IT1213182B - Derivati di composti a struttura catecolamminica. - Google Patents

Derivati di composti a struttura catecolamminica.

Info

Publication number
IT1213182B
IT1213182B IT8421583A IT2158384A IT1213182B IT 1213182 B IT1213182 B IT 1213182B IT 8421583 A IT8421583 A IT 8421583A IT 2158384 A IT2158384 A IT 2158384A IT 1213182 B IT1213182 B IT 1213182B
Authority
IT
Italy
Prior art keywords
compounds
derivatives
catecolaminical
effectiveness
disclosed
Prior art date
Application number
IT8421583A
Other languages
English (en)
Other versions
IT8421583A0 (it
Inventor
Cesare Casagrande
Francesco Santangelo
Original Assignee
Simes
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Simes filed Critical Simes
Publication of IT8421583A0 publication Critical patent/IT8421583A0/it
Priority to IT8421583A priority Critical patent/IT1213182B/it
Priority to AT85200986T priority patent/ATE46697T1/de
Priority to DE8585200986T priority patent/DE3573259D1/de
Priority to EP85200986A priority patent/EP0167204B1/en
Priority to ZA854745A priority patent/ZA854745B/xx
Priority to CA000485015A priority patent/CA1260464A/en
Priority to US06/748,587 priority patent/US4673671A/en
Priority to AU44128/85A priority patent/AU578294B2/en
Priority to JP60138839A priority patent/JP2520590B2/ja
Priority to ES545014A priority patent/ES8703483A1/es
Priority to FI852510A priority patent/FI83420C/fi
Application granted granted Critical
Publication of IT1213182B publication Critical patent/IT1213182B/it
Priority to MX9203207A priority patent/MX9203207A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/62Isoquinoline or hydrogenated isoquinoline ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/12Esters of phosphoric acids with hydroxyaryl compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/5532Seven-(or more) membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Liquid Crystal Substances (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
IT8421583A 1984-06-25 1984-06-25 Derivati di composti a struttura catecolamminica. IT1213182B (it)

Priority Applications (12)

Application Number Priority Date Filing Date Title
IT8421583A IT1213182B (it) 1984-06-25 1984-06-25 Derivati di composti a struttura catecolamminica.
AT85200986T ATE46697T1 (de) 1984-06-25 1985-06-20 Verfahren zur verbesserung der absorbierung und wirkung einer catecholaminverbindung.
DE8585200986T DE3573259D1 (en) 1984-06-25 1985-06-20 Method for improving the absorption and effectiveness of a catecholamine compound
EP85200986A EP0167204B1 (en) 1984-06-25 1985-06-20 Method for improving the absorption and effectiveness of a catecholamine compound
ZA854745A ZA854745B (en) 1984-06-25 1985-06-24 Method for improving the absorption and effectiveness of a catecholamine compound
CA000485015A CA1260464A (en) 1984-06-25 1985-06-24 Process for preparing a mono o-phosphate ester of catecholamine compound
US06/748,587 US4673671A (en) 1984-06-25 1985-06-25 Method for improving the absorption and effectiveness of a catecholamine compound
AU44128/85A AU578294B2 (en) 1984-06-25 1985-06-25 Catecholamine phosphates
JP60138839A JP2520590B2 (ja) 1984-06-25 1985-06-25 カテコ―ルアミン化合物のe/o―ホスフェ―トエステル,その製法およびそれを含有する薬剤組成物
ES545014A ES8703483A1 (es) 1984-06-25 1985-06-25 Procedimiento de preparar mono-o-fosfatoesteres de compues- tos de catecolamina
FI852510A FI83420C (fi) 1984-06-25 1985-06-25 Analogifoerfarande foer framstaellning av terapeutiskt anvaendbara mono-o-fosfatestrar av katekolaminer.
MX9203207A MX9203207A (es) 1984-06-25 1992-06-24 Compuesto de catecolamina y composicion farmaceutica que lo contiene.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8421583A IT1213182B (it) 1984-06-25 1984-06-25 Derivati di composti a struttura catecolamminica.

