AR223463A1 - PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS - Google Patents

PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS

Info

Publication number
AR223463A1
AR223463A1 AR272336A AR27233678A AR223463A1 AR 223463 A1 AR223463 A1 AR 223463A1 AR 272336 A AR272336 A AR 272336A AR 27233678 A AR27233678 A AR 27233678A AR 223463 A1 AR223463 A1 AR 223463A1
Authority
AR
Argentina
Prior art keywords
alpha
fluormethyl
amino
procedure
obtaining substituted
Prior art date
Application number
AR272336A
Other languages
Spanish (es)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/802,391 external-priority patent/US4325961A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Application granted granted Critical
Publication of AR223463A1 publication Critical patent/AR223463A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
AR272336A 1977-06-01 1978-05-26 PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS AR223463A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80238977A 1977-06-01 1977-06-01
US05/802,391 US4325961A (en) 1977-06-01 1977-06-01 Fluorinated amino acids

Publications (1)

Publication Number Publication Date
AR223463A1 true AR223463A1 (en) 1981-08-31

Family

ID=27122442

Family Applications (1)

Application Number Title Priority Date Filing Date
AR272336A AR223463A1 (en) 1977-06-01 1978-05-26 PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS

Country Status (26)

Country Link
JP (1) JPS5416423A (en)
AR (1) AR223463A1 (en)
AT (1) AT360509B (en)
AU (1) AU518479B2 (en)
CA (1) CA1120040A (en)
CH (1) CH639639A5 (en)
DD (1) DD138651A5 (en)
DE (1) DE2824116A1 (en)
DK (1) DK149841C (en)
ES (1) ES470296A1 (en)
FI (1) FI66840C (en)
FR (1) FR2392958A1 (en)
GB (1) GB1602525A (en)
GR (1) GR64495B (en)
HK (1) HK18184A (en)
HU (1) HU181911B (en)
IE (1) IE46983B1 (en)
IT (1) IT1104709B (en)
LU (1) LU79750A1 (en)
NL (1) NL190485C (en)
NO (1) NO147382C (en)
NZ (1) NZ187377A (en)
PL (1) PL115731B1 (en)
PT (1) PT68102B (en)
SE (1) SE7806440L (en)
YU (1) YU129178A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1091661A (en) * 1977-07-11 1980-12-16 Philippe Bey .alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS
ZA783273B (en) * 1977-07-11 1979-06-27 Merrell Toraude & Co A-halomethyl amino acids
IL59481A0 (en) * 1977-07-11 1980-05-30 Merrell Toraude & Co -halomethyl amino acids
US4315095A (en) * 1977-07-28 1982-02-09 Merrell Toraude Et Compagnie α-Halomethyl derivatives of amino acids
ATE3282T1 (en) * 1978-07-24 1983-05-15 Merck & Co. Inc. ALPHA-DIFLUOROMETHYL-ALPHA-AMINO ACIDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM.
IE49522B1 (en) * 1979-04-26 1985-10-16 Merrell Toraude & Co Alpha-halomethylaminoacids
CA1158657A (en) * 1979-07-26 1983-12-13 Philippe Bey Preparation of fluorinated methyl aminoalkanoic acids and novel process intermediates
ZA813018B (en) * 1980-05-09 1982-05-26 Merrell Toraude & Co Fluoromethylated tyrosine methyl ester
PH16634A (en) * 1980-06-16 1983-12-05 Merrell Dow Pharma Method of inhibiting the growth of protozoa
US4421767A (en) * 1981-06-01 1983-12-20 Merrell Toraude Et Compagnie Compounds and methods for treating depression
GB9325368D0 (en) * 1993-12-10 1994-02-16 Univ Bristol Organic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3046300A (en) * 1960-10-21 1962-07-24 Merck & Co Inc alpha-trifluoromethyloxyphenylalanines

Also Published As

Publication number Publication date
DK237978A (en) 1979-01-19
ES470296A1 (en) 1979-09-16
LU79750A1 (en) 1979-02-02
PL115731B1 (en) 1981-04-30
AT360509B (en) 1981-01-12
DK149841C (en) 1987-04-21
FI781674A (en) 1978-12-02
JPS641474B2 (en) 1989-01-11
NO781892L (en) 1978-12-04
IT7849637A0 (en) 1978-05-31
NO147382C (en) 1983-03-30
JPS5416423A (en) 1979-02-07
FI66840C (en) 1984-12-10
FI66840B (en) 1984-08-31
GB1602525A (en) 1981-11-11
AU518479B2 (en) 1981-10-01
NL7805981A (en) 1978-12-05
DK149841B (en) 1986-10-13
AU3658678A (en) 1979-12-06
DD138651A5 (en) 1979-11-14
NL190485B (en) 1993-10-18
IT1104709B (en) 1985-10-28
PT68102A (en) 1978-06-01
CH639639A5 (en) 1983-11-30
CA1120040A (en) 1982-03-16
DE2824116C2 (en) 1989-04-27
GR64495B (en) 1980-03-31
PT68102B (en) 1982-06-08
DE2824116A1 (en) 1978-12-14
HU181911B (en) 1983-11-28
SE7806440L (en) 1978-12-02
FR2392958A1 (en) 1978-12-29
ATA393278A (en) 1980-06-15
IE781078L (en) 1978-12-01
NO147382B (en) 1982-12-20
IE46983B1 (en) 1983-11-16
PL207242A1 (en) 1979-04-23
HK18184A (en) 1984-03-09
NZ187377A (en) 1981-05-15
NL190485C (en) 1994-03-16
FR2392958B1 (en) 1980-10-24
YU129178A (en) 1983-01-21

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