KR910000417B1 - 1,7-디하이드로-피롤로[3,4-e][1,4]디아제핀-2(3H)-온 유도체의 제조방법 - Google Patents

1,7-디하이드로-피롤로[3,4-e][1,4]디아제핀-2(3H)-온 유도체의 제조방법 Download PDF

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Publication number
KR910000417B1
KR910000417B1 KR1019830004230A KR830004230A KR910000417B1 KR 910000417 B1 KR910000417 B1 KR 910000417B1 KR 1019830004230 A KR1019830004230 A KR 1019830004230A KR 830004230 A KR830004230 A KR 830004230A KR 910000417 B1 KR910000417 B1 KR 910000417B1
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KR
South Korea
Prior art keywords
methyl
hydrogen
compound
formula
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019830004230A
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English (en)
Korean (ko)
Other versions
KR840006248A (ko
Inventor
마리아니 루이지
탈지아 지오지오
Original Assignee
그루포 레페티드 에스. 피. 에이
엘다 드 칼리
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by 그루포 레페티드 에스. 피. 에이, 엘다 드 칼리 filed Critical 그루포 레페티드 에스. 피. 에이
Publication of KR840006248A publication Critical patent/KR840006248A/ko
Application granted granted Critical
Publication of KR910000417B1 publication Critical patent/KR910000417B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
KR1019830004230A 1982-09-08 1983-09-08 1,7-디하이드로-피롤로[3,4-e][1,4]디아제핀-2(3H)-온 유도체의 제조방법 Expired KR910000417B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8225582 1982-09-08
GB8225582 1982-09-08

Publications (2)

Publication Number Publication Date
KR840006248A KR840006248A (ko) 1984-11-22
KR910000417B1 true KR910000417B1 (ko) 1991-01-25

Family

ID=10532762

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019830004230A Expired KR910000417B1 (ko) 1982-09-08 1983-09-08 1,7-디하이드로-피롤로[3,4-e][1,4]디아제핀-2(3H)-온 유도체의 제조방법

Country Status (14)

Country Link
US (1) US4508730A (https=)
EP (1) EP0102602B1 (https=)
JP (1) JPS5965093A (https=)
KR (1) KR910000417B1 (https=)
AT (1) ATE51230T1 (https=)
AU (1) AU566404B2 (https=)
CA (1) CA1199633A (https=)
DE (1) DE3381355D1 (https=)
DK (1) DK161077C (https=)
ES (2) ES8503000A1 (https=)
GR (1) GR79626B (https=)
IE (1) IE56043B1 (https=)
IL (1) IL69473A (https=)
ZA (1) ZA835899B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60208488A (ja) * 1984-04-03 1985-10-21 Nippon Mining Co Ltd スラグからの有価金属の回収法
WO2014128111A1 (de) 2013-02-22 2014-08-28 Bayer Pharma Aktiengesellschaft 4-substituierte pyrrolo- und pyrazolo-diazepine
EP2958922A1 (de) 2013-02-22 2015-12-30 Bayer Pharma Aktiengesellschaft Pyrrolo- und pyrazolo-triazolodiazepine als bet-proteininhibitoren zur behandlung von hyper-proliferativen erkrankungen

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3553210A (en) * 1968-12-16 1971-01-05 Parke Davis & Co 3-methyl-8-phenylpyrazolo(4,3-e)(1,4)diazepin-5(1h)-one, 7-oxide compounds
US3553207A (en) * 1968-12-16 1971-01-05 Parke Davis & Co Phenylpyrazolodiazepinone compounds
GB1433103A (en) * 1974-03-20 1976-04-22 Lepetit Spa Pharmacologically active pyrrolodiazepines
GR76455B (https=) * 1981-06-04 1984-08-10 Lepetit Spa
IT1167788B (it) * 1981-06-08 1987-05-13 Lepetit Spa Derivati pirrolo-diazepinici

Also Published As

Publication number Publication date
AU1790083A (en) 1984-03-15
DK394483D0 (da) 1983-08-30
JPH0447672B2 (https=) 1992-08-04
ES532487A0 (es) 1985-09-01
ES525442A0 (es) 1985-02-01
KR840006248A (ko) 1984-11-22
EP0102602A1 (en) 1984-03-14
IE832098L (en) 1984-03-08
AU566404B2 (en) 1987-10-22
ZA835899B (en) 1984-07-25
IE56043B1 (en) 1991-03-27
GR79626B (https=) 1984-10-31
US4508730A (en) 1985-04-02
CA1199633A (en) 1986-01-21
DK161077C (da) 1991-11-18
DK161077B (da) 1991-05-27
ES8503000A1 (es) 1985-02-01
IL69473A0 (en) 1983-11-30
ATE51230T1 (de) 1990-04-15
EP0102602B1 (en) 1990-03-21
IL69473A (en) 1985-12-31
DK394483A (da) 1984-03-09
ES8507551A1 (es) 1985-09-01
JPS5965093A (ja) 1984-04-13
DE3381355D1 (de) 1990-04-26

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