SI3866767T1 - Farmacevtski sestavek za peroralno dajanje, ki obsega derivat aminopirimidina ali njegovo sol - Google Patents

Farmacevtski sestavek za peroralno dajanje, ki obsega derivat aminopirimidina ali njegovo sol

Info

Publication number
SI3866767T1
SI3866767T1 SI201930673T SI201930673T SI3866767T1 SI 3866767 T1 SI3866767 T1 SI 3866767T1 SI 201930673 T SI201930673 T SI 201930673T SI 201930673 T SI201930673 T SI 201930673T SI 3866767 T1 SI3866767 T1 SI 3866767T1
Authority
SI
Slovenia
Prior art keywords
salt
pharmaceutical composition
oral administration
aminopyrimidine derivative
aminopyrimidine
Prior art date
Application number
SI201930673T
Other languages
English (en)
Inventor
Seongkyu Kim
Deokkyu Lee
Soo-Won Kim
Jun-Mo Yang
Yoong-Sik Park
Original Assignee
Yuhan Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yuhan Corporation filed Critical Yuhan Corporation
Publication of SI3866767T1 publication Critical patent/SI3866767T1/sl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
SI201930673T 2018-10-18 2019-10-17 Farmacevtski sestavek za peroralno dajanje, ki obsega derivat aminopirimidina ali njegovo sol SI3866767T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR1020180124171A KR20200043618A (ko) 2018-10-18 2018-10-18 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구투여용 약학 조성물
PCT/IB2019/058862 WO2020079637A1 (en) 2018-10-18 2019-10-17 Pharmaceutical composition for oral administration comprising aminopyrimidine derivative or its salt
EP19872427.0A EP3866767B1 (en) 2018-10-18 2019-10-17 Pharmaceutical composition for oral administration comprising aminopyrimidine derivative or its salt

Publications (1)

Publication Number Publication Date
SI3866767T1 true SI3866767T1 (sl) 2024-02-29

Family

ID=70282933

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201930673T SI3866767T1 (sl) 2018-10-18 2019-10-17 Farmacevtski sestavek za peroralno dajanje, ki obsega derivat aminopirimidina ali njegovo sol

Country Status (26)

Country Link
US (1) US20210322428A1 (sl)
EP (2) EP3866767B1 (sl)
JP (2) JP7369769B2 (sl)
KR (2) KR20200043618A (sl)
CN (1) CN113015521A (sl)
AR (1) AR117655A1 (sl)
AU (1) AU2019360446A1 (sl)
BR (1) BR112021007061A2 (sl)
CA (1) CA3116652A1 (sl)
DK (1) DK3866767T3 (sl)
EA (1) EA202191061A1 (sl)
FI (1) FI3866767T3 (sl)
HR (1) HRP20231670T1 (sl)
IL (1) IL282163A (sl)
LT (1) LT3866767T (sl)
MA (1) MA53927B1 (sl)
MX (1) MX2021004457A (sl)
PE (1) PE20211818A1 (sl)
PH (1) PH12021550687A1 (sl)
PL (1) PL3866767T3 (sl)
PT (1) PT3866767T (sl)
RS (1) RS65012B1 (sl)
SG (1) SG11202103057RA (sl)
SI (1) SI3866767T1 (sl)
TW (1) TWI831848B (sl)
WO (1) WO2020079637A1 (sl)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JOP20210304A1 (ar) 2019-05-14 2023-01-30 Janssen Biotech Inc علاجات مركبة باستخدام الأجسام المضادة ثنائية النوعية المضادة لمستقبل عامل نمو البشرة (EGFR)/ مستقبل عامل نمو خلايا الكبد (c-Met) ومثبطات كيناز التيروسين الخاصة بمستقبل عامل نمو البشرة (EGFR) من الجيل الثالث
US11850248B2 (en) 2019-05-14 2023-12-26 Yuhan Corporation Therapies with 3rd generation EGFR tyrosine kinase inhibitors
TW202207940A (zh) * 2020-04-14 2022-03-01 美商健生生物科技公司 包含胺基嘧啶衍生物或其醫藥上可接受之鹽、水合物、或溶劑化物之用於經口投予之醫藥組成物
EP4349835A1 (en) 2021-06-01 2024-04-10 Hangzhou Solipharma Co., Ltd. Hydrate crystal form of lazertinib methanesulfonate, preparation method therefor and use thereof

