MA53927A - Composition pharmaceutique pour une administration par voie orale comprenant un dérivé d'aminopyrimidine ou son sel - Google Patents

Composition pharmaceutique pour une administration par voie orale comprenant un dérivé d'aminopyrimidine ou son sel

Info

Publication number
MA53927A
MA53927A MA053927A MA53927A MA53927A MA 53927 A MA53927 A MA 53927A MA 053927 A MA053927 A MA 053927A MA 53927 A MA53927 A MA 53927A MA 53927 A MA53927 A MA 53927A
Authority
MA
Morocco
Prior art keywords
salt
pharmaceutical composition
oral administration
aminopyrimidine derivative
aminopyrimidine
Prior art date
Application number
MA053927A
Other languages
English (en)
Other versions
MA53927B1 (fr
Inventor
Seongkyu Kim
Soo-Won Kim
Deokkyu Lee
Yoong-Sik Park
Jun-Mo Yang
Original Assignee
Yuhan Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yuhan Corp filed Critical Yuhan Corp
Publication of MA53927A publication Critical patent/MA53927A/fr
Publication of MA53927B1 publication Critical patent/MA53927B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
MA53927A 2018-10-18 2019-10-17 Composition pharmaceutique pour une administration par voie orale comprenant un dérivé d'aminopyrimidine ou son sel MA53927B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020180124171A KR20200043618A (ko) 2018-10-18 2018-10-18 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구투여용 약학 조성물
PCT/IB2019/058862 WO2020079637A1 (fr) 2018-10-18 2019-10-17 Composition pharmaceutique pour une administration par voie orale comprenant un dérivé d'aminopyrimidine ou son sel

Publications (2)

Publication Number Publication Date
MA53927A true MA53927A (fr) 2021-09-15
MA53927B1 MA53927B1 (fr) 2023-12-29

Family

ID=70282933

Family Applications (1)

Application Number Title Priority Date Filing Date
MA53927A MA53927B1 (fr) 2018-10-18 2019-10-17 Composition pharmaceutique pour une administration par voie orale comprenant un dérivé d'aminopyrimidine ou son sel

Country Status (27)

Country Link
US (1) US20210322428A1 (fr)
EP (2) EP4306113A3 (fr)
JP (2) JP7369769B2 (fr)
KR (2) KR20200043618A (fr)
CN (1) CN113015521A (fr)
AR (1) AR117655A1 (fr)
AU (1) AU2019360446A1 (fr)
BR (1) BR112021007061A2 (fr)
CA (1) CA3116652A1 (fr)
DK (1) DK3866767T3 (fr)
EA (1) EA202191061A1 (fr)
ES (1) ES2968966T3 (fr)
FI (1) FI3866767T3 (fr)
HR (1) HRP20231670T1 (fr)
IL (1) IL282163A (fr)
LT (1) LT3866767T (fr)
MA (1) MA53927B1 (fr)
MX (1) MX2021004457A (fr)
PE (1) PE20211818A1 (fr)
PH (1) PH12021550687A1 (fr)
PL (1) PL3866767T3 (fr)
PT (1) PT3866767T (fr)
RS (1) RS65012B1 (fr)
SG (1) SG11202103057RA (fr)
SI (1) SI3866767T1 (fr)
TW (1) TWI831848B (fr)
WO (1) WO2020079637A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020230091A1 (fr) 2019-05-14 2020-11-19 Janssen Biotech, Inc. Polythérapies avec des anticorps anti-egfr/c-met bispécifiques et des inhibiteurs de tyrosine kinase egfr de troisième génération
US11850248B2 (en) 2019-05-14 2023-12-26 Yuhan Corporation Therapies with 3rd generation EGFR tyrosine kinase inhibitors
TW202207940A (zh) * 2020-04-14 2022-03-01 美商健生生物科技公司 包含胺基嘧啶衍生物或其醫藥上可接受之鹽、水合物、或溶劑化物之用於經口投予之醫藥組成物
EP4349835A1 (fr) 2021-06-01 2024-04-10 Hangzhou Solipharma Co., Ltd. Forme cristalline d'hydrate de méthanesulfonate de lazertinib, son procédé de préparation et son utilisation

