BRPI1008008A2 - usos de antagonistas do receptor de nk - Google Patents

usos de antagonistas do receptor de nk

Info

Publication number
BRPI1008008A2
BRPI1008008A2 BRPI1008008A BRPI1008008A BRPI1008008A2 BR PI1008008 A2 BRPI1008008 A2 BR PI1008008A2 BR PI1008008 A BRPI1008008 A BR PI1008008A BR PI1008008 A BRPI1008008 A BR PI1008008A BR PI1008008 A2 BRPI1008008 A2 BR PI1008008A2
Authority
BR
Brazil
Prior art keywords
receptor antagonists
antagonists
receptor
Prior art date
Application number
BRPI1008008A
Other languages
English (en)
Inventor
Anton Stuetz
Barbara Wolff-Winiski
Lina Williamson
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42102184&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI1008008(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BRPI1008008A2 publication Critical patent/BRPI1008008A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/16Emollients or protectives, e.g. against radiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BRPI1008008A 2009-02-24 2010-02-23 usos de antagonistas do receptor de nk BRPI1008008A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15497309P 2009-02-24 2009-02-24
PCT/EP2010/052273 WO2010097381A1 (en) 2009-02-24 2010-02-23 Uses of nk receptor antagonists

Publications (1)

Publication Number Publication Date
BRPI1008008A2 true BRPI1008008A2 (pt) 2016-02-23

Family

ID=42102184

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1008008A BRPI1008008A2 (pt) 2009-02-24 2010-02-23 usos de antagonistas do receptor de nk

Country Status (17)

Country Link
US (1) US20120077803A1 (pt)
EP (1) EP2400953A1 (pt)
JP (1) JP5425229B2 (pt)
KR (1) KR20110118830A (pt)
CN (1) CN102395358A (pt)
AU (1) AU2010217615C1 (pt)
BR (1) BRPI1008008A2 (pt)
CA (1) CA2753330A1 (pt)
CL (1) CL2011002045A1 (pt)
EA (1) EA201101207A1 (pt)
IL (1) IL214731A0 (pt)
MA (1) MA33059B1 (pt)
MX (1) MX2011008878A (pt)
SG (1) SG173758A1 (pt)
TN (1) TN2011000428A1 (pt)
TW (1) TW201034674A (pt)
WO (1) WO2010097381A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9603849B2 (en) * 2012-10-11 2017-03-28 Nerre Therapeutics Limited Uses of orvepitant
US20140179727A1 (en) 2012-12-14 2014-06-26 Trevi Therapeutics, Inc. Methods for treating pruritus
US8987289B2 (en) * 2012-12-14 2015-03-24 Trevi Therapeutics, Inc. Methods for treating pruritus
US9198898B2 (en) 2013-06-24 2015-12-01 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
US8906951B1 (en) 2013-06-24 2014-12-09 Tigercat Pharma, Inc. Use of NK-1 receptor antagonists in pruritus
CN109640981A (zh) * 2016-06-29 2019-04-16 曼隆治疗公司 神经激肽-1拮抗剂用于治疗多种瘙痒病症的用途
SG11202100580UA (en) 2018-07-23 2021-02-25 Trevi Therapeutics Inc Treatment of chronic cough, breathlessness and dyspnea

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2728166A1 (fr) * 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2740040B1 (fr) * 1995-10-23 1997-12-05 Oreal Utilisation d'au moins un agoniste beta-adrenergique en tant qu'antagoniste de substance p
DE19541283A1 (de) * 1995-11-06 1997-05-07 Boehringer Ingelheim Kg Neue Aminosäurederivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
MY132550A (en) * 1996-08-22 2007-10-31 Novartis Ag Acylaminoalkenylene-amide derivatives as nk1 and nk2 antogonists
JP3793612B2 (ja) * 1996-11-28 2006-07-05 花王株式会社 皮膚外用剤
CA2432543A1 (en) * 2000-12-22 2002-07-04 Takeda Chemical Industries, Ltd. Combination drugs
JP2003238986A (ja) * 2002-02-22 2003-08-27 Shiseido Co Ltd サブスタンスp増加抑制剤
ITFI20030113A1 (it) * 2003-04-24 2004-10-25 Menarini Ricerche Spa Composti lineari nk-2 antagonisti con caratteristiche basiche e formulazioni che li contengono.
JO2630B1 (en) * 2006-04-13 2012-06-17 نوفارتيس ايه جي Organic compounds
CN101600724B (zh) * 2006-10-16 2013-03-13 狮王株式会社 Nk1受体拮抗剂组合物
EP1938804A1 (en) * 2006-12-22 2008-07-02 Novartis AG Pharmaceutical formulation comprising neurokinin antagonist
WO2009000038A1 (en) * 2007-06-28 2008-12-31 Cnsbio Pty Ltd Combination methods and compositions for treatment of neuropathic pain

