KR880007520A - 카바모일이미다졸 유도체, 이의 제조방법 및 살진균제로서의 이의 용도 - Google Patents

카바모일이미다졸 유도체, 이의 제조방법 및 살진균제로서의 이의 용도 Download PDF

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KR880007520A
KR880007520A KR870013692A KR870013692A KR880007520A KR 880007520 A KR880007520 A KR 880007520A KR 870013692 A KR870013692 A KR 870013692A KR 870013692 A KR870013692 A KR 870013692A KR 880007520 A KR880007520 A KR 880007520A
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alkyl
compound
phenyl
halo
formula
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KR870013692A
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에르하르트 하인쯔
밀덴베르거 힐마
마이어 토마스
샬러 라이너
쟈크세 부르크하르트
브라운 페터
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하인리히 벡커, 베른하르트 베크
휄스트 아크리엔게젤샤프트
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Publication of KR880007520A publication Critical patent/KR880007520A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

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  • Life Sciences & Earth Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
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Abstract

내용 없음.

Description

카바모일이미다졸 유도체, 이의 제조 방법 및 살진균제로서의 이의 용도
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (6)

  1. 일반식(Ⅰ)의 화합물 및 이의 금속염착 화합물.
    상기식에서, n은 2,3,4,5 또는 6이고, m은 1 또는 2 이며, R은 또는 -CH2CH2CH2OR1이고, R1은 (C1-C10)-알킬 또는 (C3-C10)-알케닐 [이들은 1 내지 6개의 불소, 염소 또는 브롬 원자, 히드록실, (C1-C4)-알콕시, 페닐 또는 페녹시(마지막으로 언급한 두 치환체인 페닐 또는 페녹시는 비치환되거나, 할로겐, (C1-C4)-알킬또는 (C1-C4)-알콕시에 의해 치환된다)에 의해 치환될 수 있다] : 또는 C3-알키닐, (C3-C6)-사이클로알킬, (C5-C6)-사이클로알케닐, 페닐, 벤질, 벤조히드릴, 트리딜, 비페닐, 페녹시 페닐, 페닐티오페닐, 나프틸, 1,2,3,4-테트라히드로 나프틸, 인다닐, 플뤄오레닐, 피리딘, 벤조티아졸릴, 벤즈옥사졸릴, 퀴놀리닐, 티오크로마닐, 벤조푸라닐 메틸, 퀴놀리닐메틸 또는 펜아실(여기서, 언급된 환 시스템은 비치환되거나, 할로겐, (C1-C8)-알킬, 할로(C1-C8)알킬, (C3-C8)-사이클로알킬, (C1-C8)-알킬시, 할로(C1-C8)-알콕시, (C3-C8)-사이클로알킬-(C1-C4)알킬, (C1-C8)알킬티오, 할로(C1-C4)알킬티오, (C1-C8)알킬설피닐, (C1-C8)알킬설포닐, NO2, -CN, -CHO 및 (C1-C4)알킬카보닐로 이루어진 그룹으로부터 선택된 1 내지 5개의 치환체에 의해 치환된다) : 또는 (C4-C10)-알카디에닐이며, R2는 H 또는 (C1-C4)알킬이고, Y는 서로 독립적으로 H, (C1-C4)알킬, 페닐 또는 할로페닐이다.
  2. 제1항에 있어서, Y가 H이고, n이 4 또는 5이며, m이 1이고, R이 OR1, CH2OR1또는 CH2CH2OR1이며, R1이 페닐, 벤질, 벤조히드릴, 비페닐, 피리딜 또는 퀴놀릴(여기서, 언급된 환 시스템은 비치환되거나, F, Cl, Br,(C1-C3)-알킬, 할로(C1-C3)알킬, (C1-C3)-알콕시, 할로(C1-C3)알콕시, (C1-C3)-알킬티오, CF3S, CF3CH2S, NO2, CN, CHO 및 -COCH3로 이루어진 그룹으로부터 선택된 1 내지 3개의 치환체에 의해 치환된다)인 일반식(Ⅰ)의 화합물 및 이의 금속염 착화합물.
  3. a) 일반식(Ⅱ)의 화합물을 일반식(Ⅲ)의 N, N′-카보닐디이미다졸과 반응시키거나, b) 일반식(Ⅳ)의 화합물을 일반식(V)의 이미다졸 화합물과 반응시키고, 수득된 화합물을, 경우에 따라, 금속 착화합물로 전환시킴을 특징으로 하여 제1항 또는 제2항에서 청구한 일반식(Ⅰ)의 화합물 및 이의 금속염 착화합물을 제조하는 방법.
    상기식에서, n·m·R·R1·R2및 Y는 제1항에서 정의한 바와 같고, M은 알칼리 금속이다.
  4. 제1항 또는 제2항에 따르는 일반식(Ⅰ)의 화합물을 함유하는 살진균제.
  5. 해로운 진균을 퇴치하기 위한 일반식(Ⅰ)의 화합물의 용도.
  6. 제1항 또는 제2항에 따르는 일반식(Ⅰ)의 화합물의 유효량을 해로운 진균, 보호할 식물, 경작지 또는 기질에 적용하여 해로운 진균을 퇴치하는 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR870013692A 1986-12-03 1987-12-02 카바모일이미다졸 유도체, 이의 제조방법 및 살진균제로서의 이의 용도 KR880007520A (ko)

