MX2014000463A - Formas de dosificacion estables de aterolane y piperaquina. - Google Patents
Formas de dosificacion estables de aterolane y piperaquina.Info
- Publication number
- MX2014000463A MX2014000463A MX2014000463A MX2014000463A MX2014000463A MX 2014000463 A MX2014000463 A MX 2014000463A MX 2014000463 A MX2014000463 A MX 2014000463A MX 2014000463 A MX2014000463 A MX 2014000463A MX 2014000463 A MX2014000463 A MX 2014000463A
- Authority
- MX
- Mexico
- Prior art keywords
- dosage form
- active compound
- piperaquine
- solid oral
- stable solid
- Prior art date
Links
- 229950006717 piperaquine Drugs 0.000 title claims abstract description 78
- UCRHFBCYFMIWHC-UHFFFAOYSA-N piperaquine Chemical compound ClC1=CC=C2C(N3CCN(CC3)CCCN3CCN(CC3)C=3C4=CC=C(C=C4N=CC=3)Cl)=CC=NC2=C1 UCRHFBCYFMIWHC-UHFFFAOYSA-N 0.000 title claims abstract description 77
- 239000002552 dosage form Substances 0.000 title claims abstract description 49
- BRJULSXZDFYSPG-MSMJXPJBSA-N CC(C)(N)NC(=O)C[C@H]1CC[C@]2(CC1)OOC1(O2)[C@H]2CC3CC(C2)C[C@H]1C3 Chemical compound CC(C)(N)NC(=O)C[C@H]1CC[C@]2(CC1)OOC1(O2)[C@H]2CC3CC(C2)C[C@H]1C3 BRJULSXZDFYSPG-MSMJXPJBSA-N 0.000 title description 2
- 229950007854 arterolane Drugs 0.000 title description 2
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13/183,119 US8664265B2 (en) | 2005-05-18 | 2011-07-14 | Stable dosage forms of spiro and dispiro 1,2,4-trioxolane antimalarials |
| IN2703DE2011 | 2011-09-19 | ||
| IN2156DE2012 | 2012-07-12 | ||
| PCT/IB2012/053614 WO2013008218A1 (en) | 2011-07-14 | 2012-07-13 | Stable dosage forms of arterolane and piperaquine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2014000463A true MX2014000463A (es) | 2014-07-09 |
Family
ID=47505579
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2014000463A MX2014000463A (es) | 2011-07-14 | 2012-07-13 | Formas de dosificacion estables de aterolane y piperaquina. |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP2731603A1 (zh) |
| JP (1) | JP2014522856A (zh) |
| KR (1) | KR20140053169A (zh) |
| CN (1) | CN103930107A (zh) |
| AP (1) | AP2014007413A0 (zh) |
| AU (1) | AU2012282077A1 (zh) |
| CA (1) | CA2850089A1 (zh) |
| EA (1) | EA201490233A8 (zh) |
| MX (1) | MX2014000463A (zh) |
| WO (1) | WO2013008218A1 (zh) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AP2015008748A0 (en) | 2013-02-28 | 2015-09-30 | Sun Pharmaceutical Ind Ltd | Stable dispersible formulation of arterolane maleate and piperaquine and process of preparation thereof |
| KR101698003B1 (ko) * | 2016-06-20 | 2017-01-19 | 여오영 | 퀴닌 염 현탁액을 포함하는 항암 치료를 위한 국소 투여용 주사제 조성물 |
| BR112020011506A2 (pt) * | 2017-12-12 | 2020-11-17 | Intervet International B.V. | composições farmacêuticas de isoxazolina implantáveis e usos das mesmas |
| TW202220645A (zh) * | 2020-08-14 | 2022-06-01 | 印度商太陽製藥工業有限公司 | 用於治療瘧疾的固定劑量組合藥物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6486199B1 (en) | 2001-06-21 | 2002-11-26 | Medicines For Malaria Venture Mmv International Centre Cointrin | Spiro and dispiro 1,2,4-trioxolane antimalarials |
| US6906205B2 (en) | 2002-06-21 | 2005-06-14 | Medicines For Malaria Venture Mmv | Spiro and dispiro 1,2,4-trioxolane antimalarials |
| US6825230B2 (en) | 2002-06-21 | 2004-11-30 | Medicines For Malaria Venture Mmv | Spiro and dispiro 1,2,4-trixolane antimalarials |
| CN101272777B (zh) * | 2005-05-18 | 2013-01-30 | 兰贝克赛实验室有限公司 | 螺和二螺1,2,4-三氧戊环抗疟药的稳定剂型 |
| AP2525A (en) * | 2006-05-17 | 2012-12-05 | Ranbaxy Lab Ltd | Antimarial therapy using a combination of synthetic artemisinin derivative and bisquinoline derivative |
-
2012
- 2012-07-13 AP AP2014007413A patent/AP2014007413A0/xx unknown
- 2012-07-13 JP JP2014519689A patent/JP2014522856A/ja active Pending
- 2012-07-13 AU AU2012282077A patent/AU2012282077A1/en not_active Abandoned
- 2012-07-13 KR KR1020147003043A patent/KR20140053169A/ko not_active Application Discontinuation
- 2012-07-13 EP EP12743776.2A patent/EP2731603A1/en not_active Withdrawn
- 2012-07-13 EA EA201490233A patent/EA201490233A8/ru unknown
- 2012-07-13 CA CA2850089A patent/CA2850089A1/en not_active Abandoned
- 2012-07-13 WO PCT/IB2012/053614 patent/WO2013008218A1/en active Application Filing
- 2012-07-13 CN CN201280044576.7A patent/CN103930107A/zh active Pending
- 2012-07-13 MX MX2014000463A patent/MX2014000463A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2731603A1 (en) | 2014-05-21 |
| JP2014522856A (ja) | 2014-09-08 |
| CA2850089A1 (en) | 2013-01-17 |
| AP2014007413A0 (en) | 2014-02-28 |
| KR20140053169A (ko) | 2014-05-07 |
| CN103930107A (zh) | 2014-07-16 |
| WO2013008218A1 (en) | 2013-01-17 |
| EA201490233A1 (ru) | 2014-07-30 |
| AU2012282077A1 (en) | 2014-01-30 |
| AP3777A (zh) | 2016-08-31 |
| EA201490233A8 (ru) | 2015-01-30 |
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