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL193673B1 (pl) * 1998-07-20 2007-03-30 Smithkline Beecham Corp Bezpostaciowa sól amonowa eprosartanu,jej granulat i biologicznie ulepszony preparat oraz sposoby ich wytwarzania i zastosowanie
DE10319450A1 (de) 2003-04-30 2004-11-18 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmazeutische Formulierung des Telmisartan Natriumsalzes
ES2359377T3 (es) * 2006-10-27 2011-05-23 Fmc Corporation Celulosa microcristalina coprocesada y alcohol de azúcar como excipiente para formulaciones de comprimidos.
JP5410290B2 (ja) 2006-10-27 2014-02-05 エフ エム シー コーポレーション 共処理組成物とその製造方法、打錠可能な錠剤処方物、錠剤の製造方法及び錠剤
WO2013016694A2 (fr) * 2011-07-27 2013-01-31 Cornell University Procédé pour la détection et la quantification d'arn
KR20140063808A (ko) 2011-09-14 2014-05-27 셀진 코포레이션 시클로프로판카르복실 산{2-[(1s)-1-(3-에톡시-4-메톡시-페닐)-2-메탄술포닐-에틸]-3-옥소-2,3-디하이드로-1h-이소인돌-4-일}-아마이드의 제제
CN104039319B (zh) 2011-11-29 2017-12-29 吉利德制药有限责任公司 用于治疗hcv的组合物和方法
WO2014175986A2 (fr) * 2013-04-23 2014-10-30 RevOrtho LLC Procédé et système de reconstruction de hanche modulaire
GB201400034D0 (en) 2014-01-02 2014-02-19 Astrazeneca Ab Pharmaceutical Compositions comprising AZD9291
SG11201701960XA (en) * 2014-10-13 2017-04-27 Yuhan Corp Compounds and compositions for modulating egfr mutant kinase activities
KR102606253B1 (ko) 2014-12-16 2023-11-27 시그날 파마소티칼 엘엘씨 2-(tert-부틸아미노)-4-((1r,3r,4r)-3-하이드록시-4-메틸사이클로헥실아미노)-피리미딘-5-카복사마이드의 제형
CN104788427B (zh) * 2015-02-05 2017-05-31 上海泓博智源医药股份有限公司 3‑(2‑嘧啶氨基)苯基丙烯酰胺类化合物及其应用
CN107847448A (zh) 2015-05-22 2018-03-27 诺华股份有限公司 药物组合物
KR102488488B1 (ko) 2015-10-07 2023-01-12 쿄와 기린 가부시키가이샤 아릴알킬아민 화합물 함유 의약 조성물
CA3019391A1 (fr) 2016-04-07 2017-10-12 Chemocentryx, Inc. Reduction de la charge tumorale par l'administration d'antagonistes de ccr1 en association avec des inhibiteurs de pd-1 ou des inhibiteurs de pd-l1
AR111469A1 (es) * 2017-04-21 2019-07-17 Yuhan Corp Sal de un compuesto del derivado de aminopiridina, una forma cristalina de la misma, y un proceso para preparar la misma
TW202207940A (zh) * 2020-04-14 2022-03-01 美商健生生物科技公司 包含胺基嘧啶衍生物或其醫藥上可接受之鹽、水合物、或溶劑化物之用於經口投予之醫藥組成物

Also Published As

Publication number Publication date
SI3866767T1 (sl) 2024-02-29
AR117655A1 (es) 2021-08-25
WO2020079637A1 (fr) 2020-04-23
ES2968966T3 (es) 2024-05-14
JP2024016052A (ja) 2024-02-06
EP3866767A4 (fr) 2022-07-20
DK3866767T3 (da) 2024-01-29
US20210322428A1 (en) 2021-10-21
JP2022504943A (ja) 2022-01-13
CN113015521A (zh) 2021-06-22
EA202191061A1 (ru) 2021-07-09
FI3866767T3 (fi) 2024-01-30
SG11202103057RA (en) 2021-05-28
KR20210061457A (ko) 2021-05-27
WO2020079637A9 (fr) 2020-07-23
TW202034903A (zh) 2020-10-01
EP3866767B1 (fr) 2023-11-29
BR112021007061A2 (pt) 2021-07-20
HRP20231670T1 (hr) 2024-03-15
PL3866767T3 (pl) 2024-04-02
CA3116652A1 (fr) 2020-04-23
EP3866767A1 (fr) 2021-08-25
EP4306113A2 (fr) 2024-01-17
EP4306113A3 (fr) 2024-02-14
MA53927B1 (fr) 2023-12-29
PT3866767T (pt) 2024-01-18
IL282163A (en) 2021-05-31
RS65012B1 (sr) 2024-01-31
PH12021550687A1 (en) 2022-02-14
LT3866767T (lt) 2023-12-27
AU2019360446A1 (en) 2021-04-22
TWI831848B (zh) 2024-02-11
JP7369769B2 (ja) 2023-10-26
PE20211818A1 (es) 2021-09-14
KR20200043618A (ko) 2020-04-28
MX2021004457A (es) 2021-07-07

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