KR920005494B1 - 치환된 아자비사이클로헵탄의 제조방법 - Google Patents

치환된 아자비사이클로헵탄의 제조방법 Download PDF

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Publication number
KR920005494B1
KR920005494B1 KR1019850004322A KR850004322A KR920005494B1 KR 920005494 B1 KR920005494 B1 KR 920005494B1 KR 1019850004322 A KR1019850004322 A KR 1019850004322A KR 850004322 A KR850004322 A KR 850004322A KR 920005494 B1 KR920005494 B1 KR 920005494B1
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KR
South Korea
Prior art keywords
formula
group
hydrogen
lower alkyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019850004322A
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English (en)
Korean (ko)
Other versions
KR860000265A (ko
Inventor
알더 알렉스
스타네크 야로슬라브
벨루스 다니엘
Original Assignee
시바-가이기 에이지
아놀트 자일러, 에른스트 알테르
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Publication date
Application filed by 시바-가이기 에이지, 아놀트 자일러, 에른스트 알테르 filed Critical 시바-가이기 에이지
Publication of KR860000265A publication Critical patent/KR860000265A/ko
Application granted granted Critical
Publication of KR920005494B1 publication Critical patent/KR920005494B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/08—Oxygen atoms
    • C07D223/10—Oxygen atoms attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Indole Compounds (AREA)
KR1019850004322A 1984-06-20 1985-06-19 치환된 아자비사이클로헵탄의 제조방법 Expired KR920005494B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH298784 1984-06-20
CH2987/84-7 1984-06-20

Publications (2)

Publication Number Publication Date
KR860000265A KR860000265A (ko) 1986-01-27
KR920005494B1 true KR920005494B1 (ko) 1992-07-06

Family

ID=4246108

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019850004322A Expired KR920005494B1 (ko) 1984-06-20 1985-06-19 치환된 아자비사이클로헵탄의 제조방법

Country Status (20)

Country Link
US (3) US4677129A (enExample)
EP (1) EP0166692B1 (enExample)
JP (1) JPH0625127B2 (enExample)
KR (1) KR920005494B1 (enExample)
AT (1) ATE54446T1 (enExample)
AU (1) AU584098B2 (enExample)
DD (2) DD234419A5 (enExample)
DE (1) DE3578608D1 (enExample)
DK (1) DK164052C (enExample)
ES (4) ES8801261A1 (enExample)
FI (1) FI83214C (enExample)
GR (1) GR851498B (enExample)
HU (2) HU192231B (enExample)
IE (1) IE58069B1 (enExample)
IL (1) IL75545A0 (enExample)
NO (1) NO166444C (enExample)
NZ (1) NZ212482A (enExample)
PH (1) PH21957A (enExample)
PT (1) PT80659B (enExample)
ZA (1) ZA854613B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3378208D1 (en) * 1982-12-21 1988-11-17 Ciba Geigy Ag Substituted azabicycloalkanes, their use, pharmaceutical preparations containing these compounds and process for preparing these compounds
EP0166692B1 (de) * 1984-06-20 1990-07-11 Ciba-Geigy Ag Substituierte Azabicycloheptane, ihre Verwendung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verfahren zur Herstellung dieser Verbindungen
US4883877A (en) * 1987-11-13 1989-11-28 Ciba-Geigy Corporation Azabicycloheptanes and process for their preparation
DE3843481A1 (de) * 1988-12-23 1990-06-28 Boehringer Ingelheim Kg Substituierte 3-azabicyclo/3.1.1/heptane, ihre herstellung und ihre verwendung
CH683151A5 (de) * 1991-04-24 1994-01-31 Ciba Geigy Ag Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.
JP3170798B2 (ja) 1991-05-14 2001-05-28 セイコーエプソン株式会社 画像形成装置

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE548074A (enExample) *
US2673205A (en) * 1951-02-13 1954-03-23 Ciba Pharm Prod Inc 3-disubstituted dioxopiperidines and the manufacture thereof
DE1088957B (de) * 1955-07-18 1960-09-15 Ciba Geigy Verfahren zur Herstellung von ª‡-(p-Amino-phenyl)-ª‡-alkyl-glutarimiden
US2848455A (en) * 1955-07-18 1958-08-19 Ciba Pharm Prod Inc Alpha-(p-amino-phenyl)-alpha-lower alkyl glutarimides
GB1015618A (en) * 1962-04-10 1966-01-05 Aspro Nicholas Ltd Glutarimide therapeutic compositions
DE1299617B (de) * 1965-01-13 1969-07-24 Degussa Verfahren zur Herstellung von feinverteiltem gefaelltem Siliciumdioxid
US4231935A (en) * 1975-07-31 1980-11-04 American Cyanamid Company 1-Phenyl-3-azabicyclo[3.1.0]hexanes
US4131611A (en) * 1975-07-31 1978-12-26 American Cyanamid Company Azabicyclohexanes
US4435419A (en) * 1981-07-01 1984-03-06 American Cyanamid Company Method of treating depression using azabicyclohexanes
DE3378208D1 (en) * 1982-12-21 1988-11-17 Ciba Geigy Ag Substituted azabicycloalkanes, their use, pharmaceutical preparations containing these compounds and process for preparing these compounds
EP0166692B1 (de) * 1984-06-20 1990-07-11 Ciba-Geigy Ag Substituierte Azabicycloheptane, ihre Verwendung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verfahren zur Herstellung dieser Verbindungen

Also Published As

Publication number Publication date
EP0166692A3 (en) 1986-11-12
FI852429L (fi) 1985-12-21
AU4385885A (en) 1986-01-02
US4764640A (en) 1988-08-16
DK277485D0 (da) 1985-06-19
HU194180B (en) 1988-01-28
US4857660A (en) 1989-08-15
DK164052C (da) 1992-09-28
PT80659B (en) 1987-05-04
ES8801261A1 (es) 1987-12-16
FI83214C (fi) 1991-06-10
ATE54446T1 (de) 1990-07-15
FI83214B (fi) 1991-02-28
DK277485A (da) 1985-12-21
JPS6112666A (ja) 1986-01-21
ES557123A0 (es) 1987-12-16
HUT38346A (en) 1986-05-28
ZA854613B (en) 1986-02-26
EP0166692A2 (de) 1986-01-02
NZ212482A (en) 1988-08-30
JPH0625127B2 (ja) 1994-04-06
FI852429A0 (fi) 1985-06-19
ES557121A0 (es) 1988-01-01
IE851519L (en) 1985-12-20
ES544319A0 (es) 1987-12-16
DE3578608D1 (de) 1990-08-16
DD245871A5 (de) 1987-05-20
ES8802388A1 (es) 1988-05-16
NO852478L (no) 1985-12-23
ES557122A0 (es) 1988-05-16
DD234419A5 (de) 1986-04-02
ES8801278A1 (es) 1987-12-16
ES8801214A1 (es) 1988-01-01
US4677129A (en) 1987-06-30
IL75545A0 (en) 1985-10-31
NO166444B (no) 1991-04-15
GR851498B (enExample) 1985-11-25
KR860000265A (ko) 1986-01-27
NO166444C (no) 1991-08-07
DK164052B (da) 1992-05-04
AU584098B2 (en) 1989-05-18
EP0166692B1 (de) 1990-07-11
IE58069B1 (en) 1993-06-30
HU192231B (en) 1987-05-28
PT80659A (en) 1985-07-01
PH21957A (en) 1988-04-15

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