MX2015012146A - Forma cristalina de una sal de acido tiazolilacetico sustituido y trietilamina. - Google Patents

Forma cristalina de una sal de acido tiazolilacetico sustituido y trietilamina.

Info

Publication number
MX2015012146A
MX2015012146A MX2015012146A MX2015012146A MX2015012146A MX 2015012146 A MX2015012146 A MX 2015012146A MX 2015012146 A MX2015012146 A MX 2015012146A MX 2015012146 A MX2015012146 A MX 2015012146A MX 2015012146 A MX2015012146 A MX 2015012146A
Authority
MX
Mexico
Prior art keywords
crystalline form
triethylamine salt
acid triethylamine
substituted
thiazolylacetic acid
Prior art date
Application number
MX2015012146A
Other languages
English (en)
Other versions
MX351963B (es
Inventor
Weijiang Zhang
Michael R Tracey
Junning Lee
Original Assignee
Theravance Biopharma Antibiotics Ip Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theravance Biopharma Antibiotics Ip Llc filed Critical Theravance Biopharma Antibiotics Ip Llc
Publication of MX2015012146A publication Critical patent/MX2015012146A/es
Publication of MX351963B publication Critical patent/MX351963B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/40—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • C07D277/593—Z being doubly bound oxygen or doubly bound nitrogen, which nitrogen is part of a possibly substituted oximino radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)

Abstract

Una forma cristalina de una sal con trietilamina del ácido (2Z)-2-(2-amino-5-clorotiazol-4-il)-2-(3-N-tert-butoxicarbonilami nopropoxiimino)acético. También, procesos e intermediarios para preparar la forma cristalina. La forma cristalina es útil como intermediario para preparar antibióticos de glicopéptido reticulado-cefalosporina.
MX2015012146A 2013-03-13 2014-03-06 Forma cristalina de una sal de ácido tiazolilacético sustituido y trietilamina. MX351963B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361779091P 2013-03-13 2013-03-13
PCT/US2014/021080 WO2014164187A1 (en) 2013-03-13 2014-03-06 Crystalline form of a substituted thiazolylacetic acid triethylamine salt

Publications (2)

Publication Number Publication Date
MX2015012146A true MX2015012146A (es) 2015-11-25
MX351963B MX351963B (es) 2017-11-06

Family

ID=50382685

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015012146A MX351963B (es) 2013-03-13 2014-03-06 Forma cristalina de una sal de ácido tiazolilacético sustituido y trietilamina.

Country Status (20)

Country Link
US (1) US9139542B2 (es)
EP (1) EP2970164B1 (es)
JP (2) JP6404309B2 (es)
KR (1) KR20150126368A (es)
CN (1) CN105121417B (es)
AU (1) AU2014249611B2 (es)
BR (1) BR112015022600A2 (es)
CA (1) CA2902724A1 (es)
EA (1) EA027911B1 (es)
ES (1) ES2634019T3 (es)
GE (1) GEP201706779B (es)
HK (1) HK1214596A1 (es)
IL (1) IL240600A0 (es)
MD (1) MD4719C1 (es)
MX (1) MX351963B (es)
PH (1) PH12015502067A1 (es)
SG (1) SG11201507221VA (es)
TW (1) TWI627165B (es)
UA (1) UA115087C2 (es)
WO (1) WO2014164187A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2021014751A (es) * 2019-05-31 2022-01-18 Hyundai Pharm Co Ltd Forma cristalina novedosa de derivado de acido 3-(4-(benciloxi)fenil)hex-4-inoico.

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4372952A (en) 1978-07-31 1983-02-08 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4284631A (en) 1978-07-31 1981-08-18 Fujisawa Pharmaceutical Co., Ltd. 7-Substituted cephem compounds and pharmaceutical antibacterial compositions containing them
US4341775A (en) 1978-09-11 1982-07-27 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
GB2033377B (en) 1978-09-11 1983-05-05 Fujisawa Pharmaceuticalco Ltd Cephem compounds and processes for preparation thereof
US4220761A (en) 1978-09-12 1980-09-02 Fujisawa Pharmaceutical Co., Ltd. 7-[Substituted oximinoacetamido]-3-[hydroxy alkyltetrazolo]cephalosporin derivatives
DE2945248A1 (de) 1978-11-13 1980-05-22 Fujisawa Pharmaceutical Co Cephem-verbindungen, verfahren zu ihrer herstellung und sie enthaltende antibakterielle pharmazeutische mittel
DE3177090D1 (en) * 1980-12-31 1989-09-28 Fujisawa Pharmaceutical Co 7-acylaminocephalosporanic acid derivatives and processes for the preparation thereof
JP2519054B2 (ja) 1986-06-09 1996-07-31 武田薬品工業株式会社 新規セフェム化合物
AU1630988A (en) 1987-05-30 1988-12-01 Kyoto Pharmaceutical Industries, Ltd. Cephalosporin compound and pharmaceutical composition thereof
JPH04221388A (ja) * 1990-12-20 1992-08-11 Asahi Chem Ind Co Ltd セファロスポリン化合物およびその製造法
TWI335332B (en) * 2001-10-12 2011-01-01 Theravance Inc Cross-linked vancomycin-cephalosporin antibiotics
ITMI20012363A1 (it) 2001-11-09 2003-05-09 Antibioticos Spa Metodo per la sintesi di catene laterali di cefalosporine
ES2384707T3 (es) 2002-05-24 2012-07-11 Theravance, Inc. Antibióticos entrecruzados de glucopéptidos y cefalosporinas
GB0416379D0 (en) 2004-07-22 2004-08-25 Sandoz Ag Organic compounds
TW200637559A (en) 2005-03-29 2006-11-01 Shionogi & Co 3-propenylcefem derivative

Also Published As

Publication number Publication date
CN105121417A (zh) 2015-12-02
AU2014249611B2 (en) 2017-12-21
SG11201507221VA (en) 2015-10-29
EP2970164A1 (en) 2016-01-20
WO2014164187A1 (en) 2014-10-09
CN105121417B (zh) 2017-11-17
EA027911B1 (ru) 2017-09-29
US20140275554A1 (en) 2014-09-18
TWI627165B (zh) 2018-06-21
MX351963B (es) 2017-11-06
US9139542B2 (en) 2015-09-22
ES2634019T3 (es) 2017-09-26
UA115087C2 (uk) 2017-09-11
MD4719B1 (ro) 2020-10-31
BR112015022600A2 (pt) 2017-07-18
JP2018197256A (ja) 2018-12-13
CA2902724A1 (en) 2014-10-09
MD4719C1 (ro) 2021-05-31
MD20150099A2 (ro) 2016-02-29
EA201591708A1 (ru) 2016-01-29
JP6404309B2 (ja) 2018-10-10
TW201444810A (zh) 2014-12-01
GEP201706779B (en) 2017-11-27
EP2970164B1 (en) 2017-05-03
AU2014249611A1 (en) 2015-09-17
JP2016512257A (ja) 2016-04-25
IL240600A0 (en) 2015-09-24
PH12015502067B1 (en) 2016-01-25
HK1214596A1 (zh) 2016-07-29
KR20150126368A (ko) 2015-11-11
PH12015502067A1 (en) 2016-01-25

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