MA46752A - Traitement de maladies du snc au moyen de stimulateurs de gcs - Google Patents

Traitement de maladies du snc au moyen de stimulateurs de gcs

Info

Publication number
MA46752A
MA46752A MA046752A MA46752A MA46752A MA 46752 A MA46752 A MA 46752A MA 046752 A MA046752 A MA 046752A MA 46752 A MA46752 A MA 46752A MA 46752 A MA46752 A MA 46752A
Authority
MA
Morocco
Prior art keywords
gcs
stimulators
treatment
cns diseases
cns
Prior art date
Application number
MA046752A
Other languages
English (en)
Inventor
Peter Germano
Rajesh R Iyengar
Joon Jung
Thomas Wai-Ho Lee
Nicholas Robert Perl
Maria D Ribadeneira
Kim Tang
Original Assignee
Cyclerion Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cyclerion Therapeutics Inc filed Critical Cyclerion Therapeutics Inc
Publication of MA46752A publication Critical patent/MA46752A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/5025Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA046752A 2016-11-08 2017-11-07 Traitement de maladies du snc au moyen de stimulateurs de gcs MA46752A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662419059P 2016-11-08 2016-11-08

Publications (1)

Publication Number Publication Date
MA46752A true MA46752A (fr) 2019-09-18

Family

ID=60452769

Family Applications (1)

Application Number Title Priority Date Filing Date
MA046752A MA46752A (fr) 2016-11-08 2017-11-07 Traitement de maladies du snc au moyen de stimulateurs de gcs

Country Status (18)

Country Link
US (2) US11690828B2 (fr)
EP (1) EP3538096B1 (fr)
JP (2) JP7150740B2 (fr)
KR (1) KR102475124B1 (fr)
CN (1) CN110267658B (fr)
AU (2) AU2017359018C1 (fr)
BR (1) BR112019009449A2 (fr)
CA (1) CA3042548A1 (fr)
CL (1) CL2019001256A1 (fr)
EA (1) EA201991147A1 (fr)
ES (1) ES2972711T3 (fr)
IL (1) IL266275B2 (fr)
MA (1) MA46752A (fr)
MX (2) MX2019005342A (fr)
PH (1) PH12019501016A1 (fr)
SG (1) SG10202104865UA (fr)
TW (1) TWI812601B (fr)
WO (1) WO2018089328A1 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3538520A2 (fr) * 2016-11-08 2019-09-18 Cyclerion Therapeutics, Inc. Stimulateurs de sgc
US11389449B2 (en) 2017-09-14 2022-07-19 Cyclerion Therapeutics, Inc. Treatment of metabolic syndrome with an sGC stimulator
BR112021000358A2 (pt) 2018-07-11 2021-04-06 Cyclerion Therapeutics, Inc. Uso de estimulantes de sgc para o tratamento de distúrbios mitocondriais
US20220087970A1 (en) * 2019-01-18 2022-03-24 The Johns Hopkins University Prevention of anesthetic-induced neurocognitive dysfunction
US20230012071A1 (en) * 2019-12-05 2023-01-12 Zydus Lifesciences Limited Modified release pharmaceutical compositions of riociguat
CN112924573B (zh) * 2021-01-21 2022-01-04 山东英盛生物技术有限公司 一种阿比多尔、利巴韦林、氯喹的hplc-ms/ms检测方法
WO2023130028A1 (fr) * 2021-12-31 2023-07-06 Tenax Therapeutics, Inc. Formulations orales de levosimendan pour le traitement de l'hypertension pulmonaire avec insuffisance cardiaque à fraction d'éjection préservée
WO2024163888A1 (fr) * 2023-02-03 2024-08-08 R.P. Scherer Technologies, Llc Capsules pharmaceutiques osmotiques