Applications Claiming Priority (2)

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DE19863641343 DE3641343A1 (de) 1986-12-03 1986-12-03 Carbamoylimidazol-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
DEP3641343.7 1986-12-03

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KR880007520A true KR880007520A (ko) 1988-08-27

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US (1) US4889864A (ko)
EP (1) EP0270074A3 (ko)
JP (1) JPS63145277A (ko)
KR (1) KR880007520A (ko)
CN (1) CN87108072A (ko)
AU (1) AU598066B2 (ko)
BR (1) BR8706535A (ko)
CS (1) CS269997B2 (ko)
DD (1) DD264607A5 (ko)
DE (1) DE3641343A1 (ko)
DK (1) DK633287A (ko)
HU (1) HU201052B (ko)
IE (1) IE873280L (ko)
IL (1) IL84663A0 (ko)
PL (1) PL269186A1 (ko)
PT (1) PT86271B (ko)
ZA (1) ZA879043B (ko)

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KR20020012116A (ko) * 2000-08-05 2002-02-15 주정호 항암제로서 유용한 이미다졸릴우레아 유도체 및 그의제조방법

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JPH0710862B2 (ja) * 1989-08-08 1995-02-08 宇部興産株式会社 アゾリジン誘導体、その製法及び農園芸用殺菌剤
EP0449445A3 (en) * 1990-03-27 1993-08-25 Pfizer Inc. Preparation of beta-ketoesters useful in preparing quinolone antibiotics
US5629325A (en) * 1996-06-06 1997-05-13 Abbott Laboratories 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission
US6437138B1 (en) 1996-06-06 2002-08-20 Abbott Laboratories 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission
US20040192673A1 (en) * 2001-05-05 2004-09-30 Pascale Gaillard N-aroyl cyclic amine derivatives as orexin receptor antagonists
AU2002332659A1 (en) * 2001-08-21 2003-03-03 Sepracor, Inc. 2-substituted piperidines that are ligands for monoamine receptors and transporters
WO2011058766A1 (en) * 2009-11-16 2011-05-19 Raqualia Pharma Inc. Aryl carboxamide derivatives as ttx-s blockers
US9545105B2 (en) 2010-10-21 2017-01-17 Bayer Intellectual Property Gmbh 1-(heterocyclic carbonyl) piperidines
US8614242B2 (en) 2010-10-21 2013-12-24 Bayer Intellectual Property Gmbh 1-(heterocyclic carbonyl)-2-substituted pyrrolidines
CN104245687B (zh) 2012-04-12 2016-12-14 拜尔农科股份公司 作为杀真菌剂的n-酰基-2-(环)烷基吡咯烷和哌啶
WO2014176142A1 (en) * 2013-04-23 2014-10-30 Merck Sharp & Dohme Corp. Hydroxy-substituted orexin receptor antagonists

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GB1567521A (en) * 1977-03-26 1980-05-14 Boots Co Ltd Funigicidal complexes of metal salts with imidazoles
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JPS61227506A (ja) * 1985-04-01 1986-10-09 Nippon Tokushu Noyaku Seizo Kk カルバモイルイミダゾ−ル類、その中間体、それらの製法並びに除草剤又は農園芸用殺菌剤

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20020012116A (ko) * 2000-08-05 2002-02-15 주정호 항암제로서 유용한 이미다졸릴우레아 유도체 및 그의제조방법

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AU598066B2 (en) 1990-06-14
IE873280L (en) 1988-06-03
CS872487A2 (en) 1989-09-12
EP0270074A2 (de) 1988-06-08
ZA879043B (en) 1988-05-26
DD264607A5 (de) 1989-02-08
AU8198987A (en) 1988-06-09
JPS63145277A (ja) 1988-06-17
CS269997B2 (en) 1990-05-14
DE3641343A1 (de) 1988-06-16
EP0270074A3 (de) 1989-07-26
US4889864A (en) 1989-12-26
HU201052B (en) 1990-09-28
HUT46688A (en) 1988-11-28
PT86271A (en) 1988-01-01
DK633287D0 (da) 1987-12-02
DK633287A (da) 1988-06-04
IL84663A0 (en) 1988-05-31
PT86271B (pt) 1990-11-07
CN87108072A (zh) 1988-08-10
PL269186A1 (en) 1989-03-20
BR8706535A (pt) 1988-07-12

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