AR223463A1 - PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS - Google Patents

PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS

Info

Publication number
AR223463A1
AR223463A1 AR272336A AR27233678A AR223463A1 AR 223463 A1 AR223463 A1 AR 223463A1 AR 272336 A AR272336 A AR 272336A AR 27233678 A AR27233678 A AR 27233678A AR 223463 A1 AR223463 A1 AR 223463A1
Authority
AR
Argentina
Prior art keywords
alpha
fluormethyl
amino
procedure
obtaining substituted
Prior art date
Application number
AR272336A
Other languages
Spanish (es)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/802,391 external-priority patent/US4325961A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Application granted granted Critical
Publication of AR223463A1 publication Critical patent/AR223463A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
AR272336A 1977-06-01 1978-05-26 PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS AR223463A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80238977A 1977-06-01 1977-06-01
US05/802,391 US4325961A (en) 1977-06-01 1977-06-01 Fluorinated amino acids

Publications (1)

Publication Number Publication Date
AR223463A1 true AR223463A1 (en) 1981-08-31

Family

ID=27122442

Family Applications (1)

Application Number Title Priority Date Filing Date
AR272336A AR223463A1 (en) 1977-06-01 1978-05-26 PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS

Country Status (26)

Country Link
JP (1) JPS5416423A (en)
AR (1) AR223463A1 (en)
AT (1) AT360509B (en)
AU (1) AU518479B2 (en)
CA (1) CA1120040A (en)
CH (1) CH639639A5 (en)
DD (1) DD138651A5 (en)
DE (1) DE2824116A1 (en)
DK (1) DK149841C (en)
ES (1) ES470296A1 (en)
FI (1) FI66840C (en)
FR (1) FR2392958A1 (en)
GB (1) GB1602525A (en)
GR (1) GR64495B (en)
HK (1) HK18184A (en)
HU (1) HU181911B (en)
IE (1) IE46983B1 (en)
IT (1) IT1104709B (en)
LU (1) LU79750A1 (en)
NL (1) NL190485C (en)
NO (1) NO147382C (en)
NZ (1) NZ187377A (en)
PL (1) PL115731B1 (en)
PT (1) PT68102B (en)
SE (1) SE7806440L (en)
YU (1) YU129178A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1091661A (en) * 1977-07-11 1980-12-16 Philippe Bey .alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS
IL59481A0 (en) * 1977-07-11 1980-05-30 Merrell Toraude & Co -halomethyl amino acids
ZA783273B (en) * 1977-07-11 1979-06-27 Merrell Toraude & Co A-halomethyl amino acids
US4315095A (en) * 1977-07-28 1982-02-09 Merrell Toraude Et Compagnie α-Halomethyl derivatives of amino acids
EP0007600B1 (en) * 1978-07-24 1983-05-11 Merck & Co. Inc. Alpha-difluoromethyl amino acids and pharmaceutical composition containing the same
IE49522B1 (en) * 1979-04-26 1985-10-16 Merrell Toraude & Co Alpha-halomethylaminoacids
NZ194347A (en) * 1979-07-26 1982-11-23 Merrell Toraude & Co Fluorinated alkenylamines intermediate alkenyl fluorinated methyl ketimine magnesium halides and preparation of certain amino alkanoic acids
ZA813018B (en) * 1980-05-09 1982-05-26 Merrell Toraude & Co Fluoromethylated tyrosine methyl ester
PH16634A (en) * 1980-06-16 1983-12-05 Merrell Dow Pharma Method of inhibiting the growth of protozoa
US4421767A (en) * 1981-06-01 1983-12-20 Merrell Toraude Et Compagnie Compounds and methods for treating depression
GB9325368D0 (en) * 1993-12-10 1994-02-16 Univ Bristol Organic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3046300A (en) * 1960-10-21 1962-07-24 Merck & Co Inc alpha-trifluoromethyloxyphenylalanines

