MX2016017147A - Compuestos de indazole substituidos como inhibidores de irak4. - Google Patents

Compuestos de indazole substituidos como inhibidores de irak4.

Info

Publication number
MX2016017147A
MX2016017147A MX2016017147A MX2016017147A MX2016017147A MX 2016017147 A MX2016017147 A MX 2016017147A MX 2016017147 A MX2016017147 A MX 2016017147A MX 2016017147 A MX2016017147 A MX 2016017147A MX 2016017147 A MX2016017147 A MX 2016017147A
Authority
MX
Mexico
Prior art keywords
substituted indazole
indazole compounds
irak4 inhibitors
irak4
inhibitors
Prior art date
Application number
MX2016017147A
Other languages
English (en)
Spanish (es)
Inventor
Rao Gummadi Venkateshwar
Samajdar Susanta
Original Assignee
Aurigene Discovery Tech Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aurigene Discovery Tech Ltd filed Critical Aurigene Discovery Tech Ltd
Publication of MX2016017147A publication Critical patent/MX2016017147A/es

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
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  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Neurosurgery (AREA)
  • Otolaryngology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2016017147A 2014-06-20 2015-06-19 Compuestos de indazole substituidos como inhibidores de irak4. MX2016017147A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN3017CH2014 2014-06-20
PCT/IB2015/054620 WO2015193846A1 (en) 2014-06-20 2015-06-19 Substituted indazole compounds as irak4 inhibitors

Publications (1)

Publication Number Publication Date
MX2016017147A true MX2016017147A (es) 2017-06-07

Family

ID=54934936

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016017147A MX2016017147A (es) 2014-06-20 2015-06-19 Compuestos de indazole substituidos como inhibidores de irak4.

Country Status (16)

Country Link
US (1) US20170152263A1 (enExample)
EP (1) EP3157521A4 (enExample)
JP (1) JP2017518348A (enExample)
KR (1) KR20170016500A (enExample)
CN (1) CN106456609A (enExample)
AU (1) AU2015275730A1 (enExample)
BR (1) BR112016029853A2 (enExample)
CA (1) CA2952188A1 (enExample)
CU (1) CU20160188A7 (enExample)
EA (1) EA201692418A1 (enExample)
HK (1) HK1231411A1 (enExample)
IL (1) IL249345A0 (enExample)
MX (1) MX2016017147A (enExample)
PH (1) PH12016502382A1 (enExample)
SG (1) SG11201610009XA (enExample)
WO (1) WO2015193846A1 (enExample)

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TW201701879A (zh) 2015-04-30 2017-01-16 拜耳製藥公司 Ｉｒａｋ４抑制劑組合
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JP2020524663A (ja) 2017-06-21 2020-08-20 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ Ｉｒａｋ４調節因子としてのイソインドリノン誘導体
EP3642204A1 (en) 2017-06-21 2020-04-29 H. Hoffnabb-La Roche Ag PYRAZOLO[1,5a]PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS
US10722495B2 (en) 2017-09-08 2020-07-28 Incyte Corporation Cyanoindazole compounds and uses thereof
JP7366031B2 (ja) 2017-09-22 2023-10-20 カイメラ セラピューティクス， インコーポレイテッド タンパク質分解剤およびそれらの使用
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