AR223463A1 - PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS - Google Patents
PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDSInfo
- Publication number
- AR223463A1 AR223463A1 AR272336A AR27233678A AR223463A1 AR 223463 A1 AR223463 A1 AR 223463A1 AR 272336 A AR272336 A AR 272336A AR 27233678 A AR27233678 A AR 27233678A AR 223463 A1 AR223463 A1 AR 223463A1
- Authority
- AR
- Argentina
- Prior art keywords
- alpha
- fluormethyl
- amino
- procedure
- obtaining substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US80238977A | 1977-06-01 | 1977-06-01 | |
US05/802,391 US4325961A (en) | 1977-06-01 | 1977-06-01 | Fluorinated amino acids |
Publications (1)
Publication Number | Publication Date |
---|---|
AR223463A1 true AR223463A1 (en) | 1981-08-31 |
Family
ID=27122442
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR272336A AR223463A1 (en) | 1977-06-01 | 1978-05-26 | PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS |
Country Status (26)
Country | Link |
---|---|
JP (1) | JPS5416423A (en) |
AR (1) | AR223463A1 (en) |
AT (1) | AT360509B (en) |
AU (1) | AU518479B2 (en) |
CA (1) | CA1120040A (en) |
CH (1) | CH639639A5 (en) |
DD (1) | DD138651A5 (en) |
DE (1) | DE2824116A1 (en) |
DK (1) | DK149841C (en) |
ES (1) | ES470296A1 (en) |
FI (1) | FI66840C (en) |
FR (1) | FR2392958A1 (en) |
GB (1) | GB1602525A (en) |
GR (1) | GR64495B (en) |
HK (1) | HK18184A (en) |
HU (1) | HU181911B (en) |
IE (1) | IE46983B1 (en) |
IT (1) | IT1104709B (en) |
LU (1) | LU79750A1 (en) |
NL (1) | NL190485C (en) |
NO (1) | NO147382C (en) |
NZ (1) | NZ187377A (en) |
PL (1) | PL115731B1 (en) |
PT (1) | PT68102B (en) |
SE (1) | SE7806440L (en) |
YU (1) | YU129178A (en) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1091661A (en) * | 1977-07-11 | 1980-12-16 | Philippe Bey | .alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS |
ZA783273B (en) * | 1977-07-11 | 1979-06-27 | Merrell Toraude & Co | A-halomethyl amino acids |
IL59481A0 (en) * | 1977-07-11 | 1980-05-30 | Merrell Toraude & Co | -halomethyl amino acids |
US4315095A (en) * | 1977-07-28 | 1982-02-09 | Merrell Toraude Et Compagnie | α-Halomethyl derivatives of amino acids |
ATE3282T1 (en) * | 1978-07-24 | 1983-05-15 | Merck & Co. Inc. | ALPHA-DIFLUOROMETHYL-ALPHA-AMINO ACIDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM. |
IE49522B1 (en) * | 1979-04-26 | 1985-10-16 | Merrell Toraude & Co | Alpha-halomethylaminoacids |
CA1158657A (en) * | 1979-07-26 | 1983-12-13 | Philippe Bey | Preparation of fluorinated methyl aminoalkanoic acids and novel process intermediates |
ZA813018B (en) * | 1980-05-09 | 1982-05-26 | Merrell Toraude & Co | Fluoromethylated tyrosine methyl ester |
PH16634A (en) * | 1980-06-16 | 1983-12-05 | Merrell Dow Pharma | Method of inhibiting the growth of protozoa |
US4421767A (en) * | 1981-06-01 | 1983-12-20 | Merrell Toraude Et Compagnie | Compounds and methods for treating depression |
GB9325368D0 (en) * | 1993-12-10 | 1994-02-16 | Univ Bristol | Organic compounds |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3046300A (en) * | 1960-10-21 | 1962-07-24 | Merck & Co Inc | alpha-trifluoromethyloxyphenylalanines |
-
1978
- 1978-05-25 FR FR7815567A patent/FR2392958A1/en active Granted
- 1978-05-25 GR GR56328A patent/GR64495B/en unknown
- 1978-05-25 NZ NZ187377A patent/NZ187377A/en unknown
- 1978-05-26 FI FI781674A patent/FI66840C/en not_active IP Right Cessation
- 1978-05-26 AR AR272336A patent/AR223463A1/en active
- 1978-05-29 CA CA000304318A patent/CA1120040A/en not_active Expired
- 1978-05-29 AU AU36586/78A patent/AU518479B2/en not_active Expired
- 1978-05-29 ES ES470296A patent/ES470296A1/en not_active Expired
- 1978-05-30 DK DK237978A patent/DK149841C/en not_active IP Right Cessation
- 1978-05-30 GB GB24330/78A patent/GB1602525A/en not_active Expired
- 1978-05-30 YU YU01291/78A patent/YU129178A/en unknown
- 1978-05-30 PT PT68102A patent/PT68102B/en unknown
- 1978-05-30 HU HU78ME2169A patent/HU181911B/en unknown
- 1978-05-30 IE IE1078/78A patent/IE46983B1/en unknown
- 1978-05-30 AT AT393278A patent/AT360509B/en not_active IP Right Cessation
- 1978-05-30 DD DD78205669A patent/DD138651A5/en unknown
- 1978-05-31 CH CH597978A patent/CH639639A5/en not_active IP Right Cessation
- 1978-05-31 IT IT49637/78A patent/IT1104709B/en active
- 1978-05-31 NO NO781892A patent/NO147382C/en unknown
- 1978-05-31 PL PL1978207242A patent/PL115731B1/en unknown
- 1978-06-01 JP JP6501678A patent/JPS5416423A/en active Granted
- 1978-06-01 DE DE19782824116 patent/DE2824116A1/en active Granted
- 1978-06-01 SE SE7806440A patent/SE7806440L/en unknown
- 1978-06-01 NL NLAANVRAGE7805981,A patent/NL190485C/en not_active IP Right Cessation
- 1978-06-01 LU LU79750A patent/LU79750A1/en unknown
-
1984
- 1984-03-01 HK HK181/84A patent/HK18184A/en not_active IP Right Cessation
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