Also Published As

Publication number Publication date
CA1120040A (en) 1982-03-16
NO781892L (en) 1978-12-04
NO147382C (en) 1983-03-30
NL7805981A (en) 1978-12-05
DK237978A (en) 1979-01-19
IE46983B1 (en) 1983-11-16
IE781078L (en) 1978-12-01
LU79750A1 (en) 1979-02-02
PT68102B (en) 1982-06-08
FI781674A7 (en) 1978-12-02
PL207242A1 (en) 1979-04-23
IT7849637A0 (en) 1978-05-31
ATA393278A (en) 1980-06-15
FR2392958B1 (en) 1980-10-24
ES470296A1 (en) 1979-09-16
DD138651A5 (en) 1979-11-14
IT1104709B (en) 1985-10-28
NL190485C (en) 1994-03-16
NZ187377A (en) 1981-05-15
GR64495B (en) 1980-03-31
HU181911B (en) 1983-11-28
SE7806440L (en) 1978-12-02
DE2824116A1 (en) 1978-12-14
DK149841B (en) 1986-10-13
AU518479B2 (en) 1981-10-01
FI66840C (en) 1984-12-10
JPS641474B2 (en) 1989-01-11
PL115731B1 (en) 1981-04-30
PT68102A (en) 1978-06-01
GB1602525A (en) 1981-11-11
DE2824116C2 (en) 1989-04-27
AT360509B (en) 1981-01-12
NO147382B (en) 1982-12-20
AU3658678A (en) 1979-12-06
CH639639A5 (en) 1983-11-30
HK18184A (en) 1984-03-09
DK149841C (en) 1987-04-21
YU129178A (en) 1983-01-21
JPS5416423A (en) 1979-02-07
FI66840B (en) 1984-08-31
NL190485B (en) 1993-10-18
FR2392958A1 (en) 1978-12-29

Similar Documents

Publication Publication Date Title
MX5449E (en) PROCEDURE FOR PREPARING HYDROXIDIPHOSPHONIC ACIDS
MX147446A (en) IMPROVED PROCEDURE FOR BENCHENE ETILATION
AR230452A1 (en) PROCEDURE FOR PREPARING ACID COMPOUNDS 7-SUBSTITUTED-3-CEFEM-4-CARBOXYLICS
MX147968A (en) PROCEDURE FOR PREPARING POLYETHERAMIDE ACIDS
MX5535E (en) PROCEDURE FOR PREPARING 2-ALPHA-CIANO-3-OXO-STEROIDS
MX148160A (en) IMPROVED PROCEDURE FOR OBTAINING ALCOXISILANES
MX5352E (en) IMPROVED PROCEDURE FOR OBTAINING ALQUENILSUCCINIMIDAS
MX147874A (en) PROCEDURE FOR PREPARING COMPOUNDS 2-PHENOXY-5-TRIFLUOROMETILPIRIDINA
AR224238A1 (en) PROCEDURE FOR OBTAINING TETRAPEPTIDES
MX148906A (en) PROCEDURE FOR OBTAINING DIHYDROXYPOLIURETHANES
AR223463A1 (en) PROCEDURE FOR OBTAINING SUBSTITUTED ALPHA-FLUORMETHYL-ALPHA-AMINO-ALCANOIC ACIDS
MX151851A (en) IMPROVED PROCEDURE FOR PREPARING TRIACINE DERIVATIVES
AR223656A1 (en) PROCEDURE FOR OBTAINING 2-PHENYLIMINOIMIDAZOLIDINE DERIVATIVES
MX149268A (en) PROCEDURE FOR PREPARING ALIPHATIC DIPEROXIDICARBOXYLLIC ACIDS
AR222815A1 (en) PROCEDURE FOR THE PREPARATION OF ACIDS (ALPHA-TRIFLUOROMETIL-MERCAPTO-PROPIONIL) -PIRROLIDINIL-O TIAZOLIDINIL-CARBOXILICOS
AR219727A1 (en) PROCEDURE FOR OBTAINING SUBSTITUTED NONATETRAENE FENILE
AR221845A1 (en) PROCEDURE FOR OBTAINING NEW N1-GLUCOFURANOSID-6-I1-N3-UREAS
MX5434E (en) PROCEDURE FOR PREPARING CYCLOPROFILCARBOXYLATES
MX5160E (en) IMPROVED PROCEDURE FOR PREPARING AMINOALCOHOLE DERIVATIVES
AR213652A1 (en) PROCEDURE FOR OBTAINING 5-M-TOLIL OXYURACILO
AR218933A1 (en) PROCEDURE FOR OBTAINING OXAZOLIDONE-2 DERIVATIVES
MX5398E (en) PROCEDURE FOR PREPARING ALPHA-CYANO-BENCILO ESTERS
MX150015A (en) IMPROVED PROCEDURE FOR MAKING SIGNS
MX5186E (en) PROCEDURE FOR PREPARING BENCILOXIME ETERS
MX5208E (en) PROCEDURE FOR PREPARING DICLOROVINILCICLOBUTANONAS