MX2007008334A - Derivados aminofenilo como moduladores de receptor de androgeno selectivos. - Google Patents
Derivados aminofenilo como moduladores de receptor de androgeno selectivos.Info
- Publication number
- MX2007008334A MX2007008334A MX2007008334A MX2007008334A MX2007008334A MX 2007008334 A MX2007008334 A MX 2007008334A MX 2007008334 A MX2007008334 A MX 2007008334A MX 2007008334 A MX2007008334 A MX 2007008334A MX 2007008334 A MX2007008334 A MX 2007008334A
- Authority
- MX
- Mexico
- Prior art keywords
- substituted
- group
- endo
- alkyl
- chloro
- Prior art date
Links
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- PBMFSQRYOILNGV-UHFFFAOYSA-N pyridazine Chemical compound C1=CC=NN=C1 PBMFSQRYOILNGV-UHFFFAOYSA-N 0.000 description 1
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- FKHIFSZMMVMEQY-UHFFFAOYSA-N talc Chemical compound [Mg+2].[O-][Si]([O-])=O FKHIFSZMMVMEQY-UHFFFAOYSA-N 0.000 description 1
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- ITMCEJHCFYSIIV-UHFFFAOYSA-M triflate Chemical compound [O-]S(=O)(=O)C(F)(F)F ITMCEJHCFYSIIV-UHFFFAOYSA-M 0.000 description 1
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- AHZJKOKFZJYCLG-UHFFFAOYSA-K trifluoromethanesulfonate;ytterbium(3+) Chemical compound [Yb+3].[O-]S(=O)(=O)C(F)(F)F.[O-]S(=O)(=O)C(F)(F)F.[O-]S(=O)(=O)C(F)(F)F AHZJKOKFZJYCLG-UHFFFAOYSA-K 0.000 description 1
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Classifications
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- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64284105P | 2005-01-10 | 2005-01-10 | |
| PCT/US2006/000733 WO2006076317A2 (en) | 2005-01-10 | 2006-01-09 | Aminophenyl derivatives as selective androgen receptor modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007008334A true MX2007008334A (es) | 2007-09-11 |
Family
ID=36591321
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007008334A MX2007008334A (es) | 2005-01-10 | 2006-01-09 | Derivados aminofenilo como moduladores de receptor de androgeno selectivos. |
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| Country | Link |
|---|---|
| US (2) | US7585877B2 (enExample) |
| EP (1) | EP1836202B1 (enExample) |
| JP (1) | JP5203712B2 (enExample) |
| KR (1) | KR20070112775A (enExample) |
| CN (1) | CN101119993B (enExample) |
| AU (1) | AU2006205066B2 (enExample) |
| CA (1) | CA2594340C (enExample) |
| MX (1) | MX2007008334A (enExample) |
| NZ (1) | NZ555974A (enExample) |
| RU (1) | RU2007130558A (enExample) |
| WO (1) | WO2006076317A2 (enExample) |
| ZA (1) | ZA200705458B (enExample) |
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| US20070004679A1 (en) * | 2004-05-17 | 2007-01-04 | Nathalie Schlienger | Androgen receptor modulators and methods of treating disease using the same |
| US20060173037A1 (en) * | 2005-01-10 | 2006-08-03 | Nathalie Schlienger | Aminophenyl derivatives as selective androgen receptor modulators |
| NZ555974A (en) | 2005-01-10 | 2010-11-26 | Acadia Pharm Inc | Aminophenyl derivatives as selective androgen receptor modulators |
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-
2006
- 2006-01-09 NZ NZ555974A patent/NZ555974A/en not_active IP Right Cessation
- 2006-01-09 WO PCT/US2006/000733 patent/WO2006076317A2/en not_active Ceased
- 2006-01-09 US US11/329,267 patent/US7585877B2/en not_active Expired - Fee Related
- 2006-01-09 JP JP2007550547A patent/JP5203712B2/ja not_active Expired - Fee Related
- 2006-01-09 CA CA2594340A patent/CA2594340C/en not_active Expired - Fee Related
- 2006-01-09 ZA ZA200705458A patent/ZA200705458B/xx unknown
- 2006-01-09 RU RU2007130558/04A patent/RU2007130558A/ru not_active Application Discontinuation
- 2006-01-09 EP EP06733660.2A patent/EP1836202B1/en not_active Expired - Lifetime
- 2006-01-09 MX MX2007008334A patent/MX2007008334A/es not_active Application Discontinuation
- 2006-01-09 AU AU2006205066A patent/AU2006205066B2/en not_active Ceased
- 2006-01-09 KR KR1020077018305A patent/KR20070112775A/ko not_active Withdrawn
- 2006-01-09 CN CN200680002003.2A patent/CN101119993B/zh not_active Expired - Fee Related
-
2009
- 2009-06-30 US US12/495,514 patent/US20090270449A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20070112775A (ko) | 2007-11-27 |
| WO2006076317A2 (en) | 2006-07-20 |
| US7585877B2 (en) | 2009-09-08 |
| NZ555974A (en) | 2010-11-26 |
| US20060160845A1 (en) | 2006-07-20 |
| AU2006205066A1 (en) | 2006-07-20 |
| JP2008526888A (ja) | 2008-07-24 |
| AU2006205066B2 (en) | 2012-05-17 |
| ZA200705458B (en) | 2008-12-31 |
| EP1836202A2 (en) | 2007-09-26 |
| CA2594340A1 (en) | 2006-07-20 |
| CA2594340C (en) | 2015-11-10 |
| EP1836202B1 (en) | 2016-12-21 |
| US20090270449A1 (en) | 2009-10-29 |
| RU2007130558A (ru) | 2009-02-20 |
| CN101119993B (zh) | 2015-03-04 |
| WO2006076317A9 (en) | 2007-09-27 |
| JP5203712B2 (ja) | 2013-06-05 |
| CN101119993A (zh) | 2008-02-06 |
| WO2006076317A3 (en) | 2006-11-23 |
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