MA28946B1 - Utilisation de 4-(4-methylpiperazin-1-ylmethyl) -n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide pour inhiber le recepteur c-fms de la tyrosine kinase - Google Patents

Utilisation de 4-(4-methylpiperazin-1-ylmethyl) -n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide pour inhiber le recepteur c-fms de la tyrosine kinase

Info

Publication number
MA28946B1
MA28946B1 MA29848A MA29848A MA28946B1 MA 28946 B1 MA28946 B1 MA 28946B1 MA 29848 A MA29848 A MA 29848A MA 29848 A MA29848 A MA 29848A MA 28946 B1 MA28946 B1 MA 28946B1
Authority
MA
Morocco
Prior art keywords
methylpiperazin
ylamino
benzamide
pyrimidin
ylmethyl
Prior art date
Application number
MA29848A
Other languages
English (en)
Inventor
Andrea Louis Dewar
Timothy Peter Hughes
Alan Bruce Lyons
Original Assignee
Medvet Science Pty Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medvet Science Pty Ltd filed Critical Medvet Science Pty Ltd
Publication of MA28946B1 publication Critical patent/MA28946B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
MA29848A 2004-10-18 2007-04-25 Utilisation de 4-(4-methylpiperazin-1-ylmethyl) -n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide pour inhiber le recepteur c-fms de la tyrosine kinase MA28946B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US61974404P 2004-10-18 2004-10-18

Publications (1)

Publication Number Publication Date
MA28946B1 true MA28946B1 (fr) 2007-10-01

Family

ID=36202610

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29848A MA28946B1 (fr) 2004-10-18 2007-04-25 Utilisation de 4-(4-methylpiperazin-1-ylmethyl) -n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide pour inhiber le recepteur c-fms de la tyrosine kinase

Country Status (19)

Country Link
US (1) US20080255139A1 (fr)
EP (1) EP1804800B1 (fr)
JP (1) JP2008516898A (fr)
KR (1) KR20070083705A (fr)
CN (1) CN101035535A (fr)
AT (1) ATE492277T1 (fr)
AU (1) AU2005297321A1 (fr)
BR (1) BRPI0517083A (fr)
CA (1) CA2580976A1 (fr)
DE (1) DE602005025514D1 (fr)
IL (1) IL182419A0 (fr)
MA (1) MA28946B1 (fr)
MX (1) MX2007004660A (fr)
NO (1) NO20072501L (fr)
NZ (1) NZ554009A (fr)
RU (1) RU2007118420A (fr)
TN (1) TNSN07141A1 (fr)
WO (1) WO2006042362A1 (fr)
ZA (1) ZA200702316B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011502266A (ja) * 2007-10-31 2011-01-20 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Fms治療に対する応答を評価するバイオマーカー
EP3246046A4 (fr) * 2015-01-13 2018-12-05 Kyoto University Agent pour la prévention et/ou le traitement de la sclérose latérale amyotrophique

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4837237A (en) * 1985-07-09 1989-06-06 Fred Hutchinson Cancer Research Center Therapy using glucosidase processing inhibitors
CA2446939C (fr) * 2001-05-16 2005-08-02 Matthias Stein-Gerlach Derives de pyridylpyrimidine utilises comme composes actifs contre des infections et des maladies a prions
AU2003295320A1 (en) * 2002-06-26 2004-04-08 The Ohio State University Research Foundation The method for reducing inflammation using sti-571 or its salt

Also Published As

Publication number Publication date
KR20070083705A (ko) 2007-08-24
AU2005297321A1 (en) 2006-04-27
MX2007004660A (es) 2007-10-17
NO20072501L (no) 2007-05-15
ATE492277T1 (de) 2011-01-15
US20080255139A1 (en) 2008-10-16
TNSN07141A1 (en) 2008-11-21
JP2008516898A (ja) 2008-05-22
EP1804800A4 (fr) 2008-03-19
CN101035535A (zh) 2007-09-12
DE602005025514D1 (de) 2011-02-03
CA2580976A1 (fr) 2006-04-27
EP1804800A1 (fr) 2007-07-11
WO2006042362A1 (fr) 2006-04-27
NZ554009A (en) 2010-09-30
EP1804800B1 (fr) 2010-12-22
ZA200702316B (en) 2008-09-25
RU2007118420A (ru) 2008-11-27
BRPI0517083A (pt) 2008-09-30
IL182419A0 (en) 2007-09-20

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