MC1333A1 - Derives de quinazoline - Google Patents

Derives de quinazoline

Info

Publication number
MC1333A1
MC1333A1 MC801458A MC1458A MC1333A1 MC 1333 A1 MC1333 A1 MC 1333A1 MC 801458 A MC801458 A MC 801458A MC 1458 A MC1458 A MC 1458A MC 1333 A1 MC1333 A1 MC 1333A1
Authority
MC
Monaco
Prior art keywords
quinazoline derivatives
quinazoline
derivatives
Prior art date
Application number
MC801458A
Other languages
English (en)
French (fr)
Inventor
W Nason
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1333A1 publication Critical patent/MC1333A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/90Oxygen atoms with acyclic radicals attached in position 2 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MC801458A 1979-07-09 1980-07-07 Derives de quinazoline MC1333A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5572879A 1979-07-09 1979-07-09
US06/142,903 US4281127A (en) 1979-07-09 1980-04-23 Trans-3-(4-oxo-4H-quinazolin-3-yl)-2-propenoic acid derivatives

Publications (1)

Publication Number Publication Date
MC1333A1 true MC1333A1 (fr) 1981-04-21

Family

ID=26734565

Family Applications (1)

Application Number Title Priority Date Filing Date
MC801458A MC1333A1 (fr) 1979-07-09 1980-07-07 Derives de quinazoline

Country Status (21)

Country Link
US (1) US4281127A (no)
EP (1) EP0023594B1 (no)
AR (1) AR226854A1 (no)
AU (1) AU521014B2 (no)
CA (1) CA1134825A (no)
DE (1) DE3067830D1 (no)
DK (1) DK150483C (no)
ES (2) ES493203A0 (no)
FI (1) FI74279C (no)
GR (1) GR65952B (no)
HK (1) HK52187A (no)
HU (1) HU184797B (no)
IE (1) IE49938B1 (no)
IL (1) IL60514A (no)
MC (1) MC1333A1 (no)
NO (1) NO154426C (no)
NZ (1) NZ194259A (no)
PH (1) PH16413A (no)
PT (1) PT71512B (no)
SG (1) SG20887G (no)
YU (1) YU42348B (no)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4599336A (en) * 1983-08-08 1986-07-08 Hoffmann-La Roche Inc. Derivatives of (E)-3-(4-oxo-4H-quinazolin-3-yl)-2-propenamide
GB9404485D0 (en) * 1994-03-09 1994-04-20 Cancer Res Campaign Tech Benzamide analogues
US6706721B1 (en) * 1998-04-29 2004-03-16 Osi Pharmaceuticals, Inc. N-(3-ethynylphenylamino)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine mesylate anhydrate and monohydrate
US6545004B1 (en) 1999-10-27 2003-04-08 Cytokinetics, Inc. Methods and compositions utilizing quinazolinones
US7230000B1 (en) * 1999-10-27 2007-06-12 Cytokinetics, Incorporated Methods and compositions utilizing quinazolinones
US7087613B2 (en) * 1999-11-11 2006-08-08 Osi Pharmaceuticals, Inc. Treating abnormal cell growth with a stable polymorph of N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine hydrochloride
UA74803C2 (uk) 1999-11-11 2006-02-15 Осі Фармасьютікалз, Інк. Стійкий поліморф гідрохлориду n-(3-етинілфеніл)-6,7-біс(2-метоксіетокси)-4-хіназолінаміну, спосіб його одержання (варіанти) та фармацевтичне застосування
AU2003213092A1 (en) * 2002-02-15 2003-09-09 Smithkline Beecham Corporation Syntheses of quinazolinones
BR0309892A2 (pt) * 2002-05-09 2011-04-05 Cytokinetics Inc composto, composição, métodos para modular a atividade da cinesina de ksp, para inibir a ksp, e para o tratamento de uma doença proliferativa celular, e, uso de um composto
JP2005530785A (ja) * 2002-05-09 2005-10-13 サイトキネティクス・インコーポレーテッド 化合物、組成物、及び方法
US7038048B2 (en) * 2002-05-23 2006-05-02 Cytokinetics, Inc. 3H-pyridopyrimidin-4-one compounds, compositions, and methods of their use
EP1556357A4 (en) * 2002-06-14 2006-09-13 Cytokinetics Inc COMPOUNDS, COMPOSITIONS AND METHODS
AU2003256805A1 (en) * 2002-07-23 2004-02-09 Cytokinetics, Inc. Compounds compositions and methods
US20040048853A1 (en) * 2002-08-21 2004-03-11 Gustave Bergnes Compounds, compositions, and methods
EP1558083A4 (en) * 2002-09-30 2008-04-16 Cytokinetics Inc COMPOUNDS, COMPOSITIONS AND METHODS
JP2007510652A (ja) * 2003-11-03 2007-04-26 サイトキネティクス・インコーポレーテッド ピリミジン−4−オン化合物、組成物、および方法
EP1680420A4 (en) * 2003-11-07 2008-09-24 Cytokinetics Inc COMPOUNDS, COMPOSITIONS AND METHODS
JP2007513154A (ja) * 2003-12-08 2007-05-24 サイトキネティクス・インコーポレーテッド 化合物、組成物及び方法
UY29198A1 (es) * 2004-11-09 2006-05-31 Cancer Rec Tech Ltd Derivados sustituidos de quinazolinona y derivados sustituidos de quinazolina-2, 4-diona, composiciones conteniéndolos, procedimientos de preparación y aplicaciones

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2786055A (en) * 1955-02-10 1957-03-19 Mallinckrodt Chemical Works Carboxyalkyl-iodoquinazolones
US3517005A (en) * 1967-10-26 1970-06-23 Pfizer & Co C Certain 2- and 4-substituted quinazolines
US3696102A (en) * 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones

Also Published As

Publication number Publication date
NO154426C (no) 1986-09-17
FI74279B (fi) 1987-09-30
PT71512A (en) 1980-08-01
IE801412L (en) 1981-01-09
FI74279C (fi) 1988-01-11
DK150483B (da) 1987-03-09
ES8106302A1 (es) 1981-05-16
CA1134825A (en) 1982-11-02
NZ194259A (en) 1984-09-28
AU6024480A (en) 1981-03-12
IL60514A0 (en) 1980-09-16
NO802056L (no) 1981-01-12
IL60514A (en) 1985-03-31
DE3067830D1 (en) 1984-06-20
EP0023594B1 (de) 1984-05-16
YU176680A (en) 1984-12-31
PT71512B (en) 1981-12-11
ES499035A0 (es) 1982-09-16
AR226854A1 (es) 1982-08-31
DK294780A (da) 1981-01-10
US4281127A (en) 1981-07-28
IE49938B1 (en) 1986-01-08
ES8207155A1 (es) 1982-09-16
SG20887G (en) 1988-09-16
YU42348B (en) 1988-08-31
DK150483C (da) 1987-11-09
FI802195A (fi) 1981-01-10
GR65952B (no) 1981-01-09
HU184797B (en) 1984-10-29
ES493203A0 (es) 1981-05-16
AU521014B2 (en) 1982-03-11
PH16413A (en) 1983-09-29
NO154426B (no) 1986-06-09
EP0023594A1 (de) 1981-02-11
HK52187A (en) 1987-07-17

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