LT3081B - Novel pilocarpine derivatives and process for their preparation - Google Patents

Novel pilocarpine derivatives and process for their preparation Download PDF

Info

Publication number
LT3081B
LT3081B LTIP576A LTIP576A LT3081B LT 3081 B LT3081 B LT 3081B LT IP576 A LTIP576 A LT IP576A LT IP576 A LTIP576 A LT IP576A LT 3081 B LT3081 B LT 3081B
Authority
LT
Lithuania
Prior art keywords
bispilocarpate
formula
ethylene
propylene
derivatives
Prior art date
Application number
LTIP576A
Other languages
English (en)
Lithuanian (lt)
Inventor
Tomi Jaervinen
Pekka Peura
Pekka Suhonen
Arto Urtti
Hannu Hanhijaervi
Esko Pohjala
Original Assignee
Leiras Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leiras Oy filed Critical Leiras Oy
Publication of LTIP576A publication Critical patent/LTIP576A/xx
Publication of LT3081B publication Critical patent/LT3081B/lt

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
LTIP576A 1992-05-29 1993-05-28 Novel pilocarpine derivatives and process for their preparation LT3081B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FI922518A FI98910C (fi) 1992-05-29 1992-05-29 Menetelmä farmaseuttisesti käyttökelpoisten pilokarpiinijohdannaisten valmistamiseksi

Publications (2)

Publication Number Publication Date
LTIP576A LTIP576A (en) 1994-06-15
LT3081B true LT3081B (en) 1994-11-25

Family

ID=8535384

Family Applications (1)

Application Number Title Priority Date Filing Date
LTIP576A LT3081B (en) 1992-05-29 1993-05-28 Novel pilocarpine derivatives and process for their preparation

Country Status (2)

Country Link
FI (1) FI98910C (fi)
LT (1) LT3081B (fi)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4061722A (en) 1976-04-26 1977-12-06 Interx Research Corporation Selected quaternary ammonium salts of pilocarpine useful in reducing intraocular pressure in warm-blooded animals
EP0106541A2 (en) 1982-09-17 1984-04-25 Hans Bundgaard Pilocarpine prodrugs

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4061722A (en) 1976-04-26 1977-12-06 Interx Research Corporation Selected quaternary ammonium salts of pilocarpine useful in reducing intraocular pressure in warm-blooded animals
EP0106541A2 (en) 1982-09-17 1984-04-25 Hans Bundgaard Pilocarpine prodrugs

Also Published As

Publication number Publication date
FI922518A0 (fi) 1992-05-29
FI98910C (fi) 1997-09-10
FI922518A (fi) 1993-11-30
FI98910B (fi) 1997-05-30
LTIP576A (en) 1994-06-15

Similar Documents

Publication Publication Date Title
KR100858464B1 (ko) 콤브레타스타틴 a-4 인산염 프로드럭 모노- 및 디-유기아민 염, 모노- 및 디-아미노산 염, 그리고 모노- 및디-아미노산 에스테르 염
TW201240662A (en) Ester pro-drugs of [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl] methanol for treating retinal diseases
US20100093770A1 (en) Therapeutic agent for glaucoma containing adenosine derivative as active ingredient
CN105849117B (zh) Na,K‑ATP酶的α2亚型的选择性抑制剂和用于降低眼内压的用途
EP0087378B1 (fr) Ethers-oximes d'alcoylaminoalcools comme médicaments, produits nouveaux et procédés pour leur préparation
JP2016056207A (ja) プロスタグランジンアゴニストのプロドラッグの安定した水性組成物およびその使用方法
RU2100352C1 (ru) Производные сложного эфира биспилокарпиновой кислоты и способы их получения
LT3081B (en) Novel pilocarpine derivatives and process for their preparation
US20090186857A1 (en) Combretastatin A-4 Phosphate Prodrug Mono- and Di- Organic Amine Salts, Mono- and Di- Amino Acid Salts, and Mono- and Di- Amino Acid Ester Salts
RU2276138C2 (ru) Вещество, обладающее антиоксидантной, геропротекторной и противоишемической активностью, и способ его получения
HUT61002A (en) Process for producing 2-aminopyrimdine-4-carboxamide derivatives and pharmaceutical compositions comprising such compounds
TW202114981A (zh) Trpv1激動劑及其製備方法和用途
LV10257B (en) Novel pilocarpine derivatives and process for their preparation
US5436350A (en) Bispilocarpic acid ester derivatives and process for their preparation
CN113710320A (zh) 硫辛酸前药
JP3094474B2 (ja) イソキノリノン誘導体とその製造方法
EP4159209A1 (en) Sulfur-containing compound useful for treating or preventing presbyopia
BRPI0910391A2 (pt) Compostos moduladores do receptor prostaciclina (pgi2), forma cristalina dos referidos compostos, composição farmacêutica, usos dos mesmos e processo para preparação da referida composição
CZ20003126A3 (cs) Deriváty indolu a farmaceutické prostředky, které je obsahují

Legal Events

Date Code Title Description
PC9A Transfer of patents

Free format text: SANTEN OY,NIITTYHAANKATU 20, FIN-33720 TAMPERE,FI,971017

MM9A Lapsed patents

Effective date: 19990528