MX2019015747A - Compuesto heterociclico. - Google Patents
Compuesto heterociclico.Info
- Publication number
- MX2019015747A MX2019015747A MX2019015747A MX2019015747A MX2019015747A MX 2019015747 A MX2019015747 A MX 2019015747A MX 2019015747 A MX2019015747 A MX 2019015747A MX 2019015747 A MX2019015747 A MX 2019015747A MX 2019015747 A MX2019015747 A MX 2019015747A
- Authority
- MX
- Mexico
- Prior art keywords
- heterocyclic compound
- formula
- present
- compound
- constipation
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4355—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención tiene como objetivo proporcionar un compuesto que puede ser útil para la profilaxis o tratamiento del estreñimiento y similares. La presente invención proporciona un compuesto representado por la siguiente fórmula (I): (ver Fórmula) en donde cada símbolo es como se describe en la especificación, o una sal del mismo.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2017120859 | 2017-06-20 | ||
JP2018005960 | 2018-01-17 | ||
US201862683418P | 2018-06-11 | 2018-06-11 | |
PCT/JP2018/023357 WO2018235838A1 (ja) | 2017-06-20 | 2018-06-19 | 複素環化合物 |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2019015747A true MX2019015747A (es) | 2020-02-20 |
Family
ID=69178190
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2019015747A MX2019015747A (es) | 2017-06-20 | 2018-06-19 | Compuesto heterociclico. |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP3643718B1 (es) |
JP (1) | JP7123042B2 (es) |
KR (1) | KR102658949B1 (es) |
CN (1) | CN110709401B (es) |
AU (1) | AU2018289939B2 (es) |
BR (1) | BR112019026096A2 (es) |
CA (1) | CA3068209A1 (es) |
MX (1) | MX2019015747A (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN114958325B (zh) * | 2021-02-24 | 2023-06-27 | 中国石油化工股份有限公司 | 一种耐高温缓蚀剂、制备方法及其在井筒防腐中的应用 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP4710445B2 (ja) * | 2004-07-08 | 2011-06-29 | 田辺三菱製薬株式会社 | 医薬組成物 |
KR101494059B1 (ko) | 2009-12-17 | 2015-02-16 | 머크 샤프 앤드 돔 코포레이션 | 퀴놀린 아미드 m1 수용체 양성 알로스테릭 조절제 |
EP2821401B1 (en) * | 2012-03-02 | 2020-09-09 | Takeda Pharmaceutical Company Limited | Dihydroquinolinone compounds as modulators of the muscarininc m1 receptor |
JP6211530B2 (ja) | 2012-11-19 | 2017-10-11 | 武田薬品工業株式会社 | 含窒素複素環化合物 |
CA2946519C (en) | 2014-04-23 | 2022-07-19 | Takeda Pharmaceutical Company Limited | Isoindoline-1-one derivatives as cholinergic muscarinic m1 receptor positive alloesteric modulator activity for the treatment of alzheimers disease |
WO2015174534A1 (ja) | 2014-05-16 | 2015-11-19 | 武田薬品工業株式会社 | 含窒素複素環化合物 |
WO2015190564A1 (ja) | 2014-06-13 | 2015-12-17 | 武田薬品工業株式会社 | 含窒素複素環化合物 |
WO2016009297A1 (en) * | 2014-07-18 | 2016-01-21 | Pfizer Inc. | Pyridine derivatives as muscarinic m1 receptor positive allosteric modulators |
US9878989B2 (en) | 2015-06-26 | 2018-01-30 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
US11111251B2 (en) * | 2016-02-16 | 2021-09-07 | Vanderbilt University | Positive allosteric modulators of the muscarinic acetylcholine receptor M1 |
MX2019002180A (es) * | 2016-09-02 | 2019-08-16 | Suven Life Sciences Ltd | Moduladores alostericos positivos del receptor m1 muscarinico. |
