KR20210091139A - 피하 투여용 약제학적 제형 - Google Patents

피하 투여용 약제학적 제형 Download PDF

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Publication number
KR20210091139A
KR20210091139A KR1020217013385A KR20217013385A KR20210091139A KR 20210091139 A KR20210091139 A KR 20210091139A KR 1020217013385 A KR1020217013385 A KR 1020217013385A KR 20217013385 A KR20217013385 A KR 20217013385A KR 20210091139 A KR20210091139 A KR 20210091139A
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KR
South Korea
Prior art keywords
pharmaceutical composition
levodopa
liquid aqueous
stable liquid
carbidopa
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020217013385A
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English (en)
Korean (ko)
Inventor
에하브 무사
매튜 로제브라우
페로즈 자밀
낸시 세버
마우리지오 에프. 파셔리스
웨이닝 제트. 로비슨
찰스 에스. 록
스벤 슈토트만
Original Assignee
애브비 인코포레이티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 애브비 인코포레이티드 filed Critical 애브비 인코포레이티드
Publication of KR20210091139A publication Critical patent/KR20210091139A/ko
Ceased legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0021—Intradermal administration, e.g. through microneedle arrays or needleless injectors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020217013385A 2018-11-15 2019-11-15 피하 투여용 약제학적 제형 Ceased KR20210091139A (ko)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
US201862767546P 2018-11-15 2018-11-15
US62/767,546 2018-11-15
US201962843945P 2019-05-06 2019-05-06
US62/843,945 2019-05-06
US201962863093P 2019-06-18 2019-06-18
US201962863113P 2019-06-18 2019-06-18
US201962863101P 2019-06-18 2019-06-18
US62/863,113 2019-06-18
US62/863,093 2019-06-18
US62/863,101 2019-06-18
US201962898214P 2019-09-10 2019-09-10
US62/898,214 2019-09-10
PCT/US2019/061626 WO2020102628A1 (en) 2018-11-15 2019-11-15 Pharmaceutical formulations for subcutaneous administration

Publications (1)

Publication Number Publication Date
KR20210091139A true KR20210091139A (ko) 2021-07-21

Family

ID=68835352

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020217013385A Ceased KR20210091139A (ko) 2018-11-15 2019-11-15 피하 투여용 약제학적 제형

Country Status (14)

Country Link
US (3) US12251365B2 (https=)
EP (1) EP3880210A1 (https=)
JP (2) JP2022507528A (https=)
KR (1) KR20210091139A (https=)
CN (1) CN113015531A (https=)
AU (2) AU2019379806B2 (https=)
BR (1) BR112021009353A2 (https=)
CA (1) CA3117983A1 (https=)
IL (1) IL282842A (https=)
MX (1) MX2021005776A (https=)
SG (1) SG11202104499RA (https=)
TW (1) TW202031265A (https=)
UY (1) UY38473A (https=)
WO (1) WO2020102628A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021009353A2 (pt) 2018-11-15 2021-11-23 Abbvie Inc Formulações farmacêuticas para administração subcutânea
WO2023049534A2 (en) 2021-10-27 2023-03-30 Abbvie Inc. Subcutaneously administered treatments for advanced parkinson's disease

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Also Published As

Publication number Publication date
US20250186382A1 (en) 2025-06-12
US20250325507A1 (en) 2025-10-23
WO2020102628A1 (en) 2020-05-22
US20200155578A1 (en) 2020-05-21
EP3880210A1 (en) 2021-09-22
JP2024174894A (ja) 2024-12-17
UY38473A (es) 2020-06-30
US12251365B2 (en) 2025-03-18
MX2021005776A (es) 2021-07-02
JP2022507528A (ja) 2022-01-18
BR112021009353A2 (pt) 2021-11-23
IL282842A (en) 2021-06-30
AU2019379806A1 (en) 2021-05-27
AU2019379806B2 (en) 2025-08-14
CA3117983A1 (en) 2020-05-22
SG11202104499RA (en) 2021-05-28
TW202031265A (zh) 2020-09-01
AU2025256148A1 (en) 2025-11-13
CN113015531A (zh) 2021-06-22

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