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US4627850A (en) 1983-11-02 1986-12-09 Alza Corporation Osmotic capsule
EP0192963B1 (fr) 1985-02-27 1988-07-20 Werkzeugmaschinenfabrik Oerlikon-Bührle AG Installation de mesure des vibrations d'une transmission à roues coniques dentées en spirale sur une machine d'essai de roues dentées
IL92966A (en) 1989-01-12 1995-07-31 Pfizer Hydrogel-operated release devices
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US5324280A (en) 1990-04-02 1994-06-28 Alza Corporation Osmotic dosage system for delivering a formulation comprising liquid carrier and drug
US5994341A (en) 1993-07-19 1999-11-30 Angiogenesis Technologies, Inc. Anti-angiogenic Compositions and methods for the treatment of arthritis
JP2928079B2 (ja) 1994-02-14 1999-07-28 永信薬品工業股▲ふん▼有限公司 1−(置換ベンジル)−3−(置換アリール)縮合ピラゾール類、その製造法及びその用途
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DE19830430A1 (de) 1998-07-08 2000-01-13 Hoechst Marion Roussel De Gmbh Schwefelsubstituierte Sulfonylamino-carbonsäure-N-arylamide, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate
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AU2009322836B2 (en) 2008-11-25 2013-04-04 Merck Sharp & Dohme Corp. Soluble guanylate cyclase activators
CA2753434C (fr) 2009-02-26 2014-07-15 Merck Sharp & Dohme Corp. Activateurs solubles de guanylate cyclase
WO2011119518A1 (fr) 2010-03-25 2011-09-29 Merck Sharp & Dohme Corp. Activateurs de guanylate cyclase solubles
MA34330B1 (fr) 2010-05-27 2013-06-01 Merck Sharp & Dohme Activateurs de guanylate cyclase soluble
EP2632551B1 (fr) 2010-10-28 2016-07-06 Merck Sharp & Dohme Corp. Activateurs de la guanylate cyclase soluble
EA201891416A1 (ru) * 2015-12-14 2018-12-28 Айронвуд Фармасьютикалз, Инк. ПРИМЕНЕНИЕ СТИМУЛЯТОРОВ sGC ДЛЯ ЛЕЧЕНИЯ ДИСФУНКЦИИ ЖЕЛУДОЧНО-КИШЕЧНОГО СФИНКТЕРА
WO2017108441A1 (fr) 2015-12-22 2017-06-29 Universiteit Maastricht Traitement de la déficience cognitive à l'aide d'un stimulateur de la sgc
WO2017121700A1 (fr) 2016-01-15 2017-07-20 Bayer Pharma Aktiengesellschaft Dérivés de 1h-pyrazolo[3,4-b]pyridine 1,3-disubstitués et leur utilisation en tant que stimulateurs de la guanylacte cyclase soluble
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Also Published As

Publication number Publication date
CA3042548A1 (fr) 2018-05-17
AU2017359018C1 (en) 2023-12-21
ES2972711T3 (es) 2024-06-14
EP3538096C0 (fr) 2024-02-28
CN110267658B (zh) 2024-02-02
AU2023270267A1 (en) 2023-12-07
WO2018089328A8 (fr) 2019-03-28
US11690828B2 (en) 2023-07-04
MX2022010852A (es) 2022-09-27
IL266275B2 (en) 2023-12-01
JP7150740B2 (ja) 2022-10-11
PH12019501016A1 (en) 2019-09-09
IL266275B1 (en) 2023-08-01
JP2022160605A (ja) 2022-10-19
EP3538096A1 (fr) 2019-09-18
MX2019005342A (es) 2019-10-02
KR20190094167A (ko) 2019-08-12
IL266275A (en) 2019-06-30
BR112019009449A2 (pt) 2019-07-30
JP2019534327A (ja) 2019-11-28
KR102475124B1 (ko) 2022-12-08
TW201822765A (zh) 2018-07-01
SG10202104865UA (en) 2021-06-29
AU2017359018B2 (en) 2023-08-31
CN110267658A (zh) 2019-09-20
WO2018089328A1 (fr) 2018-05-17
AU2017359018A1 (en) 2019-05-30
EA201991147A1 (ru) 2019-11-29
US20190343813A1 (en) 2019-11-14
CL2019001256A1 (es) 2019-10-04
TWI812601B (zh) 2023-08-21
EP3538096B1 (fr) 2024-02-28
US20230381153A1 (en) 2023-11-30

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