CN110177776B - 5-羟色胺受体7的新型调节剂及其使用方法 - Google Patents

5-羟色胺受体7的新型调节剂及其使用方法 Download PDF

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CN110177776B
CN110177776B CN201780079945.9A CN201780079945A CN110177776B CN 110177776 B CN110177776 B CN 110177776B CN 201780079945 A CN201780079945 A CN 201780079945A CN 110177776 B CN110177776 B CN 110177776B
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ethyl
azaspiro
oxa
piperazin
decan
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CN110177776A (zh
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D·J·坎尼
B·E·布拉斯
K·M·布拉特纳
D·A·皮平
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Plewetix Co ltd
Tempel University Commonwealth Higher Education System
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Tempel University Commonwealth Higher Education System
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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CN201780079945.9A 2016-11-15 2017-11-15 5-羟色胺受体7的新型调节剂及其使用方法 Active CN110177776B (zh)

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WO2014164756A1 (en) 2013-03-11 2014-10-09 Temple University Of The Commonwealth System Of Higher Education Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use
US10544117B2 (en) 2014-09-10 2020-01-28 Temple University—Of the Commonwealth System of Higher Education 5-hydroxytryptamine receptor 7 activity modulators and their method of use
CA3043319A1 (en) 2016-11-15 2018-05-24 Temple University-Of The Commonwealth System Of Higher Education Modulators of the 5-hydroxytryptamine receptor 7 and their method of use
US11220505B2 (en) * 2017-03-21 2022-01-11 Temple University-Of The Commonwealth System Of Higher Education 5-hydroxytryptamine receptor 7 modulators and their use as therapeutic agents
MA49019A (fr) * 2017-03-21 2020-02-05 Univ Temple Nouveaux modulateurs du récepteur sigma 2 et leur procédé d'utilisation
CN112437768B (zh) * 2018-05-11 2025-06-24 英联邦高等教育系统坦普尔大学 作为5-羟色胺受体7调节剂的新型官能化内酰胺及其使用方法
JP2023501576A (ja) * 2019-11-13 2023-01-18 テンプル・ユニバーシティ－オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクトンおよびその使用方法
US20230002383A1 (en) * 2019-11-13 2023-01-05 Temple University-Of The Commonwealth System Of Higher Education Novel functionalized lactams as modulators of the 5-hydroxytryptamine receptor 7 and their method of use
TW202328148A (zh) * 2021-09-22 2023-07-16 日商塩野義製藥股份有限公司 具有血清素受體結合活性之螺雜環衍生物

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