MA27643A1 - Utilisation de n-alkyl-4-methyleneamino-3-hydroxy-2-pyridones en tant qu'agents antimicrobiens - Google Patents

Utilisation de n-alkyl-4-methyleneamino-3-hydroxy-2-pyridones en tant qu'agents antimicrobiens

Info

Publication number
MA27643A1
MA27643A1 MA28269A MA28269A MA27643A1 MA 27643 A1 MA27643 A1 MA 27643A1 MA 28269 A MA28269 A MA 28269A MA 28269 A MA28269 A MA 28269A MA 27643 A1 MA27643 A1 MA 27643A1
Authority
MA
Morocco
Prior art keywords
methyleneamino
pyridones
hydroxy
alkyl
antimicrobial agents
Prior art date
Application number
MA28269A
Other languages
English (en)
Inventor
Namal Chithranga Warshakoon
Rodney Dean Bush
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of MA27643A1 publication Critical patent/MA27643A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/69—Two or more oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

L'invention se rapporte à des composés représentés par la formuie (I), qui sont permettent de traiter efficacement des infections microbiennes
MA28269A 2002-11-09 2005-05-09 Utilisation de n-alkyl-4-methyleneamino-3-hydroxy-2-pyridones en tant qu'agents antimicrobiens MA27643A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42507002P 2002-11-09 2002-11-09

Publications (1)

Publication Number Publication Date
MA27643A1 true MA27643A1 (fr) 2005-12-01

Family

ID=32312926

Family Applications (1)

Application Number Title Priority Date Filing Date
MA28269A MA27643A1 (fr) 2002-11-09 2005-05-09 Utilisation de n-alkyl-4-methyleneamino-3-hydroxy-2-pyridones en tant qu'agents antimicrobiens

Country Status (26)

Country Link
US (5) US6930117B2 (fr)
EP (1) EP1558579B1 (fr)
JP (1) JP4496083B2 (fr)
KR (2) KR100896675B1 (fr)
CN (1) CN1708481A (fr)
AT (1) ATE372985T1 (fr)
AU (1) AU2003291382B2 (fr)
BR (1) BR0316107A (fr)
CA (1) CA2502264C (fr)
CO (1) CO5570678A2 (fr)
CY (1) CY1106958T1 (fr)
DE (1) DE60316338T2 (fr)
DK (1) DK1558579T3 (fr)
EG (1) EG25017A (fr)
ES (1) ES2293036T3 (fr)
HR (1) HRP20050516B1 (fr)
IL (1) IL168119A (fr)
MA (1) MA27643A1 (fr)
MX (1) MXPA05004896A (fr)
NO (1) NO330810B1 (fr)
NZ (1) NZ539386A (fr)
PL (1) PL377226A1 (fr)
PT (1) PT1558579E (fr)
RU (1) RU2311410C2 (fr)
WO (1) WO2004043927A1 (fr)
ZA (1) ZA200503683B (fr)

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EP2542077A4 (fr) * 2010-03-04 2013-08-21 Merck Sharp & Dohme Inhibiteurs de catéchol o-méthyl transférase et utilisation associée dans le traitement de troubles psychotiques
WO2011109267A1 (fr) 2010-03-04 2011-09-09 Merck Sharp & Dohme Corp. Inhibiteurs de catéchol o-méthyl transférase et utilisation associée dans le traitement de troubles psychotiques
PL2649069T3 (pl) 2010-11-08 2016-01-29 Janssen Pharmaceuticals Inc Pochodne 1,2,4-triazolo[4,3-a]pirydyny i ich zastosowanie jako dodatnich allosterycznych modulatorów receptorów mGluR2
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Also Published As

Publication number Publication date
RU2005114489A (ru) 2005-11-20
RU2311410C2 (ru) 2007-11-27
ZA200503683B (en) 2006-08-30
AU2003291382A1 (en) 2004-06-03
NZ539386A (en) 2008-02-29
EP1558579A1 (fr) 2005-08-03
US8133894B2 (en) 2012-03-13
NO20052787D0 (no) 2005-06-09
WO2004043927A1 (fr) 2004-05-27
US20040097560A1 (en) 2004-05-20
US7247648B2 (en) 2007-07-24
ES2293036T3 (es) 2008-03-16
HRP20050516A2 (en) 2005-12-31
US20050234045A1 (en) 2005-10-20
KR20050055792A (ko) 2005-06-13
BR0316107A (pt) 2005-09-27
NO330810B1 (no) 2011-07-25
US7790748B2 (en) 2010-09-07
DE60316338D1 (de) 2007-10-25
CY1106958T1 (el) 2012-09-26
KR100896675B1 (ko) 2009-05-08
US20120115876A1 (en) 2012-05-10
DE60316338T2 (de) 2008-06-05
CA2502264C (fr) 2009-12-15
PL377226A1 (pl) 2006-01-23
ATE372985T1 (de) 2007-09-15
CO5570678A2 (es) 2005-10-31
NO20052787L (no) 2005-06-09
PT1558579E (pt) 2007-11-27
HRP20050516B1 (hr) 2013-11-08
US20100305097A1 (en) 2010-12-02
CN1708481A (zh) 2005-12-14
KR20070026891A (ko) 2007-03-08
AU2003291382B2 (en) 2008-07-31
IL168119A (en) 2011-11-30
MXPA05004896A (es) 2005-07-22
EP1558579B1 (fr) 2007-09-12
DK1558579T3 (da) 2008-01-14
JP4496083B2 (ja) 2010-07-07
EG25017A (en) 2011-05-25
JP2006508133A (ja) 2006-03-09
US6930117B2 (en) 2005-08-16
US20070270407A1 (en) 2007-11-22
CA2502264A1 (fr) 2004-05-27

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