AR096178A1 - Procedimiento para la preparacion de intermediarios de acido boronico. - Google Patents

Procedimiento para la preparacion de intermediarios de acido boronico.

Info

Publication number
AR096178A1
AR096178A1 ARP140101825A AR096178A1 AR 096178 A1 AR096178 A1 AR 096178A1 AR P140101825 A ARP140101825 A AR P140101825A AR 096178 A1 AR096178 A1 AR 096178A1
Authority
AR
Argentina
Prior art keywords
intermediaries
procedure
preparation
boronic acid
boronic
Prior art date
Application number
Other languages
English (en)
Inventor
Torsten Busch
Michael Nonnenmacher
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR096178A1 publication Critical patent/AR096178A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • C07D491/044Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/048Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
ARP140101825 2013-05-06 2014-05-05 Procedimiento para la preparacion de intermediarios de acido boronico. AR096178A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP13166587 2013-05-06

Publications (1)

Publication Number Publication Date
AR096178A1 true AR096178A1 (es) 2015-12-09

Family

ID=48227048

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140101825 AR096178A1 (es) 2013-05-06 2014-05-05 Procedimiento para la preparacion de intermediarios de acido boronico.

Country Status (12)

Country Link
US (1) US9102689B2 (es)
EP (1) EP2994472B1 (es)
JP (1) JP6456925B2 (es)
KR (1) KR101813775B1 (es)
CN (1) CN105189519B (es)
AR (1) AR096178A1 (es)
BR (1) BR112015027475B1 (es)
CA (1) CA2910541C (es)
HK (1) HK1213554A1 (es)
MX (1) MX361673B (es)
RU (1) RU2658915C2 (es)
WO (1) WO2014180752A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2801577A1 (en) * 2013-05-06 2014-11-12 Euticals S.P.A. Process for the preparation of aminoaryl- and aminoheteroaryl boronic acids and esters

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10322843A1 (de) * 2003-05-19 2004-12-16 Clariant Gmbh Verfahren zur Herstellung von Anilinboronsäuren und ihren Derivaten
NZ578162A (en) 2006-12-07 2011-12-22 Genentech Inc Phosphoinositide 3-kinase inhibitor compounds and methods of use
EP1988095B1 (de) * 2007-04-27 2016-01-27 Euticals GmbH Verfarhen zur Herstellung von Aminoaryl- bzw. heteroarylboronsaeuren und ihren Derivaten
CN102399235A (zh) * 2011-10-25 2012-04-04 江苏弘和药物研发有限公司 一种2-氨基-5-嘧啶硼酸频哪醇酯的合成方法
CN102367260A (zh) * 2011-12-12 2012-03-07 南京药石药物研发有限公司 2-氨基嘧啶-5-硼酸的合成方法
WO2014056955A1 (en) * 2012-10-10 2014-04-17 F. Hoffmann-La Roche Ag Process for making thienopyrimidine compounds

Also Published As

Publication number Publication date
JP2016522820A (ja) 2016-08-04
KR20160004385A (ko) 2016-01-12
CN105189519A (zh) 2015-12-23
EP2994472B1 (en) 2017-11-22
RU2015148570A (ru) 2017-06-13
JP6456925B2 (ja) 2019-01-23
CN105189519B (zh) 2018-01-30
RU2658915C2 (ru) 2018-06-26
CA2910541A1 (en) 2014-11-13
BR112015027475A2 (es) 2017-08-29
KR101813775B1 (ko) 2017-12-29
MX361673B (es) 2018-12-11
EP2994472A1 (en) 2016-03-16
WO2014180752A1 (en) 2014-11-13
MX2015015346A (es) 2016-03-04
US9102689B2 (en) 2015-08-11
HK1213554A1 (zh) 2016-07-08
US20140330008A1 (en) 2014-11-06
CA2910541C (en) 2020-07-21
BR112015027475B1 (pt) 2022-08-23

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