MX2012008644A - Inhibidores de cinasa de pirazolopiridinas. - Google Patents
Inhibidores de cinasa de pirazolopiridinas.Info
- Publication number
- MX2012008644A MX2012008644A MX2012008644A MX2012008644A MX2012008644A MX 2012008644 A MX2012008644 A MX 2012008644A MX 2012008644 A MX2012008644 A MX 2012008644A MX 2012008644 A MX2012008644 A MX 2012008644A MX 2012008644 A MX2012008644 A MX 2012008644A
- Authority
- MX
- Mexico
- Prior art keywords
- independently
- compound
- alkyl
- substituted
- absent
- Prior art date
Links
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Classifications
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Landscapes
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- Psychiatry (AREA)
- Emergency Medicine (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29864910P | 2010-01-27 | 2010-01-27 | |
| US41042610P | 2010-11-05 | 2010-11-05 | |
| PCT/US2011/022522 WO2011094273A1 (en) | 2010-01-27 | 2011-01-26 | Pyrazolopyridine kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2012008644A true MX2012008644A (es) | 2012-11-23 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2012008644A MX2012008644A (es) | 2010-01-27 | 2011-01-26 | Inhibidores de cinasa de pirazolopiridinas. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US9067932B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2528917B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP5769733B2 (cg-RX-API-DMAC7.html) |
| CN (1) | CN102858769A (cg-RX-API-DMAC7.html) |
| AR (1) | AR080856A1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2011209726A1 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2787315A1 (cg-RX-API-DMAC7.html) |
| MX (1) | MX2012008644A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2011094273A1 (cg-RX-API-DMAC7.html) |
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| US8569337B2 (en) | 2008-07-23 | 2013-10-29 | Vertex Pharmaceuticals Incorporated | Tri-cyclic pyrazolopyridine kinase inhibitors |
| CA2732765A1 (en) * | 2008-08-06 | 2010-02-11 | Vertex Pharmaceuticals Incorporated | Aminopyridine kinase inhibitors |
| EP2528916A1 (en) * | 2010-01-27 | 2012-12-05 | Vertex Pharmaceuticals Incorporated | Pyrazolopyridine kinase inhibitors |
| EP2582702A1 (en) * | 2010-01-27 | 2013-04-24 | Vertex Pharmaceuticals Incorporated | Pyrazolopyrimidine kinase inhibitors |
| EP3046560B1 (en) | 2013-09-18 | 2021-01-06 | EpiAxis Therapeutics Pty Ltd | Stem cell modulation ii |
| AU2015309686B2 (en) * | 2014-08-25 | 2020-05-14 | Epiaxis Therapeutics Pty Ltd | Compositions for modulating cancer stem cells and uses therefor |
| CN111587120A (zh) * | 2017-11-08 | 2020-08-25 | 艾比克斯治疗私人有限公司 | 免疫原性组合物及其用途 |
| CN118923682B (zh) * | 2024-07-22 | 2025-09-05 | 中国农业大学 | 一种化合物作为病原真菌Pmk1的抑制剂的应用 |
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| DE3827253A1 (de) | 1987-08-20 | 1989-03-02 | Sandoz Ag | Ester und amide von cyclischen carbonsaeuren und cyclischen alkoholen und aminen sowie verfahren zu deren herstellung und sie enthaltende therapeutische zusammensetzungen |
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-
2011
- 2011-01-26 MX MX2012008644A patent/MX2012008644A/es active IP Right Grant
- 2011-01-26 US US13/014,505 patent/US9067932B2/en active Active
- 2011-01-26 JP JP2012551251A patent/JP5769733B2/ja active Active
- 2011-01-26 WO PCT/US2011/022522 patent/WO2011094273A1/en not_active Ceased
- 2011-01-26 EP EP11703958.6A patent/EP2528917B1/en active Active
- 2011-01-26 CA CA2787315A patent/CA2787315A1/en not_active Abandoned
- 2011-01-26 CN CN2011800130461A patent/CN102858769A/zh active Pending
- 2011-01-26 AU AU2011209726A patent/AU2011209726A1/en not_active Abandoned
- 2011-01-27 AR ARP110100282A patent/AR080856A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP5769733B2 (ja) | 2015-08-26 |
| AU2011209726A1 (en) | 2012-08-09 |
| CA2787315A1 (en) | 2011-08-04 |
| CN102858769A (zh) | 2013-01-02 |
| EP2528917A1 (en) | 2012-12-05 |
| WO2011094273A1 (en) | 2011-08-04 |
| US9067932B2 (en) | 2015-06-30 |
| JP2013518111A (ja) | 2013-05-20 |
| AR080856A1 (es) | 2012-05-16 |
| EP2528917B1 (en) | 2016-10-19 |
| US20120071494A1 (en) | 2012-03-22 |
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