LU79750A1 - PROCESS FOR THE PREPARATION OF NEW FLUORINE AMINO ACIDS - Google Patents

PROCESS FOR THE PREPARATION OF NEW FLUORINE AMINO ACIDS

Info

Publication number
LU79750A1
LU79750A1 LU79750A LU79750A LU79750A1 LU 79750 A1 LU79750 A1 LU 79750A1 LU 79750 A LU79750 A LU 79750A LU 79750 A LU79750 A LU 79750A LU 79750 A1 LU79750 A1 LU 79750A1
Authority
LU
Luxembourg
Prior art keywords
preparation
amino acids
new fluorine
fluorine amino
new
Prior art date
Application number
LU79750A
Other languages
French (fr)
Inventor
A Patchett
J Kollonitsch
S Marburg
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/802,391 external-priority patent/US4325961A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of LU79750A1 publication Critical patent/LU79750A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
LU79750A 1977-06-01 1978-06-01 PROCESS FOR THE PREPARATION OF NEW FLUORINE AMINO ACIDS LU79750A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80238977A 1977-06-01 1977-06-01
US05/802,391 US4325961A (en) 1977-06-01 1977-06-01 Fluorinated amino acids

Publications (1)

Publication Number Publication Date
LU79750A1 true LU79750A1 (en) 1979-02-02

Family

ID=27122442

Family Applications (1)

Application Number Title Priority Date Filing Date
LU79750A LU79750A1 (en) 1977-06-01 1978-06-01 PROCESS FOR THE PREPARATION OF NEW FLUORINE AMINO ACIDS

Country Status (26)

Country Link
JP (1) JPS5416423A (en)
AR (1) AR223463A1 (en)
AT (1) AT360509B (en)
AU (1) AU518479B2 (en)
CA (1) CA1120040A (en)
CH (1) CH639639A5 (en)
DD (1) DD138651A5 (en)
DE (1) DE2824116A1 (en)
DK (1) DK149841C (en)
ES (1) ES470296A1 (en)
FI (1) FI66840C (en)
FR (1) FR2392958A1 (en)
GB (1) GB1602525A (en)
GR (1) GR64495B (en)
HK (1) HK18184A (en)
HU (1) HU181911B (en)
IE (1) IE46983B1 (en)
IT (1) IT1104709B (en)
LU (1) LU79750A1 (en)
NL (1) NL190485C (en)
NO (1) NO147382C (en)
NZ (1) NZ187377A (en)
PL (1) PL115731B1 (en)
PT (1) PT68102B (en)
SE (1) SE7806440L (en)
YU (1) YU129178A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA783273B (en) * 1977-07-11 1979-06-27 Merrell Toraude & Co A-halomethyl amino acids
IL59481A0 (en) * 1977-07-11 1980-05-30 Merrell Toraude & Co -halomethyl amino acids
CA1091661A (en) * 1977-07-11 1980-12-16 Philippe Bey .alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS
US4315095A (en) * 1977-07-28 1982-02-09 Merrell Toraude Et Compagnie α-Halomethyl derivatives of amino acids
ATE3282T1 (en) * 1978-07-24 1983-05-15 Merck & Co. Inc. ALPHA-DIFLUOROMETHYL-ALPHA-AMINO ACIDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM.
IE49522B1 (en) * 1979-04-26 1985-10-16 Merrell Toraude & Co Alpha-halomethylaminoacids
CA1158657A (en) * 1979-07-26 1983-12-13 Philippe Bey Preparation of fluorinated methyl aminoalkanoic acids and novel process intermediates
ZA813018B (en) * 1980-05-09 1982-05-26 Merrell Toraude & Co Fluoromethylated tyrosine methyl ester
NZ197394A (en) * 1980-06-16 1984-09-28 Merrell Dow Pharma Inhibition of protozoal growth in animals with certain-substituted-amines or amino acids
US4421767A (en) * 1981-06-01 1983-12-20 Merrell Toraude Et Compagnie Compounds and methods for treating depression
GB9325368D0 (en) * 1993-12-10 1994-02-16 Univ Bristol Organic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3046300A (en) * 1960-10-21 1962-07-24 Merck & Co Inc alpha-trifluoromethyloxyphenylalanines

Also Published As

Publication number Publication date
AT360509B (en) 1981-01-12
DK237978A (en) 1979-01-19
DD138651A5 (en) 1979-11-14
DE2824116A1 (en) 1978-12-14
PT68102B (en) 1982-06-08
GB1602525A (en) 1981-11-11
FR2392958A1 (en) 1978-12-29
DK149841B (en) 1986-10-13
IT7849637A0 (en) 1978-05-31
NL190485C (en) 1994-03-16
JPS5416423A (en) 1979-02-07
DE2824116C2 (en) 1989-04-27
YU129178A (en) 1983-01-21
JPS641474B2 (en) 1989-01-11
AR223463A1 (en) 1981-08-31
NL7805981A (en) 1978-12-05
SE7806440L (en) 1978-12-02
NO147382C (en) 1983-03-30
HU181911B (en) 1983-11-28
NO781892L (en) 1978-12-04
CA1120040A (en) 1982-03-16
ATA393278A (en) 1980-06-15
PL115731B1 (en) 1981-04-30
FR2392958B1 (en) 1980-10-24
GR64495B (en) 1980-03-31
IE781078L (en) 1978-12-01
CH639639A5 (en) 1983-11-30
FI781674A (en) 1978-12-02
PL207242A1 (en) 1979-04-23
NZ187377A (en) 1981-05-15
AU3658678A (en) 1979-12-06
HK18184A (en) 1984-03-09
IE46983B1 (en) 1983-11-16
NO147382B (en) 1982-12-20
NL190485B (en) 1993-10-18
IT1104709B (en) 1985-10-28
FI66840B (en) 1984-08-31
DK149841C (en) 1987-04-21
AU518479B2 (en) 1981-10-01
FI66840C (en) 1984-12-10
PT68102A (en) 1978-06-01
ES470296A1 (en) 1979-09-16

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