-01-12
CN112638383A (zh) 2021-04-09
LT3846810T (lt) 2024-01-10
SI3846810T1 (sl) 2023-12-29
MA53551B1 (fr) 2023-11-30
AU2022291568A1 (en) 2023-02-02

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