NO20072501L - Anvendelse av 4-(4-metyopiperazin-1-ylmetyl)-N-[4-metyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)fenyl]-benzamid for a inhibere tyrosin kinasereseptor C-FMS - Google Patents

Anvendelse av 4-(4-metyopiperazin-1-ylmetyl)-N-[4-metyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)fenyl]-benzamid for a inhibere tyrosin kinasereseptor C-FMS

Info

Publication number
NO20072501L
NO20072501L NO20072501A NO20072501A NO20072501L NO 20072501 L NO20072501 L NO 20072501L NO 20072501 A NO20072501 A NO 20072501A NO 20072501 A NO20072501 A NO 20072501A NO 20072501 L NO20072501 L NO 20072501L
Authority
NO
Norway
Prior art keywords
fms
ylamino
benzamide
pyrimidin
ylmethyl
Prior art date
Application number
NO20072501A
Other languages
English (en)
Inventor
Andrea Louis Dewar
Timothy Peter Hughes
Alan Bruce Lyons
Original Assignee
Medvet Science Pty Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medvet Science Pty Ltd filed Critical Medvet Science Pty Ltd
Publication of NO20072501L publication Critical patent/NO20072501L/no

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Foreliggende oppfinnelse angår anvendelse av 4-(4-metylpiperazin-l-ylmetyl)-N-[4-metyl-3-(4-pyridin-3-yl)pyrimidin-2-ylamino)fenyl]-benzamid (også kjent som imatinib, gleevee, glivec, cgp57148b eller 8T1571), eller et farmasøytisk akseptabelt salt av denne, for fremstilling av et medikament for behandling av c-fms-assosierte sykdommer inkludert: koriokarsinom, malign histiocytose, embryonale karsinom, endometrialt karsinom, hjerne mikroblia tumorer, sarkoidose, mikroglia celleinvolvering ved normal og variant Creutzfeld-Jacob sykdom eller amyotrof lateral sklerose.
NO20072501A 2004-10-18 2007-05-15 Anvendelse av 4-(4-metyopiperazin-1-ylmetyl)-N-[4-metyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)fenyl]-benzamid for a inhibere tyrosin kinasereseptor C-FMS NO20072501L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61974404P 2004-10-18 2004-10-18
PCT/AU2005/001602 WO2006042362A1 (en) 2004-10-18 2005-10-17 Use of 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide to inhibit the tyrosine kinase receptor c-fms

Publications (1)

Publication Number Publication Date
NO20072501L true NO20072501L (no) 2007-05-15

Family

ID=36202610

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20072501A NO20072501L (no) 2004-10-18 2007-05-15 Anvendelse av 4-(4-metyopiperazin-1-ylmetyl)-N-[4-metyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)fenyl]-benzamid for a inhibere tyrosin kinasereseptor C-FMS

Country Status (19)

Country Link
US (1) US20080255139A1 (no)
EP (1) EP1804800B1 (no)
JP (1) JP2008516898A (no)
KR (1) KR20070083705A (no)
CN (1) CN101035535A (no)
AT (1) ATE492277T1 (no)
AU (1) AU2005297321A1 (no)
BR (1) BRPI0517083A (no)
CA (1) CA2580976A1 (no)
DE (1) DE602005025514D1 (no)
IL (1) IL182419A0 (no)
MA (1) MA28946B1 (no)
MX (1) MX2007004660A (no)
NO (1) NO20072501L (no)
NZ (1) NZ554009A (no)
RU (1) RU2007118420A (no)
TN (1) TNSN07141A1 (no)
WO (1) WO2006042362A1 (no)
ZA (1) ZA200702316B (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2215482A2 (en) * 2007-10-31 2010-08-11 Janssen Pharmaceutica N.V. Biomarker for assessing response to fms treatment
EP3789027A1 (en) * 2015-01-13 2021-03-10 Kyoto University Bosutinib, sunitinib, tivozanib, imatinib, nilotinib, rebastinib or bafetinib for preventing and/or treating amyotrophic lateral sclerosis

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4837237A (en) * 1985-07-09 1989-06-06 Fred Hutchinson Cancer Research Center Therapy using glucosidase processing inhibitors
AU2002342878A1 (en) * 2001-05-16 2002-11-25 Axxima Pharmaceuticals Ag Pyridylpyrimidine derivatives as effective compounds against prion diseases
WO2004026930A2 (en) * 2002-06-26 2004-04-01 The Ohio State University Research Foundation The method for reducing inflammation using sti-571 or its salt

Also Published As

Publication number Publication date
MX2007004660A (es) 2007-10-17
TNSN07141A1 (en) 2008-11-21
US20080255139A1 (en) 2008-10-16
AU2005297321A1 (en) 2006-04-27
ZA200702316B (en) 2008-09-25
EP1804800A4 (en) 2008-03-19
EP1804800A1 (en) 2007-07-11
ATE492277T1 (de) 2011-01-15
IL182419A0 (en) 2007-09-20
BRPI0517083A (pt) 2008-09-30
EP1804800B1 (en) 2010-12-22
RU2007118420A (ru) 2008-11-27
NZ554009A (en) 2010-09-30
MA28946B1 (fr) 2007-10-01
WO2006042362A1 (en) 2006-04-27
JP2008516898A (ja) 2008-05-22
KR20070083705A (ko) 2007-08-24
CA2580976A1 (en) 2006-04-27
CN101035535A (zh) 2007-09-12
DE602005025514D1 (de) 2011-02-03

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