ECSP21015491A - Administración prolongada de lasmiditan por la noche para la prevención de la migraña - Google Patents

Administración prolongada de lasmiditan por la noche para la prevención de la migraña

Info

Publication number
ECSP21015491A
ECSP21015491A ECSENADI202115491A ECDI202115491A ECSP21015491A EC SP21015491 A ECSP21015491 A EC SP21015491A EC SENADI202115491 A ECSENADI202115491 A EC SENADI202115491A EC DI202115491 A ECDI202115491 A EC DI202115491A EC SP21015491 A ECSP21015491 A EC SP21015491A
Authority
EC
Ecuador
Prior art keywords
migraine
prevention
night
meditan
prolonged administration
Prior art date
Application number
ECSENADI202115491A
Other languages
English (en)
Inventor
Gudarz Davar
Kirk Willis Johnson
Robert Russell Conley
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of ECSP21015491A publication Critical patent/ECSP21015491A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Saccharide Compounds (AREA)

Abstract

La presente invención se refiere al uso prolongado de lasmiditan por la noche para la prevención de la migraña, particularmente la migraña resistente al tratamiento que se define en el presente documento como migraña refractaria a dos o más esquemas de prevención o tratamiento previos de monoterapia y/o terapia doble.
ECSENADI202115491A 2018-09-04 2021-03-04 Administración prolongada de lasmiditan por la noche para la prevención de la migraña ECSP21015491A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862726585P 2018-09-04 2018-09-04

Publications (1)

Publication Number Publication Date
ECSP21015491A true ECSP21015491A (es) 2021-04-29

Family

ID=68051892

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSENADI202115491A ECSP21015491A (es) 2018-09-04 2021-03-04 Administración prolongada de lasmiditan por la noche para la prevención de la migraña

Country Status (35)

Country Link
US (1) US20210338655A1 (es)
EP (2) EP3846810B1 (es)
JP (2) JP7321256B2 (es)
KR (1) KR102649644B1 (es)
CN (1) CN112638383A (es)
AU (2) AU2019336667B2 (es)
BR (1) BR112021002945A2 (es)
CA (1) CA3111205A1 (es)
CL (1) CL2021000529A1 (es)
CO (1) CO2021002766A2 (es)
CR (1) CR20210126A (es)
DK (1) DK3846810T3 (es)
DO (1) DOP2021000039A (es)
EA (1) EA202190440A1 (es)
EC (1) ECSP21015491A (es)
ES (1) ES2967665T3 (es)
FI (1) FI3846810T3 (es)
HR (1) HRP20231587T1 (es)
HU (1) HUE064519T2 (es)
IL (1) IL281208A (es)
JO (1) JOP20210033A1 (es)
LT (1) LT3846810T (es)
MA (1) MA53551B1 (es)
MD (1) MD3846810T2 (es)
MX (1) MX2021002474A (es)
NZ (1) NZ774400A (es)
PE (1) PE20211599A1 (es)
PH (1) PH12021550448A1 (es)
PL (1) PL3846810T3 (es)
PT (1) PT3846810T (es)
RS (1) RS64857B1 (es)
SG (1) SG11202101530PA (es)
SI (1) SI3846810T1 (es)
TW (1) TWI826514B (es)
WO (1) WO2020051137A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2937315A1 (en) 2014-02-05 2015-08-13 Merck Sharp & Dohme Corp. Tablet formulation for cgrp-active compounds
BR112023001615A2 (pt) * 2020-07-29 2023-04-04 Allergan Pharmaceuticals Int Ltd Tratamento para enxaqueca
US11717515B2 (en) 2020-12-22 2023-08-08 Allergan Pharmaceuticals International Limited Treatment of migraine

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5698571A (en) * 1994-10-05 1997-12-16 Eli Lilly And Company 5-HT1F mediated inhibition of neurogenic meningeal extravasation: a method for the treatment of migraine
TWI263497B (en) * 2002-03-29 2006-10-11 Lilly Co Eli Pyridinoylpiperidines as 5-HT1F agonists
NZ596161A (en) * 2009-04-02 2013-11-29 Colucid Pharmaceuticals Inc Composition of 2,4,6-trifluoro-n-[6-(1-methyl-piperidin-4-carbonyl)-pyridin-2-yl]-benzamide
US8697876B2 (en) * 2010-04-02 2014-04-15 Colucid Pharmaceuticals, Inc. Compositions and methods of synthesis of pyridinolypiperidine 5-HT1F agonists

Also Published As

Publication number Publication date
EA202190440A1 (ru) 2021-06-24
SG11202101530PA (en) 2021-03-30
TW202033197A (zh) 2020-09-16
DOP2021000039A (es) 2021-03-31
KR20210039419A (ko) 2021-04-09
JP2021535913A (ja) 2021-12-23
DK3846810T3 (da) 2023-12-04
WO2020051137A1 (en) 2020-03-12
CN112638383A (zh) 2021-04-09
RS64857B1 (sr) 2023-12-29
JP7321256B2 (ja) 2023-08-04
HUE064519T2 (hu) 2024-03-28
LT3846810T (lt) 2024-01-10
JOP20210033A1 (ar) 2021-02-25
MA53551A (fr) 2022-01-12
BR112021002945A2 (pt) 2021-05-11
AU2022291568A1 (en) 2023-02-02
HRP20231587T1 (hr) 2024-03-15
CA3111205A1 (en) 2020-03-12
FI3846810T3 (fi) 2023-12-15
EP3846810B1 (en) 2023-10-18
CR20210126A (es) 2021-04-22
IL281208A (en) 2021-04-29
KR102649644B1 (ko) 2024-03-21
NZ774400A (en) 2024-03-22
PE20211599A1 (es) 2021-08-18
SI3846810T1 (sl) 2023-12-29
MX2021002474A (es) 2021-08-24
EP4279132A3 (en) 2024-03-06
MA53551B1 (fr) 2023-11-30
EP3846810A1 (en) 2021-07-14
EP4279132A2 (en) 2023-11-22
AU2019336667A1 (en) 2021-03-11
PT3846810T (pt) 2023-12-14
ES2967665T3 (es) 2024-05-03
CO2021002766A2 (es) 2021-03-19
PH12021550448A1 (en) 2021-09-27
US20210338655A1 (en) 2021-11-04
AU2019336667B2 (en) 2022-09-29
MD3846810T2 (ro) 2024-04-30
PL3846810T3 (pl) 2024-03-18
CL2021000529A1 (es) 2021-08-13
JP2023156344A (ja) 2023-10-24
TWI826514B (zh) 2023-12-21

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