KR20180095580A - H-pgds 억제제로서의 퀴놀린-3-카르복스아미드 - Google Patents

H-pgds 억제제로서의 퀴놀린-3-카르복스아미드 Download PDF

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KR20180095580A
KR20180095580A KR1020187019904A KR20187019904A KR20180095580A KR 20180095580 A KR20180095580 A KR 20180095580A KR 1020187019904 A KR1020187019904 A KR 1020187019904A KR 20187019904 A KR20187019904 A KR 20187019904A KR 20180095580 A KR20180095580 A KR 20180095580A
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carboxamide
quinoline
chloro
difluoromethoxy
trans
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Korean (ko)
Inventor
로돌포 캐딜라
데이브 노먼 대톤
애슐리 폴 핸콕
헤더 홉스
시몬 테안비 호지슨
앤드류 엘. 라킨
조엘 르
폴 엔. 모텐슨
대니얼 제이. 프라이스
고든 삭티
리 티. 샬러
크리스티 셜트
이안 에드워드 데이빗 스미쓰
스티븐 앤드류 톰슨
조셉 웬델 윌슨
Original Assignee
아스텍스 테라퓨틱스 리미티드
글락소스미스클라인 인털렉츄얼 프로퍼티 디벨로프먼트 리미티드
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Publication of KR20180095580A publication Critical patent/KR20180095580A/ko
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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020187019904A 2015-12-17 2016-12-15 H-pgds 억제제로서의 퀴놀린-3-카르복스아미드 Withdrawn KR20180095580A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562268630P 2015-12-17 2015-12-17
US62/268,630 2015-12-17
PCT/IB2016/057676 WO2017103851A1 (en) 2015-12-17 2016-12-15 Quinoline-3-carboxamides as h-pgds inhibitors

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KR20180095580A true KR20180095580A (ko) 2018-08-27

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US (1) US20210238162A1 (https=)
EP (1) EP3390384B1 (https=)
JP (1) JP2019502691A (https=)
KR (1) KR20180095580A (https=)
CN (1) CN108430992A (https=)
AR (1) AR107044A1 (https=)
AU (1) AU2016370779B2 (https=)
BR (1) BR112018012469B1 (https=)
CA (1) CA3008358A1 (https=)
RU (1) RU2018126105A (https=)
TW (1) TW201733988A (https=)
UY (1) UY37028A (https=)
WO (1) WO2017103851A1 (https=)

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JP7403472B2 (ja) 2018-05-09 2023-12-22 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング 新規キノリン誘導体
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