IT1236843B - Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati - Google Patents

Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati

Info

Publication number
IT1236843B
IT1236843B IT02248689A IT2248689A IT1236843B IT 1236843 B IT1236843 B IT 1236843B IT 02248689 A IT02248689 A IT 02248689A IT 2248689 A IT2248689 A IT 2248689A IT 1236843 B IT1236843 B IT 1236843B
Authority
IT
Italy
Prior art keywords
dopamine
derivatives
phosphates
preparation
phosphate
Prior art date
Application number
IT02248689A
Other languages
English (en)
Other versions
IT8922486A0 (it
IT8922486A1 (it
Inventor
Cesare Casagrande
Francesco Santangelo
Original Assignee
Simes
Ora Simes Societa Italiana Med
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Simes, Ora Simes Societa Italiana Med filed Critical Simes
Publication of IT8922486A0 publication Critical patent/IT8922486A0/it
Priority to IT02248689A priority Critical patent/IT1236843B/it
Priority to US07/612,508 priority patent/US5138084A/en
Priority to AT90203034T priority patent/ATE118496T1/de
Priority to EP90203034A priority patent/EP0430336B1/en
Priority to DE69016946T priority patent/DE69016946T2/de
Priority to CA002030284A priority patent/CA2030284A1/en
Priority to FI905748A priority patent/FI905748A/fi
Priority to JP2315729A priority patent/JPH03176495A/ja
Publication of IT8922486A1 publication Critical patent/IT8922486A1/it
Application granted granted Critical
Publication of IT1236843B publication Critical patent/IT1236843B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/12Esters of phosphoric acids with hydroxyaryl compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Train Traffic Observation, Control, And Security (AREA)
IT02248689A 1989-11-22 1989-11-22 Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati IT1236843B (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IT02248689A IT1236843B (it) 1989-11-22 1989-11-22 Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati
US07/612,508 US5138084A (en) 1989-11-22 1990-11-14 Process for the preparation of 4-o-phosphates of dopamine and dopamine derivatives
DE69016946T DE69016946T2 (de) 1989-11-22 1990-11-15 Verfahren zur Herstellung von 4-O-Dopaminphosphaten und Dopaminderivate.
EP90203034A EP0430336B1 (en) 1989-11-22 1990-11-15 Process for the preparation of 4-O-phosphates of dopamine and dopamine derivatives
AT90203034T ATE118496T1 (de) 1989-11-22 1990-11-15 Verfahren zur herstellung von 4-o- dopaminphosphaten und dopaminderivate.
CA002030284A CA2030284A1 (en) 1989-11-22 1990-11-19 Process for the preparation of 4-0-phosphates of dopamine and dopamine derivatives
FI905748A FI905748A (fi) 1989-11-22 1990-11-21 Foerfarande foer framstaellning av 4-o -fosfater av dopamin och dopaminderivat.
JP2315729A JPH03176495A (ja) 1989-11-22 1990-11-22 ドーパミン及びドーパミン誘導体の4―0―リン酸エステルの製造方法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02248689A IT1236843B (it) 1989-11-22 1989-11-22 Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati

Publications (3)

Publication Number Publication Date
IT8922486A0 IT8922486A0 (it) 1989-11-22
IT8922486A1 IT8922486A1 (it) 1991-05-22
IT1236843B true IT1236843B (it) 1993-04-21

Family

ID=11196922

Family Applications (1)

Application Number Title Priority Date Filing Date
IT02248689A IT1236843B (it) 1989-11-22 1989-11-22 Processo per la preparazione di 4-0-fosfati di dopamina o suoi derivati

Country Status (8)

Country Link
US (1) US5138084A (it)
EP (1) EP0430336B1 (it)
JP (1) JPH03176495A (it)
AT (1) ATE118496T1 (it)
CA (1) CA2030284A1 (it)
DE (1) DE69016946T2 (it)
FI (1) FI905748A (it)
IT (1) IT1236843B (it)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPQ037499A0 (en) * 1999-05-14 1999-06-10 Swig Pty Ltd Improved process for phosphorylation and compounds produced by this method
MXPA01011597A (es) * 1999-05-14 2002-06-04 Swig Pty Ltd Proceso mejorado para la fosforilacion y compuestos producidos mediante este proceso.
US20040097472A1 (en) * 2000-11-14 2004-05-20 West Simon Michael Complexes of phosphate derivatives
AUPR549901A0 (en) 2001-06-06 2001-07-12 Vital Health Sciences Pty Ltd Topical formulation containing tocopheryl phosphates
CA2453823C (en) * 2001-07-27 2010-12-21 Vital Health Sciences Pty Ltd Dermal therapy using phosphate derivatives of electron transfer agents
WO2003049774A1 (en) * 2001-12-13 2003-06-19 Vital Health Sciences Pty Ltd Transdermal transport of compounds
AU2002950713A0 (en) * 2002-08-09 2002-09-12 Vital Health Sciences Pty Ltd Carrier
KR20050086954A (ko) * 2003-01-17 2005-08-30 바이탈 헬스 사이언시즈 피티와이 리미티드 항증식성 화합물
AU2003901815A0 (en) * 2003-04-15 2003-05-01 Vital Health Sciences Pty Ltd Phosphate derivatives
CA2557354C (en) * 2004-03-03 2013-05-07 Vital Health Sciences Pty Ltd. Alkaloid formulations
JP2008531602A (ja) * 2005-03-03 2008-08-14 バイタル ヘルス サイエンシズ プロプライアタリー リミティド 抗癌特性を有する化合物
US9168216B2 (en) * 2005-06-17 2015-10-27 Vital Health Sciences Pty. Ltd. Carrier comprising one or more di and/or mono-(electron transfer agent) phosphate derivatives or complexes thereof
EP1973547A1 (en) * 2005-12-23 2008-10-01 Vital Health Sciences Pty Ltd. Compounds having cytokine modulating properties
AU2011213557B2 (en) 2010-02-05 2015-05-07 Phosphagenics Limited Carrier comprising non-neutralised tocopheryl phosphate
BR112012024835A2 (pt) 2010-03-30 2016-06-07 Phosphagenics Ltd adesivo de distribuição transdérmica
WO2012122586A1 (en) 2011-03-15 2012-09-20 Phosphagenics Limited New composition
EP3383371B1 (en) 2015-12-09 2024-05-01 Avecho Biotechnology Limited Pharmaceutical formulation
CA3045702A1 (en) 2016-12-21 2018-06-28 Phosphagenics Limited Phosphorylation process of complex alcohols

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1213182B (it) * 1984-06-25 1989-12-14 Simes Derivati di composti a struttura catecolamminica.

Also Published As

Publication number Publication date
CA2030284A1 (en) 1991-05-23
EP0430336A3 (en) 1992-01-15
ATE118496T1 (de) 1995-03-15
DE69016946T2 (de) 1995-12-14
IT8922486A0 (it) 1989-11-22
EP0430336A2 (en) 1991-06-05
DE69016946D1 (de) 1995-03-23
FI905748A (fi) 1991-05-23
EP0430336B1 (en) 1995-02-15
JPH03176495A (ja) 1991-07-31
IT8922486A1 (it) 1991-05-22
FI905748A0 (fi) 1990-11-21
US5138084A (en) 1992-08-11

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19941103