MX2011008878A - Usos de antagonistas de los receptores de nk. - Google Patents

Usos de antagonistas de los receptores de nk.

Info

Publication number
MX2011008878A
MX2011008878A MX2011008878A MX2011008878A MX2011008878A MX 2011008878 A MX2011008878 A MX 2011008878A MX 2011008878 A MX2011008878 A MX 2011008878A MX 2011008878 A MX2011008878 A MX 2011008878A MX 2011008878 A MX2011008878 A MX 2011008878A
Authority
MX
Mexico
Prior art keywords
receptor antagonists
pruritus
solvate
hydrate
substituents
Prior art date
Application number
MX2011008878A
Other languages
English (en)
Inventor
Anton Stuetz
Barbara Wolff-Winiski
Lina Williamson
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42102184&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2011008878(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2011008878A publication Critical patent/MX2011008878A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/16—Emollients or protectives, e.g. against radiation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Abstract

La invención proporciona el uso de un compuesto de la fórmula (I): (ver fórmula (I)) o de un solvato o hidrato del mismo, en donde los sustituyentes son como se definen en la descripción, y combinaciones de los mismos, para el tratamiento de prurito o de un trastorno o enfermedad dermatológica.
MX2011008878A 2009-02-24 2010-02-23 Usos de antagonistas de los receptores de nk. MX2011008878A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15497309P 2009-02-24 2009-02-24
PCT/EP2010/052273 WO2010097381A1 (en) 2009-02-24 2010-02-23 Uses of nk receptor antagonists

Publications (1)

Publication Number Publication Date
MX2011008878A true MX2011008878A (es) 2011-09-21

Family

ID=42102184

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011008878A MX2011008878A (es) 2009-02-24 2010-02-23 Usos de antagonistas de los receptores de nk.

Country Status (17)

Country Link
US (1) US20120077803A1 (es)
EP (1) EP2400953A1 (es)
JP (1) JP5425229B2 (es)
KR (1) KR20110118830A (es)
CN (1) CN102395358A (es)
AU (1) AU2010217615C1 (es)
BR (1) BRPI1008008A2 (es)
CA (1) CA2753330A1 (es)
CL (1) CL2011002045A1 (es)
EA (1) EA201101207A1 (es)
IL (1) IL214731A0 (es)
MA (1) MA33059B1 (es)
MX (1) MX2011008878A (es)
SG (1) SG173758A1 (es)
TN (1) TN2011000428A1 (es)
TW (1) TW201034674A (es)
WO (1) WO2010097381A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2906219T3 (pl) * 2012-10-11 2020-02-28 Nerre Therapeutics Limited Orwepitant do leczenia przewlekłego świądu
US20140179727A1 (en) 2012-12-14 2014-06-26 Trevi Therapeutics, Inc. Methods for treating pruritus
US8987289B2 (en) * 2012-12-14 2015-03-24 Trevi Therapeutics, Inc. Methods for treating pruritus
US8906951B1 (en) 2013-06-24 2014-12-09 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
US9198898B2 (en) 2013-06-24 2015-12-01 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
JP2019519592A (ja) * 2016-06-29 2019-07-11 メンロ セラピューティクス インコーポレイテッド 様々な掻痒状態を処置するためのニューロキニン−１アンタゴニストの使用
MX2021000908A (es) 2018-07-23 2021-06-08 Trevi Therapeutics Inc Tratamiento de la tos cronica, la dificultad respiratoria y la disnea.

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2728166A1 (fr) * 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2740040B1 (fr) * 1995-10-23 1997-12-05 Oreal Utilisation d'au moins un agoniste beta-adrenergique en tant qu'antagoniste de substance p
DE19541283A1 (de) * 1995-11-06 1997-05-07 Boehringer Ingelheim Kg Neue Aminosäurederivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
MY132550A (en) * 1996-08-22 2007-10-31 Novartis Ag Acylaminoalkenylene-amide derivatives as nk1 and nk2 antogonists
JP3793612B2 (ja) * 1996-11-28 2006-07-05 花王株式会社 皮膚外用剤
US20040058914A1 (en) * 2000-12-22 2004-03-25 Takayuki Doi Combination drugs
JP2003238986A (ja) * 2002-02-22 2003-08-27 Shiseido Co Ltd サブスタンスｐ増加抑制剤
ITFI20030113A1 (it) * 2003-04-24 2004-10-25 Menarini Ricerche Spa Composti lineari nk-2 antagonisti con caratteristiche basiche e formulazioni che li contengono.
JO2630B1 (en) * 2006-04-13 2012-06-17 نوفارتيس ايه جي Organic compounds
MY177591A (en) * 2006-10-16 2020-09-22 Lion Corp Nk1 receptor antagonist composition
EP1938804A1 (en) * 2006-12-22 2008-07-02 Novartis AG Pharmaceutical formulation comprising neurokinin antagonist
WO2009000038A1 (en) * 2007-06-28 2008-12-31 Cnsbio Pty Ltd Combination methods and compositions for treatment of neuropathic pain

Also Published As

Publication number Publication date
JP2012518622A (ja) 2012-08-16
KR20110118830A (ko) 2011-11-01
CL2011002045A1 (es) 2012-01-13
SG173758A1 (en) 2011-09-29
BRPI1008008A2 (pt) 2016-02-23
IL214731A0 (en) 2011-11-30
CN102395358A (zh) 2012-03-28
TN2011000428A1 (en) 2013-03-27
EA201101207A1 (ru) 2012-04-30
EP2400953A1 (en) 2012-01-04
CA2753330A1 (en) 2010-09-02
WO2010097381A1 (en) 2010-09-02
AU2010217615C1 (en) 2013-05-23
TW201034674A (en) 2010-10-01
JP5425229B2 (ja) 2014-02-26
US20120077803A1 (en) 2012-03-29
AU2010217615A1 (en) 2011-09-08
MA33059B1 (fr) 2012-02-01

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