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IL140905A0 (en) * 1998-07-20 2002-02-10 Smithkline Beecham Corp Bioenhanced formulations comprising eprosartan in oral solid dosage form
DE10319450A1 (de) 2003-04-30 2004-11-18 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmazeutische Formulierung des Telmisartan Natriumsalzes
WO2008057267A2 (en) 2006-10-27 2008-05-15 Fmc Corporation Co-processed microcrystalline cellulose and sugar alcohol as an excipient for tablet formulations
ES2359377T3 (es) * 2006-10-27 2011-05-23 Fmc Corporation Celulosa microcristalina coprocesada y alcohol de azúcar como excipiente para formulaciones de comprimidos.
WO2013016694A2 (en) * 2011-07-27 2013-01-31 Cornell University Methods for rna detection and quantification
SG11201400632YA (en) 2011-09-14 2014-04-28 Celgene Corp Formulations of cyclopropanecarboxylic acid {2-(1s)-1-(3-ethoxy-4-methoxy-phenyl)-2-methanesulfonyl-ethyl]-3-oxo-2,3-dihydro-1h-isoindol-4-yl}-amidecelgene corporation state of incorporation:delaware
MX2014006373A (es) 2011-11-29 2014-07-22 Gilead Pharmasset Llc Composiciones y metodos para tratar el virus de la hepatitis c.
WO2014175986A2 (en) * 2013-04-23 2014-10-30 RevOrtho LLC A method and system for modular hip resurfacing
GB201400034D0 (en) 2014-01-02 2014-02-19 Astrazeneca Ab Pharmaceutical Compositions comprising AZD9291
MX2017003181A (es) 2014-10-13 2017-07-20 Yuhan Corp Compuestos y composiciones para modular actividades de quinasa de mutante de receptor del factor de crecimiento epidermico.
EA033530B1 (ru) 2014-12-16 2019-10-31 Signal Pharm Llc Композиции 2-(трет-бутиламино)-4-((1r,3r,4r)-3-гидрокси-4-метилциклогексиламино)пиримидин-5-карбоксамида
CN104788427B (zh) * 2015-02-05 2017-05-31 上海泓博智源医药股份有限公司 3‑(2‑嘧啶氨基)苯基丙烯酰胺类化合物及其应用
CA2986522A1 (en) 2015-05-22 2016-12-01 Novartis Ag Pharmaceutical compositions
WO2017061621A1 (ja) 2015-10-07 2017-04-13 協和発酵キリン株式会社 アリールアルキルアミン化合物含有医薬組成物
WO2017176965A1 (en) 2016-04-07 2017-10-12 Chemocentryx, Inc. Reducing tumor burden by administering ccr1 antagonists in combination with pd-1 inhibitors or pd-l1 inhibitors
AR111469A1 (es) * 2017-04-21 2019-07-17 Yuhan Corp Sal de un compuesto del derivado de aminopiridina, una forma cristalina de la misma, y un proceso para preparar la misma
TW202207940A (zh) * 2020-04-14 2022-03-01 美商健生生物科技公司 包含胺基嘧啶衍生物或其醫藥上可接受之鹽、水合物、或溶劑化物之用於經口投予之醫藥組成物

Also Published As

Publication number Publication date
PE20211818A1 (es) 2021-09-14
BR112021007061A2 (pt) 2021-07-20
TW202034903A (zh) 2020-10-01
FI3866767T3 (fi) 2024-01-30
PH12021550687A1 (en) 2022-02-14
JP2024016052A (ja) 2024-02-06
MA53927B1 (fr) 2023-12-29
EP4306113A3 (en) 2024-02-14
TWI831848B (zh) 2024-02-11
WO2020079637A1 (en) 2020-04-23
KR20210061457A (ko) 2021-05-27
AU2019360446A1 (en) 2021-04-22
WO2020079637A9 (en) 2020-07-23
SG11202103057RA (en) 2021-05-28
EP3866767B1 (en) 2023-11-29
PL3866767T3 (pl) 2024-04-02
AR117655A1 (es) 2021-08-25
CN113015521A (zh) 2021-06-22
CA3116652A1 (en) 2020-04-23
EP3866767A4 (en) 2022-07-20
EA202191061A1 (ru) 2021-07-09
IL282163A (en) 2021-05-31
EP3866767A1 (en) 2021-08-25
DK3866767T3 (da) 2024-01-29
RS65012B1 (sr) 2024-01-31
PT3866767T (pt) 2024-01-18
HRP20231670T1 (hr) 2024-03-15
JP7369769B2 (ja) 2023-10-26
EP4306113A2 (en) 2024-01-17
JP2022504943A (ja) 2022-01-13
US20210322428A1 (en) 2021-10-21
KR20200043618A (ko) 2020-04-28
LT3866767T (lt) 2023-12-27
MX2021004457A (es) 2021-07-07
MA53927A (fr) 2021-09-15

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