BR112017020718A2 - processos para a preparação de cloreto de 2-tiofenocarbonila - Google Patents
processos para a preparação de cloreto de 2-tiofenocarbonilaInfo
- Publication number
- BR112017020718A2 BR112017020718A2 BR112017020718A BR112017020718A BR112017020718A2 BR 112017020718 A2 BR112017020718 A2 BR 112017020718A2 BR 112017020718 A BR112017020718 A BR 112017020718A BR 112017020718 A BR112017020718 A BR 112017020718A BR 112017020718 A2 BR112017020718 A2 BR 112017020718A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- thiophenocarbonyl
- chloride
- processes
- oxadiazols
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/12—Radicals substituted by halogen atoms or nitro or nitroso radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Abstract
a presente invenção refere-se a processos para a preparação de cloreto de 2-tiofenocarbonila, que é útil, por exemplo, na preparação de 1,2,4-oxadiazóis 3,5-dissubstituídos, como tioxazafen (3-fenil-5-(2-tienil)-1,2,4-oxadiazol).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562140915P | 2015-03-31 | 2015-03-31 | |
PCT/US2016/025159 WO2016161063A1 (en) | 2015-03-31 | 2016-03-31 | Processes for the preparation of 2-thiophenecarbonyl chloride |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112017020718A2 true BR112017020718A2 (pt) | 2018-06-26 |
Family
ID=57007579
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112017020718A BR112017020718A2 (pt) | 2015-03-31 | 2016-03-31 | processos para a preparação de cloreto de 2-tiofenocarbonila |
Country Status (11)
Country | Link |
---|---|
US (1) | US10239857B2 (pt) |
EP (1) | EP3277275A4 (pt) |
JP (1) | JP6559798B2 (pt) |
KR (1) | KR102096420B1 (pt) |
CN (1) | CN107530327A (pt) |
AR (1) | AR104159A1 (pt) |
AU (1) | AU2016242884B2 (pt) |
BR (1) | BR112017020718A2 (pt) |
CA (1) | CA2981066A1 (pt) |
MX (1) | MX2017012661A (pt) |
WO (1) | WO2016161063A1 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112018069255A2 (pt) * | 2016-03-24 | 2019-01-22 | Monsanto Technology Llc | processos para a preparação de ácidos heteroaril carboxílicos |
EP3533791B1 (en) * | 2016-10-26 | 2020-12-30 | Ishihara Sangyo Kaisha, Ltd. | Method for producing 3-methyl-2-thiophenecarboxylic acid |
CN110937983A (zh) * | 2019-12-27 | 2020-03-31 | 大连奇凯医药科技有限公司 | 以六氟苯为溶剂生产三氯甲氧基苯的方法 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2229897A (en) * | 1940-03-02 | 1941-01-28 | American Cyanamid Co | Method of preparing alpha hydroxy carboxylic acids |
US3959569A (en) | 1970-07-27 | 1976-05-25 | The Dow Chemical Company | Preparation of water-absorbent articles |
US3741984A (en) * | 1971-08-19 | 1973-06-26 | Du Pont | N-sulfamoyl-2-thiopenecarboxamides |
JPS5422363A (en) * | 1977-07-19 | 1979-02-20 | Seitetsu Kagaku Co Ltd | Preparation of thiophene-substituted fatty acid halide |
JPS6081182A (ja) * | 1983-10-12 | 1985-05-09 | Kissei Pharmaceut Co Ltd | チオフエン誘導体及びその製造方法 |
US4556672A (en) * | 1984-03-19 | 1985-12-03 | Pfizer Inc. | 3-Substituted 2-oxindole-1-carboxamides as analgesic and anti-inflammatory agents |
US4565812A (en) * | 1984-11-30 | 1986-01-21 | Chevron Research Company | Fungicidal tin salts of thienyl and furyl hydroxamic acids, compositions, and method of use therefor |
DE3812175A1 (de) * | 1988-04-13 | 1989-10-26 | Bayer Ag | Verfahren zur herstellung von carbonsaeurehalogeniden |
DE4011172A1 (de) | 1990-04-06 | 1991-10-10 | Degussa | Verbindungen zur bekaempfung von pflanzenkrankheiten |
US5371240A (en) * | 1992-11-30 | 1994-12-06 | Torcan Chemical Ltd. | Process for the preparation of pure thiophene derivatives |
US20080167286A1 (en) * | 2006-12-12 | 2008-07-10 | Abbott Laboratories | Pharmaceutical compositions and their methods of use |
BR122018001851B1 (pt) * | 2007-08-13 | 2019-08-20 | Monsanto Technology Llc | Método de controle de nematódeos parasitas de plantas |
JP5578809B2 (ja) * | 2008-06-26 | 2014-08-27 | 石原産業株式会社 | 3−メチル−2−チオフェンカルボン酸の製造方法 |
CA2876215A1 (en) * | 2012-07-02 | 2014-01-09 | Monsanto Technology Llc | Processes for the preparation of 3,5-disubstituted-1,2,4-oxadiazoles |
CN103980265A (zh) * | 2014-05-14 | 2014-08-13 | 武汉工程大学 | 3-苯基-5-(噻吩-2基)-1,2,4-噁二唑的合成工艺 |
-
2016
- 2016-03-31 CN CN201680019709.3A patent/CN107530327A/zh active Pending
- 2016-03-31 JP JP2017551110A patent/JP6559798B2/ja not_active Expired - Fee Related
- 2016-03-31 KR KR1020177028582A patent/KR102096420B1/ko active IP Right Grant
- 2016-03-31 CA CA2981066A patent/CA2981066A1/en not_active Abandoned
- 2016-03-31 WO PCT/US2016/025159 patent/WO2016161063A1/en active Application Filing
- 2016-03-31 AU AU2016242884A patent/AU2016242884B2/en not_active Expired - Fee Related
- 2016-03-31 US US15/563,008 patent/US10239857B2/en not_active Expired - Fee Related
- 2016-03-31 MX MX2017012661A patent/MX2017012661A/es unknown
- 2016-03-31 EP EP16774164.4A patent/EP3277275A4/en not_active Withdrawn
- 2016-03-31 AR ARP160100874A patent/AR104159A1/es unknown
- 2016-03-31 BR BR112017020718A patent/BR112017020718A2/pt not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP3277275A1 (en) | 2018-02-07 |
KR20170137741A (ko) | 2017-12-13 |
JP6559798B2 (ja) | 2019-08-14 |
EP3277275A4 (en) | 2018-07-11 |
US10239857B2 (en) | 2019-03-26 |
CA2981066A1 (en) | 2016-10-06 |
MX2017012661A (es) | 2018-01-09 |
US20180162830A1 (en) | 2018-06-14 |
AU2016242884A1 (en) | 2017-10-05 |
WO2016161063A1 (en) | 2016-10-06 |
AR104159A1 (es) | 2017-06-28 |
CN107530327A (zh) | 2018-01-02 |
KR102096420B1 (ko) | 2020-04-02 |
JP2018511606A (ja) | 2018-04-26 |
AU2016242884B2 (en) | 2019-11-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
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B07G | Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette] | ||
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements | ||
B350 | Update of information on the portal [chapter 15.35 patent gazette] |