KR860001492B1 - 트랜스-4aR-5-n-프로필-4,4a,5,6,7,8,,8a,9-옥타하이드로-1H(및 2H) 피라졸로 [3,4-g] 퀴놀린의 제조방법 - Google Patents

트랜스-4aR-5-n-프로필-4,4a,5,6,7,8,,8a,9-옥타하이드로-1H(및 2H) 피라졸로 [3,4-g] 퀴놀린의 제조방법 Download PDF

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Publication number
KR860001492B1
KR860001492B1 KR1019830003502A KR830003502A KR860001492B1 KR 860001492 B1 KR860001492 B1 KR 860001492B1 KR 1019830003502 A KR1019830003502 A KR 1019830003502A KR 830003502 A KR830003502 A KR 830003502A KR 860001492 B1 KR860001492 B1 KR 860001492B1
Authority
KR
South Korea
Prior art keywords
trans
propyl
quinoline
octahydro
pyrazolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019830003502A
Other languages
English (en)
Korean (ko)
Other versions
KR840006654A (ko
Inventor
알렌 한 리챠드
다니엘 티터스 로버트
칼 콘펠드 에드먼드
Original Assignee
일라이 릴리 앤드 캄파니
아더 알. 웨일
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/438,833 external-priority patent/US4468401A/en
Application filed by 일라이 릴리 앤드 캄파니, 아더 알. 웨일 filed Critical 일라이 릴리 앤드 캄파니
Publication of KR840006654A publication Critical patent/KR840006654A/ko
Application granted granted Critical
Publication of KR860001492B1 publication Critical patent/KR860001492B1/ko
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1019830003502A 1982-11-03 1983-07-27 트랜스-4aR-5-n-프로필-4,4a,5,6,7,8,,8a,9-옥타하이드로-1H(및 2H) 피라졸로 [3,4-g] 퀴놀린의 제조방법 Expired KR860001492B1 (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US43923882A 1982-11-03 1982-11-03
US06/438,833 US4468401A (en) 1982-11-03 1982-11-03 Method of blocking peripheral norepinephrine release
US439238 1982-11-03
US439,238 1982-11-03
US438,833 1989-11-17
US438833 1989-11-17

Publications (2)

Publication Number Publication Date
KR840006654A KR840006654A (ko) 1984-12-01
KR860001492B1 true KR860001492B1 (ko) 1986-09-27

Family

ID=27031819

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019830003502A Expired KR860001492B1 (ko) 1982-11-03 1983-07-27 트랜스-4aR-5-n-프로필-4,4a,5,6,7,8,,8a,9-옥타하이드로-1H(및 2H) 피라졸로 [3,4-g] 퀴놀린의 제조방법

Country Status (16)

Country Link
EP (1) EP0111990B1 (enExample)
KR (1) KR860001492B1 (enExample)
AU (1) AU547185B2 (enExample)
CS (1) CS563283A2 (enExample)
DD (1) DD210044A5 (enExample)
DE (2) DE3327118A1 (enExample)
DK (1) DK343083A (enExample)
ES (1) ES8504174A1 (enExample)
FI (1) FI832718A7 (enExample)
GB (1) GB2129423B (enExample)
GR (1) GR79599B (enExample)
HU (1) HU189726B (enExample)
IL (1) IL69359A (enExample)
NZ (1) NZ205029A (enExample)
PL (1) PL243199A1 (enExample)
PT (1) PT77112A (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL72729A (en) * 1983-09-26 1988-02-29 Lilly Co Eli Trans(+_)octahydropyrazole-ring alkylated pyrazoloquinolines,their preparation and pharmaceutical compositions containing them
FI852975L (fi) * 1984-08-03 1986-02-04 Lilly Co Eli Tricykliska kinolinderivat.
US4762843A (en) * 1986-09-15 1988-08-09 Warner-Lambert Company Hetero [f] fused carbocyclic pyridines as dopaminergic agents

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4198415A (en) * 1979-01-22 1980-04-15 Eli Lilly And Company Prolactin inhibiting octahydro pyrazolo[3,4-g]quinolines

Also Published As

Publication number Publication date
ES524452A0 (es) 1985-04-16
FI832718L (fi) 1984-05-04
GB2129423B (en) 1986-05-29
EP0111990B1 (en) 1987-10-07
DD210044A5 (de) 1984-05-30
NZ205029A (en) 1985-08-30
AU1733883A (en) 1984-05-10
KR840006654A (ko) 1984-12-01
ES8504174A1 (es) 1985-04-16
EP0111990A1 (en) 1984-06-27
DE3374009D1 (en) 1987-11-12
DK343083A (da) 1984-05-04
GR79599B (enExample) 1984-10-31
DE3327118A1 (de) 1984-05-03
GB2129423A (en) 1984-05-16
PL243199A1 (en) 1984-08-13
CS563283A2 (en) 1985-07-16
PT77112A (en) 1983-08-01
IL69359A (en) 1986-09-30
AU547185B2 (en) 1985-10-10
HU189726B (en) 1986-07-28
FI832718A7 (fi) 1984-05-04
FI832718A0 (fi) 1983-07-27
GB8320250D0 (en) 1983-09-01
DK343083D0 (da) 1983-07-27

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Legal Events

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PA0109 Patent application

Patent event code: PA01091R01D

Comment text: Patent Application

Patent event date: 19830727

PA0201 Request for examination
PG1501 Laying open of application
PG1605 Publication of application before grant of patent

Comment text: Decision on Publication of Application

Patent event code: PG16051S01I

Patent event date: 19860830

E701 Decision to grant or registration of patent right
PE0701 Decision of registration

Patent event code: PE07011S01D

Comment text: Decision to Grant Registration

Patent event date: 19861206