Publications (2)

Publication Number Publication Date
IT8421583A0 IT8421583A0 (it) 1984-06-25
IT1213182B true IT1213182B (it) 1989-12-14

Family

ID=11183927

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8421583A IT1213182B (it) 1984-06-25 1984-06-25 Derivati di composti a struttura catecolamminica.

Country Status (11)

Country Link
US (1) US4673671A (it)
EP (1) EP0167204B1 (it)
JP (1) JP2520590B2 (it)
AT (1) ATE46697T1 (it)
AU (1) AU578294B2 (it)
CA (1) CA1260464A (it)
DE (1) DE3573259D1 (it)
ES (1) ES8703483A1 (it)
FI (1) FI83420C (it)
IT (1) IT1213182B (it)
ZA (1) ZA854745B (it)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2070994T3 (es) * 1989-04-20 1995-06-16 Zambon Spa Profarmaco de dopamina.
IT1236843B (it) * 1989-11-22 1993-04-21 Simes Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati
IT1255471B (it) * 1992-07-30 1995-11-02 Zambon Spa Derivati di catecolammine,processo per la loro preparazione e composizioni farmaceutiche che li contengono
US6030961A (en) * 1997-03-11 2000-02-29 Bar-Ilan Research & Development Co., Ltd. Oxyalkylene phosphate compounds and uses thereof
HK1041703A1 (zh) * 1999-01-21 2002-07-19 Board Of Regents The University Of Texas System 肠道顶膜钠/磷酸盐共同传送的抑制剂
US6787044B1 (en) * 2003-03-10 2004-09-07 Archimedes Technology Group, Inc. High frequency wave heated plasma mass filter
JP4591045B2 (ja) 2004-11-08 2010-12-01 株式会社東京ベル製作所 ベル装置の打撃機構
RU2021103000A (ru) * 2014-10-21 2021-03-01 Эббви Инк. Пролекарства карбидопа и l-dopa и их применение для лечения болезни паркинсона
EP3880210A1 (en) 2018-11-15 2021-09-22 Abbvie Inc. Pharmaceutical formulations for subcutaneous administration
US12391650B2 (en) 2019-05-21 2025-08-19 H. Lundbeck A/S Catecholamine prodrugs for use in the treatment of Parkinson's disease
CN116256439B (zh) * 2021-12-10 2025-11-07 远大医药(中国)有限公司 Hplc检测盐酸多巴胺注射液中焦亚硫酸钠含量的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE557947A (it) * 1956-05-31
US3132171A (en) * 1962-06-18 1964-05-05 Strong Cobb Arner Inc 3, 4-diphosphatophenyl-alanine and process for making same
US3914343A (en) * 1973-07-20 1975-10-21 Warner Lambert Co Phosphoric acid esters of 5-(2-aminoethoxy)-carvacrols
FR2444043A1 (fr) * 1978-12-15 1980-07-11 Bottu Nouveau derive du paracetamol, son procede de preparation et son utilisation en therapeutique
US4508706A (en) * 1983-03-30 1985-04-02 Yale University Composition for increasing melanin in mammalian skin and hair

Also Published As

Publication number Publication date
ES545014A0 (es) 1987-03-01
EP0167204B1 (en) 1989-09-27
FI852510A0 (fi) 1985-06-25
ZA854745B (en) 1986-03-26
FI83420B (fi) 1991-03-28
CA1260464A (en) 1989-09-26
FI852510L (fi) 1985-12-26
JPS6183193A (ja) 1986-04-26
DE3573259D1 (en) 1989-11-02
AU4412885A (en) 1986-01-02
FI83420C (fi) 1991-07-10
JP2520590B2 (ja) 1996-07-31
IT8421583A0 (it) 1984-06-25
US4673671A (en) 1987-06-16
ATE46697T1 (de) 1989-10-15
EP0167204A1 (en) 1986-01-08
ES8703483A1 (es) 1987-03-01
AU578294B2 (en) 1988-10-20

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