MX18736A - Inhibidores retrovirales de proteasa y procedimiento para su preparacion. - Google Patents

Inhibidores retrovirales de proteasa y procedimiento para su preparacion.

Info

Publication number
MX18736A
MX18736A MX1873689A MX1873689A MX18736A MX 18736 A MX18736 A MX 18736A MX 1873689 A MX1873689 A MX 1873689A MX 1873689 A MX1873689 A MX 1873689A MX 18736 A MX18736 A MX 18736A
Authority
MX
Mexico
Prior art keywords
procedure
preparation
protease inhibitors
retroviral protease
retroviral
Prior art date
Application number
MX1873689A
Other languages
English (en)
Inventor
Alexander Fassler
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of MX18736A publication Critical patent/MX18736A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0207Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)4-C(=0), e.g. 'isosters', replacing two amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
MX1873689A 1988-12-15 1989-12-15 Inhibidores retrovirales de proteasa y procedimiento para su preparacion. MX18736A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH464088 1988-12-15

Publications (1)

Publication Number Publication Date
MX18736A true MX18736A (es) 1994-02-28

Family

ID=4279903

Family Applications (1)

Application Number Title Priority Date Filing Date
MX1873689A MX18736A (es) 1988-12-15 1989-12-15 Inhibidores retrovirales de proteasa y procedimiento para su preparacion.

Country Status (15)

Country Link
EP (1) EP0374098A3 (es)
JP (1) JPH02300199A (es)
KR (1) KR900009692A (es)
AU (1) AU626361B2 (es)
CA (1) CA2005340A1 (es)
DD (1) DD290894A5 (es)
DK (1) DK633289A (es)
FI (1) FI895962A0 (es)
HU (1) HUT52525A (es)
IL (1) IL92672A0 (es)
MX (1) MX18736A (es)
NO (1) NO895026L (es)
NZ (1) NZ231750A (es)
PT (1) PT92554A (es)
ZA (1) ZA899558B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2010531A1 (en) * 1989-03-06 1990-09-06 Werner Neidhart Amino acid derivatives
IL98260A0 (en) * 1990-06-01 1992-06-21 Ciba Geigy Ag Hiv protease inhibiting oligopeptides,process for their preparation and pharmaceutical compositions containing them
DE4126485A1 (de) * 1991-08-10 1993-02-11 Bayer Ag Trifluormethyl-haltige pseudopeptide
US5643878A (en) * 1991-09-12 1997-07-01 Ciba-Geigy Corporation 5-amino-4-hydroxyhexanoic acid derivatives
RU2126794C1 (ru) 1992-03-11 1999-02-27 Нархекс Лимитед Аминопроизводные оксо- или гидроксизамещенных гидразинов, способ их получения и фармацевтические композиции для ингибирования ретровирусной протеазы
US5888992A (en) 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
US6071895A (en) 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
MXPA93002392A (es) 1992-03-11 2005-02-04 Narhex Ltd Derivados amino de hidrocarburos-oxo e hidroxi-substituidos.
TW217410B (es) * 1992-04-01 1993-12-11 Ciba Geigy
US5559256A (en) * 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
EP0626178A1 (de) * 1993-05-17 1994-11-30 Ciba-Geigy Ag Verwendung von Hemmstoffen von HIV-Aspartatproteasen zur Bekämpfung von Tumorerkrankungen
DE4332395A1 (de) * 1993-09-23 1995-04-13 Horst Dr Lindhofer Inhibitoren zur Hemmung der zymogenähnlichen Freispaltung der HIV-1 Protease
PL335484A1 (en) * 1997-02-26 2000-04-25 Pfizer Derivatives of heteroarylhexamide, their production and application as selective inhibitors of mip-1a being assimilated by its ccr1 receptor
US6395897B1 (en) 1999-03-02 2002-05-28 Boehringer Ingelheim Pharmaceuticals, Inc. Nitrile compounds useful as reversible inhibitors of #9 cathepsin 5
US6420364B1 (en) 1999-09-13 2002-07-16 Boehringer Ingelheim Pharmaceuticals, Inc. Compound useful as reversible inhibitors of cysteine proteases
EP1498417A1 (en) * 2000-02-04 2005-01-19 Pfizer Products Inc. Heterocyclic amide derivatives
CZ20022542A3 (cs) * 2000-02-04 2003-08-13 Pfizer Products Inc. Heterocyklické amidové deriváty

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4727060A (en) * 1984-11-13 1988-02-23 Ciba-Geigy Corporation Novel 5-amino-4-hydroxyvaleryl derivatives
WO1988003022A1 (en) * 1986-10-31 1988-05-05 Pfizer Inc. Relatively low molecular weight polypeptides as renin inhibitors

Also Published As

Publication number Publication date
AU626361B2 (en) 1992-07-30
ZA899558B (en) 1990-08-29
NZ231750A (en) 1992-08-26
DD290894A5 (de) 1991-06-13
EP0374098A3 (de) 1991-05-02
DK633289D0 (da) 1989-12-14
AU4678489A (en) 1990-06-21
KR900009692A (ko) 1990-07-05
PT92554A (pt) 1990-06-29
CA2005340A1 (en) 1990-06-15
JPH02300199A (ja) 1990-12-12
IL92672A0 (en) 1990-09-17
FI895962A0 (fi) 1989-12-13
EP0374098A2 (de) 1990-06-20
HUT52525A (en) 1990-07-28
DK633289A (da) 1990-06-16
NO895026L (no) 1990-06-18
NO895026D0 (no) 1989-12-14

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