MX361673B - Procedimiento para la preparación de intermediarios de ácido borónico. - Google Patents
Procedimiento para la preparación de intermediarios de ácido borónico.Info
- Publication number
- MX361673B MX361673B MX2015015346A MX2015015346A MX361673B MX 361673 B MX361673 B MX 361673B MX 2015015346 A MX2015015346 A MX 2015015346A MX 2015015346 A MX2015015346 A MX 2015015346A MX 361673 B MX361673 B MX 361673B
- Authority
- MX
- Mexico
- Prior art keywords
- preparation
- boronic acid
- acid intermediates
- intermediates
- pyrimidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Abstract
La presente invención se refiere a un procedimiento mejorado para la preparación de ácido 2-amino-pirimidín-5-borónico de fórmula (I). (ver Fórmula) o sales o ésteres del mismo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP13166587 | 2013-05-06 | ||
PCT/EP2014/059023 WO2014180752A1 (en) | 2013-05-06 | 2014-05-05 | Process for the preparation of boronic acid intermediates |
Publications (2)
Publication Number | Publication Date |
---|---|
MX2015015346A MX2015015346A (es) | 2016-03-04 |
MX361673B true MX361673B (es) | 2018-12-11 |
Family
ID=48227048
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2015015346A MX361673B (es) | 2013-05-06 | 2014-05-05 | Procedimiento para la preparación de intermediarios de ácido borónico. |
Country Status (12)
Country | Link |
---|---|
US (1) | US9102689B2 (es) |
EP (1) | EP2994472B1 (es) |
JP (1) | JP6456925B2 (es) |
KR (1) | KR101813775B1 (es) |
CN (1) | CN105189519B (es) |
AR (1) | AR096178A1 (es) |
BR (1) | BR112015027475B1 (es) |
CA (1) | CA2910541C (es) |
HK (1) | HK1213554A1 (es) |
MX (1) | MX361673B (es) |
RU (1) | RU2658915C2 (es) |
WO (1) | WO2014180752A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2801577A1 (en) * | 2013-05-06 | 2014-11-12 | Euticals S.P.A. | Process for the preparation of aminoaryl- and aminoheteroaryl boronic acids and esters |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10322843A1 (de) | 2003-05-19 | 2004-12-16 | Clariant Gmbh | Verfahren zur Herstellung von Anilinboronsäuren und ihren Derivaten |
ES2544082T3 (es) * | 2006-12-07 | 2015-08-27 | F. Hoffmann-La Roche Ag | Compuestos inhibidores de fosfoinosítido 3-quinasa y métodos de uso |
EP1988095B1 (de) * | 2007-04-27 | 2016-01-27 | Euticals GmbH | Verfarhen zur Herstellung von Aminoaryl- bzw. heteroarylboronsaeuren und ihren Derivaten |
CN102399235A (zh) | 2011-10-25 | 2012-04-04 | 江苏弘和药物研发有限公司 | 一种2-氨基-5-嘧啶硼酸频哪醇酯的合成方法 |
CN102367260A (zh) * | 2011-12-12 | 2012-03-07 | 南京药石药物研发有限公司 | 2-氨基嘧啶-5-硼酸的合成方法 |
ES2594078T3 (es) | 2012-10-10 | 2016-12-15 | F. Hoffmann-La Roche Ag | Proceso para preparar compuestos de tienopirimidina |
-
2014
- 2014-05-05 JP JP2016512308A patent/JP6456925B2/ja active Active
- 2014-05-05 RU RU2015148570A patent/RU2658915C2/ru active
- 2014-05-05 WO PCT/EP2014/059023 patent/WO2014180752A1/en active Application Filing
- 2014-05-05 CN CN201480025306.0A patent/CN105189519B/zh active Active
- 2014-05-05 MX MX2015015346A patent/MX361673B/es active IP Right Grant
- 2014-05-05 KR KR1020157034486A patent/KR101813775B1/ko active IP Right Grant
- 2014-05-05 CA CA2910541A patent/CA2910541C/en active Active
- 2014-05-05 EP EP14722170.9A patent/EP2994472B1/en active Active
- 2014-05-05 AR ARP140101825 patent/AR096178A1/es unknown
- 2014-05-05 US US14/269,334 patent/US9102689B2/en active Active
- 2014-05-05 BR BR112015027475-7A patent/BR112015027475B1/pt active IP Right Grant
-
2016
- 2016-02-11 HK HK16101475.4A patent/HK1213554A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
MX2015015346A (es) | 2016-03-04 |
AR096178A1 (es) | 2015-12-09 |
BR112015027475A2 (es) | 2017-08-29 |
BR112015027475B1 (pt) | 2022-08-23 |
KR101813775B1 (ko) | 2017-12-29 |
WO2014180752A1 (en) | 2014-11-13 |
CN105189519A (zh) | 2015-12-23 |
CA2910541A1 (en) | 2014-11-13 |
EP2994472A1 (en) | 2016-03-16 |
HK1213554A1 (zh) | 2016-07-08 |
US20140330008A1 (en) | 2014-11-06 |
CA2910541C (en) | 2020-07-21 |
CN105189519B (zh) | 2018-01-30 |
US9102689B2 (en) | 2015-08-11 |
JP2016522820A (ja) | 2016-08-04 |
RU2015148570A (ru) | 2017-06-13 |
KR20160004385A (ko) | 2016-01-12 |
EP2994472B1 (en) | 2017-11-22 |
JP6456925B2 (ja) | 2019-01-23 |
RU2658915C2 (ru) | 2018-06-26 |
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Legal Events
Date | Code | Title | Description |
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FG | Grant or registration |