MX2010012803A - Tieno pirimidinonas sustituidas con hidroxi como antagonistas del receptor-1 de la hormona concentradora de melanina. - Google Patents

Tieno pirimidinonas sustituidas con hidroxi como antagonistas del receptor-1 de la hormona concentradora de melanina.

Info

Publication number
MX2010012803A
MX2010012803A MX2010012803A MX2010012803A MX2010012803A MX 2010012803 A MX2010012803 A MX 2010012803A MX 2010012803 A MX2010012803 A MX 2010012803A MX 2010012803 A MX2010012803 A MX 2010012803A MX 2010012803 A MX2010012803 A MX 2010012803A
Authority
MX
Mexico
Prior art keywords
agents
compounds
antagonists
receptor
inhibitors
Prior art date
Application number
MX2010012803A
Other languages
English (en)
Spanish (es)
Inventor
Ramesh N Patel
William N Washburn
Pratik Devasthale
Jeffrey A Robl
Animesh Goswami
Zhiwei Guo
Saleem Ahmad
Original Assignee
Squibb Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb Bristol Myers Co filed Critical Squibb Bristol Myers Co
Publication of MX2010012803A publication Critical patent/MX2010012803A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
MX2010012803A 2008-05-29 2009-05-28 Tieno pirimidinonas sustituidas con hidroxi como antagonistas del receptor-1 de la hormona concentradora de melanina. MX2010012803A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5694908P 2008-05-29 2008-05-29
PCT/US2009/045452 WO2009146365A1 (en) 2008-05-29 2009-05-28 Hydroxy substituted thieno pyrimidinones as melanin concentrating hormone receptor-1 antagonists

Publications (1)

Publication Number Publication Date
MX2010012803A true MX2010012803A (es) 2010-12-07

Family

ID=41017166

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010012803A MX2010012803A (es) 2008-05-29 2009-05-28 Tieno pirimidinonas sustituidas con hidroxi como antagonistas del receptor-1 de la hormona concentradora de melanina.

Country Status (17)

Country Link
US (1) US7989433B2 (enExample)
EP (1) EP2310394A1 (enExample)
JP (1) JP2011521962A (enExample)
KR (1) KR20110021988A (enExample)
CN (1) CN102099360A (enExample)
AR (1) AR075260A1 (enExample)
AU (1) AU2009251331A1 (enExample)
BR (1) BRPI0913197A2 (enExample)
CA (1) CA2726264A1 (enExample)
CO (1) CO6280492A2 (enExample)
EA (1) EA201001882A1 (enExample)
IL (1) IL209354A0 (enExample)
MX (1) MX2010012803A (enExample)
PE (1) PE20091928A1 (enExample)
TW (1) TW201000487A (enExample)
WO (1) WO2009146365A1 (enExample)
ZA (1) ZA201008451B (enExample)

Families Citing this family (9)

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EP2788088B1 (en) 2011-12-06 2019-06-19 Unilever Plc. Skin anti-ageing composition
IL225900A0 (en) * 2013-04-22 2014-03-31 Perrigo Api Ltd A process for the preparation of nicotine that includes the enzymatic reduction of 4-(methylamino)-1-(3-pyridinyl)-1-butanone
EP2921856B1 (en) * 2014-03-18 2016-09-14 Serum Institute Of India Private Limited A quantitative assay for 4-pyrrolidinopyridine (4-ppy) in polysaccharide-protein conjugate vaccines
BR112017013758B1 (pt) * 2014-12-30 2021-11-23 Dow Agrosciences Llc Compostos de picolinamida com atividade fungicida
CA2972401C (en) 2014-12-30 2023-09-05 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
EP4151210A3 (en) * 2020-01-10 2023-06-14 Harmony Biosciences, LLC Pyridine-carboline derivatives as mchr1 antagonists for use in therapy
HUP2200222A1 (hu) 2022-06-17 2023-12-28 Richter Gedeon Nyrt MCHR1 antagonisták a Prader-Willi szindróma kezelésére

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Also Published As

Publication number Publication date
AR075260A1 (es) 2011-03-23
AU2009251331A1 (en) 2009-12-03
IL209354A0 (en) 2011-01-31
JP2011521962A (ja) 2011-07-28
EA201001882A1 (ru) 2011-06-30
CO6280492A2 (es) 2011-05-20
US20090298794A1 (en) 2009-12-03
BRPI0913197A2 (pt) 2016-01-12
WO2009146365A1 (en) 2009-12-03
ZA201008451B (en) 2012-04-25
CA2726264A1 (en) 2009-12-03
US7989433B2 (en) 2011-08-02
PE20091928A1 (es) 2009-12-31
CN102099360A (zh) 2011-06-15
KR20110021988A (ko) 2011-03-04
EP2310394A1 (en) 2011-04-20
TW201000487A (en) 2010-01-01

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