MX2017012661A - Procesos para preparar cloruro de 2-tiofenocarbonilo. - Google Patents

Procesos para preparar cloruro de 2-tiofenocarbonilo.

Info

Publication number
MX2017012661A
MX2017012661A MX2017012661A MX2017012661A MX2017012661A MX 2017012661 A MX2017012661 A MX 2017012661A MX 2017012661 A MX2017012661 A MX 2017012661A MX 2017012661 A MX2017012661 A MX 2017012661A MX 2017012661 A MX2017012661 A MX 2017012661A
Authority
MX
Mexico
Prior art keywords
preparation
processes
thiophenecarbonyl chloride
thiophenecarbonyl
chloride
Prior art date
Application number
MX2017012661A
Other languages
English (en)
Inventor
William H Miller
p walker Daniel
Original Assignee
Monsanto Technology Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Monsanto Technology Llc filed Critical Monsanto Technology Llc
Publication of MX2017012661A publication Critical patent/MX2017012661A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/12—Radicals substituted by halogen atoms or nitro or nitroso radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)

Abstract

En la presente se proporcionan procesos para la preparación cloruro de 2-tiofenocarbonilo, el cual es útil, por ejemplo, en la preparación de 1,2,4-oxadiazoles 3,5-disustituidos, como tioxazafeno (3-fenil-5-(2-tienil)-1,2,4- oxadiazol).
MX2017012661A 2015-03-31 2016-03-31 Procesos para preparar cloruro de 2-tiofenocarbonilo. MX2017012661A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562140915P 2015-03-31 2015-03-31
PCT/US2016/025159 WO2016161063A1 (en) 2015-03-31 2016-03-31 Processes for the preparation of 2-thiophenecarbonyl chloride

Publications (1)

Publication Number Publication Date
MX2017012661A true MX2017012661A (es) 2018-01-09

Family

ID=57007579

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017012661A MX2017012661A (es) 2015-03-31 2016-03-31 Procesos para preparar cloruro de 2-tiofenocarbonilo.

Country Status (11)

Country Link
US (1) US10239857B2 (es)
EP (1) EP3277275A4 (es)
JP (1) JP6559798B2 (es)
KR (1) KR102096420B1 (es)
CN (1) CN107530327A (es)
AR (1) AR104159A1 (es)
AU (1) AU2016242884B2 (es)
BR (1) BR112017020718A2 (es)
CA (1) CA2981066A1 (es)
MX (1) MX2017012661A (es)
WO (1) WO2016161063A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2017238056A1 (en) * 2016-03-24 2018-10-04 Monsanto Technology Llc Processes for the preparation of heteroaryl carboxylic acids
KR102420944B1 (ko) 2016-10-26 2022-07-15 이시하라 산교 가부시끼가이샤 3-메틸-2-티오펜카르복실산의 제조 방법
CN110937983A (zh) * 2019-12-27 2020-03-31 大连奇凯医药科技有限公司 以六氟苯为溶剂生产三氯甲氧基苯的方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2229897A (en) * 1940-03-02 1941-01-28 American Cyanamid Co Method of preparing alpha hydroxy carboxylic acids
US3959569A (en) 1970-07-27 1976-05-25 The Dow Chemical Company Preparation of water-absorbent articles
US3741984A (en) 1971-08-19 1973-06-26 Du Pont N-sulfamoyl-2-thiopenecarboxamides
JPS5422363A (en) * 1977-07-19 1979-02-20 Seitetsu Kagaku Co Ltd Preparation of thiophene-substituted fatty acid halide
JPS6081182A (ja) * 1983-10-12 1985-05-09 Kissei Pharmaceut Co Ltd チオフエン誘導体及びその製造方法
US4556672A (en) * 1984-03-19 1985-12-03 Pfizer Inc. 3-Substituted 2-oxindole-1-carboxamides as analgesic and anti-inflammatory agents
US4565812A (en) * 1984-11-30 1986-01-21 Chevron Research Company Fungicidal tin salts of thienyl and furyl hydroxamic acids, compositions, and method of use therefor
DE3812175A1 (de) * 1988-04-13 1989-10-26 Bayer Ag Verfahren zur herstellung von carbonsaeurehalogeniden
DE4011172A1 (de) * 1990-04-06 1991-10-10 Degussa Verbindungen zur bekaempfung von pflanzenkrankheiten
US5371240A (en) * 1992-11-30 1994-12-06 Torcan Chemical Ltd. Process for the preparation of pure thiophene derivatives
US20080167286A1 (en) * 2006-12-12 2008-07-10 Abbott Laboratories Pharmaceutical compositions and their methods of use
CA3081731A1 (en) * 2007-08-13 2009-02-19 Monsanto Technology Llc Compositions and methods for controlling nematodes
JP5578809B2 (ja) * 2008-06-26 2014-08-27 石原産業株式会社 ３−メチル−２−チオフェンカルボン酸の製造方法
DK2867230T3 (da) * 2012-07-02 2020-04-14 Monsanto Technology Llc Fremgangsmåde til fremstilling af 3,5-disubstitueret 1,2,4-oxadiazoler
CN103980265A (zh) * 2014-05-14 2014-08-13 武汉工程大学 3-苯基-5-(噻吩-2基)-1,2,4-噁二唑的合成工艺

Also Published As

Publication number Publication date
KR20170137741A (ko) 2017-12-13
EP3277275A4 (en) 2018-07-11
BR112017020718A2 (pt) 2018-06-26
WO2016161063A1 (en) 2016-10-06
AU2016242884A1 (en) 2017-10-05
EP3277275A1 (en) 2018-02-07
AU2016242884B2 (en) 2019-11-07
KR102096420B1 (ko) 2020-04-02
JP2018511606A (ja) 2018-04-26
CA2981066A1 (en) 2016-10-06
CN107530327A (zh) 2018-01-02
US10239857B2 (en) 2019-03-26
US20180162830A1 (en) 2018-06-14
JP6559798B2 (ja) 2019-08-14
AR104159A1 (es) 2017-06-28

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