MX2019014483A - Regimenes de dosificación de antagonistas de hormona liberadora de gonadotropina para el tratamiento de endometriosis. - Google Patents

Regimenes de dosificación de antagonistas de hormona liberadora de gonadotropina para el tratamiento de endometriosis.

Info

Publication number
MX2019014483A
MX2019014483A MX2019014483A MX2019014483A MX2019014483A MX 2019014483 A MX2019014483 A MX 2019014483A MX 2019014483 A MX2019014483 A MX 2019014483A MX 2019014483 A MX2019014483 A MX 2019014483A MX 2019014483 A MX2019014483 A MX 2019014483A
Authority
MX
Mexico
Prior art keywords
gonadotropin
endometriosis
dosing regimens
releasing hormone
treatment
Prior art date
Application number
MX2019014483A
Other languages
English (en)
Spanish (es)
Inventor
Jean-Pierre Gotteland
Ernest Loumaye
Original Assignee
ObsEva SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ObsEva SA filed Critical ObsEva SA
Publication of MX2019014483A publication Critical patent/MX2019014483A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • A61K38/09Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Reproductive Health (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Cell Biology (AREA)
  • Food Science & Technology (AREA)
  • Physics & Mathematics (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • General Physics & Mathematics (AREA)
  • Pathology (AREA)
  • Apparatus For Radiation Diagnosis (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
MX2019014483A 2017-06-05 2018-06-05 Regimenes de dosificación de antagonistas de hormona liberadora de gonadotropina para el tratamiento de endometriosis. MX2019014483A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762515268P 2017-06-05 2017-06-05
PCT/EP2018/064768 WO2018224498A1 (en) 2017-06-05 2018-06-05 Gonadotropin-releasing hormone antagonist dosing regimens for the treatment of endometriosis

Publications (1)

Publication Number Publication Date
MX2019014483A true MX2019014483A (es) 2020-08-17

Family

ID=62620835

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2019014483A MX2019014483A (es) 2017-06-05 2018-06-05 Regimenes de dosificación de antagonistas de hormona liberadora de gonadotropina para el tratamiento de endometriosis.

Country Status (12)

Country Link
US (2) US11980621B2 (cg-RX-API-DMAC7.html)
EP (1) EP3634418A1 (cg-RX-API-DMAC7.html)
JP (2) JP7348171B2 (cg-RX-API-DMAC7.html)
KR (2) KR20250117836A (cg-RX-API-DMAC7.html)
CN (1) CN110996956A (cg-RX-API-DMAC7.html)
AU (2) AU2018280742B2 (cg-RX-API-DMAC7.html)
CA (1) CA3066190A1 (cg-RX-API-DMAC7.html)
EA (1) EA201992612A1 (cg-RX-API-DMAC7.html)
MA (1) MA49256A (cg-RX-API-DMAC7.html)
MX (1) MX2019014483A (cg-RX-API-DMAC7.html)
SG (1) SG11201911598WA (cg-RX-API-DMAC7.html)
WO (1) WO2018224498A1 (cg-RX-API-DMAC7.html)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK3518933T4 (da) 2016-09-30 2025-04-22 Takeda Pharmaceuticals Co Fremgangsmåder til behandling af uterusfibromer og endometriose
MX2019014482A (es) 2017-06-05 2020-08-17 ObsEva SA Régimenes de dosificación de antagonistas de hormona liberadora de gonadotropina para tratar miomas uterinos y reducir la menstruación.
KR20250117836A (ko) 2017-06-05 2025-08-05 깃세이 야쿠힌 고교 가부시키가이샤 자궁내막증의 치료를 위한 고나도트로핀 방출 호르몬 길항제 투약 요법
EP3873465B1 (en) 2018-10-29 2025-01-15 Kissei Pharmaceutical Co., Ltd. Compositions and methods for the treatment of adenomyosis and rectovaginal endometriosis
US20220305017A1 (en) * 2019-08-08 2022-09-29 ObsEva S.A. Compositions and methods for the treatment of estrogen-dependent disorders
CN113384581B (zh) * 2020-03-12 2023-11-14 成都倍特药业股份有限公司 一种包含促性腺激素释放激素拮抗剂的药物组合物
WO2022101303A1 (en) * 2020-11-11 2022-05-19 Myovant Sciences Gmbh Methods of administering relugolix
TWI796144B (zh) * 2021-02-23 2023-03-11 大陸商南京明德新藥研發有限公司 噻吩並嘧啶二酮類化合物及其應用
CN115232144B (zh) * 2021-04-22 2024-04-02 长春金赛药业有限责任公司 含氮稠环类衍生物、药物组合物及其制备方法和应用