Also Published As

Publication number Publication date
CL2011002045A1 (es) 2012-01-13
TN2011000428A1 (en) 2013-03-27
AU2010217615C1 (en) 2013-05-23
SG173758A1 (en) 2011-09-29
AU2010217615A1 (en) 2011-09-08
EA201101207A1 (ru) 2012-04-30
JP2012518622A (ja) 2012-08-16
EP2400953A1 (en) 2012-01-04
US20120077803A1 (en) 2012-03-29
KR20110118830A (ko) 2011-11-01
CA2753330A1 (en) 2010-09-02
JP5425229B2 (ja) 2014-02-26
MX2011008878A (es) 2011-09-21
MA33059B1 (fr) 2012-02-01
CN102395358A (zh) 2012-03-28
WO2010097381A1 (en) 2010-09-02
TW201034674A (en) 2010-10-01
IL214731A0 (en) 2011-11-30

Similar Documents

Publication Publication Date Title
FR22C1044I1 (fr) Antagonistes du recepteur cgrp
CY2023022I1 (el) Ανταγωνιστες υποδοχεων cgrp αζαϊνδανιου καρβοξαμιδιου πιπεριδινονης
BR112012015873A2 (pt) antagonistas de receptores ccr2 e usos dos mesmos
BRPI0919844A2 (pt) compostos de azaindazol como antagonistas do receptor ccr1
PL2927224T3 (pl) Antagoniści receptora
BRPI0910118A2 (pt) antagonistas de receptores do glucagon
EP2411001A4 (en) P2X3 RECEPTOR ANTAGONISTS FOR PAIN TREATMENT
BR112014001030A2 (pt) anticorpos anti-receptor alfa de folato e usos destes
BRPI0913930A2 (pt) antagonistas de receptores de prostaglandinas d2
BR112012003263A2 (pt) formulações intravenosas de antagonistas de neuroquinina-1
EP2410857A4 (en) ANTAGONISTS OF THE P2X3 RECEPTOR FOR THE TREATMENT OF PAIN
DK2443104T3 (da) Disubstituerede phthalazin-hedgehog-sti-antagonister
DK2501703T3 (da) Spiropiperidinforbindelser som orl-1-receptorantagonister
SMT201600078B (it) Antagonista del recettore per cgrp
BRPI0717937A2 (pt) Compostos de pirazona como antagonistas do receptor mineralocorticóide
EP2427430A4 (en) 5-OXO-ETE RECEPTOR ANTAGONIST COMPOUNDS
EP2410858A4 (en) P2X3 RECEPTOR ANTAGONISTS FOR PAIN TREATMENT
DK2252581T3 (da) Kappa-selektiv opioidreceptorantagonist
BRPI1008008A2 (pt) usos de antagonistas do receptor de nk
BR112012003976A2 (pt) antagonistas de receptor glyt1 carbocíclico
BRPI0720078A2 (pt) 2-aminoquinolinas como antagonistas de receptores de 5-ht(5a)
BRPI0915834A2 (pt) 6-(1-piperazinil)-piridazinas substituídas como antagonistas do receptor de 5-ht6
BRPI1013617A2 (pt) derivados de piperidina como antagonistas de receptor de nk3
EP2451281A4 (en) ANTAGONISTS OF OREXIN RECEPTORS BASED ON TETRAHYDRONAPHTHYRIDINE
BRPI1014668A2 (pt) antagonistas ccr3 de arilsulfonamida

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2370 DE 07-06-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.