KR20260053219A - 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법 - Google Patents

5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법

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Publication number
KR20260053219A
KR20260053219A KR1020257041103A KR20257041103A KR20260053219A KR 20260053219 A KR20260053219 A KR 20260053219A KR 1020257041103 A KR1020257041103 A KR 1020257041103A KR 20257041103 A KR20257041103 A KR 20257041103A KR 20260053219 A KR20260053219 A KR 20260053219A
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South Korea
Prior art keywords
decane
ethyl
azaspiro
oxa
piperazine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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KR1020257041103A
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English (en)
Korean (ko)
Inventor
다니엘 제이. 캐니
벤자민 이. 블라스
케빈 엠. 블래트너
더글라스 에이. 피핀
Original Assignee
템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션
프라이벤틱스 엘엘씨
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Application filed by 템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션, 프라이벤틱스 엘엘씨 filed Critical 템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션
Publication of KR20260053219A publication Critical patent/KR20260053219A/ko
Pending legal-status Critical Current

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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
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    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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KR1020257041103A 2016-11-15 2017-11-15 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법 Pending KR20260053219A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201662422344P 2016-11-15 2016-11-15
US62/422,344 2016-11-15
PCT/US2017/061677 WO2018093818A1 (en) 2016-11-15 2017-11-15 Novel modulators of the 5-hydroxytryptamine receptor 7 and their method of use
KR1020237034770A KR102900157B1 (ko) 2016-11-15 2017-11-15 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법

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KR20260053219A true KR20260053219A (ko) 2026-04-21

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KR1020257041103A Pending KR20260053219A (ko) 2016-11-15 2017-11-15 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법
KR1020237034770A Active KR102900157B1 (ko) 2016-11-15 2017-11-15 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법
KR1020197016744A Active KR102590403B1 (ko) 2016-11-15 2017-11-15 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법

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KR1020197016744A Active KR102590403B1 (ko) 2016-11-15 2017-11-15 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법

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US (4) US10858368B2 (enExample)
EP (2) EP3541790B1 (enExample)
JP (3) JP7107955B2 (enExample)
KR (3) KR20260053219A (enExample)
CN (2) CN110177776B (enExample)
AU (2) AU2017361078B2 (enExample)
CA (1) CA3043319A1 (enExample)
CL (1) CL2019001329A1 (enExample)
EA (1) EA201990915A1 (enExample)
ES (1) ES3050660T3 (enExample)
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WO (1) WO2018093818A1 (enExample)
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Families Citing this family (9)

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Publication number Priority date Publication date Assignee Title
WO2014164756A1 (en) 2013-03-11 2014-10-09 Temple University Of The Commonwealth System Of Higher Education Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use
EP3200589B1 (en) 2014-09-10 2026-03-11 Temple University Of The Commonwealth System Of Higher Education Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use
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