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US7109171B2 (en) 2000-02-28 2006-09-19 Praecis Pharmaceuticals Inc. Methods for treating FSH related conditions with GnRH antagonists
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EP1591446B1 (en) 2003-01-29 2013-03-06 Takeda Pharmaceutical Company Limited Thienopyrimidine compounds and use thereof
ATE407679T1 (de) 2003-07-07 2008-09-15 Neurocrine Biosciences Inc Pyrimidin-2,4-dion-derivate als gonadotropin freisetzende hormon-rezeptor-antagonisten
BRPI0609625A2 (pt) 2005-03-31 2010-04-20 Astellas Pharma Inc derivados de propano-1,3-diona ou sal destes
BRPI0617436B8 (pt) 2005-10-19 2021-05-25 Kissei Pharmaceutical derivado heterocíclico fundido, composição farmacêutica compreendendo o mesmo e usos do dito derivado na prevenção ou tratamento de doença dependente de hormônio sexual e na regulação da reprodução, contracepção ou indução de ovulação
US8765948B2 (en) 2007-11-07 2014-07-01 Neurocrine Biosciences, Inc. Processes for the preparation of uracil derivatives
BR112012020110B1 (pt) 2010-02-10 2021-06-08 Kissei Pharmaceutical Co., Ltd. composto derivado heterocíclico fusionado, composição farmacêutica que compreende o mesmo e uso terapêutico do dito composto
HK1199878A1 (en) 2012-01-16 2015-07-24 Bayer Intellectual Property Gmbh Spiroindoline derivatives as gonadotropin-releasing hormone receptor antagonists
EP2817621A4 (en) 2012-02-21 2016-02-24 Univ Northwestern PROOF OF ANTI-MÜLLER-HORMON IN FULL BLOOD
CN104603114B (zh) 2012-09-07 2017-06-20 安斯泰来制药株式会社 磺酰脒化合物的制造方法
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LT3415517T (lt) 2012-09-28 2022-06-10 Takeda Pharmaceutical Company Limited Kristalinė 1-(4-(1-(2,6-difluorbenzil)-5-dimetilaminometil-3-(6-metoksipiridazin-3-il)-2,4-diokso-1,2,3,4- tetrahidrotieno(2,3-d)pirimidin-6-il)fenil)-3-metoksikarbamido forma
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CA3025760A1 (en) 2016-08-08 2018-02-15 Kissei Pharmaceutical Co., Ltd. Usage and dosage of therapeutic agents for endometriosis
DK3518933T4 (da) 2016-09-30 2025-04-22 Takeda Pharmaceuticals Co Fremgangsmåder til behandling af uterusfibromer og endometriose
KR20250117836A (ko) 2017-06-05 2025-08-05 깃세이 야쿠힌 고교 가부시키가이샤 자궁내막증의 치료를 위한 고나도트로핀 방출 호르몬 길항제 투약 요법
MX2019014482A (es) 2017-06-05 2020-08-17 ObsEva SA Régimenes de dosificación de antagonistas de hormona liberadora de gonadotropina para tratar miomas uterinos y reducir la menstruación.
EP3876943A2 (en) 2018-11-07 2021-09-15 ObsEva S.A. Compositions and methods for the treatment of estrogen-dependent disorders

Also Published As

Publication number Publication date
US20240293414A1 (en) 2024-09-05
JP2020522571A (ja) 2020-07-30
KR20200027481A (ko) 2020-03-12
JP7348171B2 (ja) 2023-09-20
JP7657855B2 (ja) 2025-04-07
CA3066190A1 (en) 2018-12-13
EA201992612A1 (ru) 2020-05-20
AU2018280742B2 (en) 2023-12-21
KR20250117836A (ko) 2025-08-05
EP3634418A1 (en) 2020-04-15
AU2024201701A1 (en) 2024-04-04
CN110996956A (zh) 2020-04-10
KR102839190B1 (ko) 2025-07-28
SG11201911598WA (en) 2020-01-30
AU2024201701B2 (en) 2025-04-10
WO2018224498A1 (en) 2018-12-13
US11980621B2 (en) 2024-05-14
US20200138819A1 (en) 2020-05-07
JP2023113715A (ja) 2023-08-16
AU2018280742A1 (en) 2020-01-30
MA49256A (fr) 2021-05-26

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