-
2018
- 2018-06-19 BR BR112019026096-0A patent/BR112019026096A2/pt unknown
- 2018-06-19 CA CA3068209A patent/CA3068209A1/en active Pending
- 2018-06-19 JP JP2019525643A patent/JP7123042B2/ja active Active
- 2018-06-19 KR KR1020207000757A patent/KR102658949B1/ko active IP Right Grant
- 2018-06-19 EP EP18819596.0A patent/EP3643718B1/en active Active
- 2018-06-19 AU AU2018289939A patent/AU2018289939B2/en active Active
- 2018-06-19 CN CN201880036933.2A patent/CN110709401B/zh active Active
- 2018-06-19 MX MX2019015747A patent/MX2019015747A/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP3643718B1 (en) | 2023-07-26 |
CA3068209A1 (en) | 2018-12-27 |
RU2019140596A (ru) | 2021-07-20 |
AU2018289939A1 (en) | 2020-01-30 |
RU2019140596A3 (es) | 2021-10-08 |
JPWO2018235838A1 (ja) | 2020-04-16 |
BR112019026096A2 (pt) | 2020-07-07 |
CN110709401B (zh) | 2023-06-13 |
JP7123042B2 (ja) | 2022-08-22 |
AU2018289939B2 (en) | 2022-06-16 |
KR20200013773A (ko) | 2020-02-07 |
EP3643718A1 (en) | 2020-04-29 |
EP3643718A4 (en) | 2021-03-03 |
CN110709401A (zh) | 2020-01-17 |
KR102658949B1 (ko) | 2024-04-18 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ZA201701299B (en) | Glycosidase inhibitors | |
SG11201901061QA (en) | Heterocyclic compound | |
MX2018010192A (es) | Inhibidores de glucosidasa. | |
MX2017006266A (es) | Compuestos de heteroarilo como inhibidores de cinasas asociadas al receptor de interleucina 1(irak) y sus usos. | |
MX2018010191A (es) | Inhibidores de glucosidasa. | |
PH12016500225B1 (en) | Novel quinoline-substituted compound | |
MX2020001757A (es) | Compuestos, sales de los mismos y metodos para el tratamiento de enfermedades. | |
JO3317B1 (ar) | مركبات تترا هيدروبيرولو ثيازين | |
PH12015501755A1 (en) | Azabenzimidazole compounds as inhibitors of pde4 isozymes for the treatment of cns and other disorders | |
PH12016502130B1 (en) | Novel pyrrolopyrimidine compound or salt thereof, pharmaceutical composition containing same, especially agent for prevention and/or treatment of tumors etc based on nae inhibitory effect | |
PH12015502611A1 (en) | Heterocyclic compounds as hedgehog signaling pathway inhibitors | |
MX2016005760A (es) | Inhibidores de glucogeno sintasa cinasa 3 (gsk-3). | |
NZ709986A (en) | Pharmaceutical compositions comprising nitroxyl donors | |
MX2019010085A (es) | Inhibidores de la glicosidasa de sulfoximina. | |
MX2021015514A (es) | Compuesto heterociclico. | |
MX2017013880A (es) | Derivados del acido tetrahidronaftiridinil propionico y usos de los mismos. | |
PH12019502248A1 (en) | Ip6k inhibitors | |
PH12015501038A1 (en) | Inhibitors of iap | |
MX2018005004A (es) | Compuestos de indazol substituidos como inhibidores de rorgammat y sus usos. | |
PH12015502032A1 (en) | Azetidinyloxyphenylpyrrolidine compounds | |
WO2018194181A8 (en) | HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF ACETYLCHOLINE RECEPTORS | |
MY193239A (en) | Novel b-lactamase inhibitors | |
GEP20186893B (en) | Pyrazines modulators of gpr6 | |
AU2016363719A8 (en) | 1,3,4-thiadiazole compounds and their use in treating cancer | |
MX2019015747A (es) | Compuesto heterociclico. |