KR20170102050A - 알파-멜라노사이트 자극 호르몬의 펩티드 유사체 - Google Patents

알파-멜라노사이트 자극 호르몬의 펩티드 유사체 Download PDF

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Publication number
KR20170102050A
KR20170102050A KR1020177023883A KR20177023883A KR20170102050A KR 20170102050 A KR20170102050 A KR 20170102050A KR 1020177023883 A KR1020177023883 A KR 1020177023883A KR 20177023883 A KR20177023883 A KR 20177023883A KR 20170102050 A KR20170102050 A KR 20170102050A
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xaa
msh
ser
ala
peptide
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Korean (ko)
Inventor
마이클 에이. 페리콘
존 라일 드주리스
티모씨 이. 위든
제임스 이. 스테파노
클락 큐. 판
안드레아 이. 에들링
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젠자임 코포레이션
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/68—Melanocyte-stimulating hormone [MSH]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/68—Melanocyte-stimulating hormone [MSH]
    • C07K14/685—Alpha-melanotropin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/33—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • A61K38/34—Melanocyte stimulating hormone [MSH], e.g. alpha- or beta-melanotropin
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    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1021—Tetrapeptides with the first amino acid being acidic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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  • Engineering & Computer Science (AREA)
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  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
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  • Biochemistry (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Diabetes (AREA)
  • Toxicology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pathology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
KR1020177023883A 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체 Ceased KR20170102050A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5637308P 2008-05-27 2008-05-27
US61/056,373 2008-05-27
PCT/US2009/037809 WO2009151708A2 (en) 2008-05-27 2009-03-20 Peptide analogs of alpha-melanocyte stimulating hormone

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KR1020167020183A Division KR101810110B1 (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체

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KR1020187030624A Division KR20180118250A (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체

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KR1020177023883A Ceased KR20170102050A (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체
KR1020187030624A Ceased KR20180118250A (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체
KR1020167020183A Expired - Fee Related KR101810110B1 (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체
KR1020107029335A Expired - Fee Related KR101666631B1 (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체

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KR1020187030624A Ceased KR20180118250A (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체
KR1020167020183A Expired - Fee Related KR101810110B1 (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체
KR1020107029335A Expired - Fee Related KR101666631B1 (ko) 2008-05-27 2009-03-20 알파-멜라노사이트 자극 호르몬의 펩티드 유사체

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US (4) US8440793B2 (cg-RX-API-DMAC7.html)
EP (2) EP2816055B1 (cg-RX-API-DMAC7.html)
JP (4) JP5624027B2 (cg-RX-API-DMAC7.html)
KR (4) KR20170102050A (cg-RX-API-DMAC7.html)
CN (2) CN107098957A (cg-RX-API-DMAC7.html)
AU (1) AU2009258054B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0912141A2 (cg-RX-API-DMAC7.html)
CA (2) CA2998948A1 (cg-RX-API-DMAC7.html)
DK (2) DK2297178T3 (cg-RX-API-DMAC7.html)
ES (2) ES2715329T3 (cg-RX-API-DMAC7.html)
IL (3) IL209369A (cg-RX-API-DMAC7.html)
MX (3) MX356295B (cg-RX-API-DMAC7.html)
PT (2) PT2297178E (cg-RX-API-DMAC7.html)
RU (1) RU2496786C2 (cg-RX-API-DMAC7.html)
TR (1) TR201903610T4 (cg-RX-API-DMAC7.html)
WO (1) WO2009151708A2 (cg-RX-API-DMAC7.html)

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WO2012158960A2 (en) 2011-05-17 2012-11-22 H. Lee Moffitt Cancer Center & Research Institute, Inc. Melanocortin 1 receptor ligands and methods of use
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CN106905432B (zh) * 2015-12-18 2018-12-21 兰州大学 一种α促黑素细胞激素的融合蛋白及其制备方法和应用
EP3448872A4 (en) * 2016-04-27 2019-12-11 The Regents of the University of California PREPARATION OF FUNCTIONAL HOMOCYSTEINRESTES IN POLYPEPTIDES AND PEPTIDES
US20220072092A1 (en) * 2016-06-24 2022-03-10 University Of Iowa Research Foundation Compositions and methods of treating melanoma
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CN109803979B (zh) * 2016-10-04 2023-01-31 帝斯曼知识产权资产管理有限公司 黑皮质素-1-受体激动剂
KR101957014B1 (ko) * 2017-04-18 2019-06-20 순천대학교 산학협력단 항염증 활성을 나타내는 펩타이드 및 이를 유효성분으로 포함하는 항염증용 조성물
MX2022003446A (es) 2019-09-23 2022-07-13 Dds Res Inc Composiciones de vesiculas lipidicas con agentes potenciadores de la penetracion.
WO2021157973A1 (ko) * 2020-02-07 2021-08-12 이화여자대학교 산학협력단 페길화된 ige-의존적 히스타민 방출인자(hrf) 결합 펩타이드 및 이의 용도
US11529335B2 (en) 2020-07-31 2022-12-20 University Of Iowa Research Foundation Compositions and methods for treating cancer
RU2766340C1 (ru) * 2021-02-10 2022-03-15 Игорь Закванович Зайцев Пептидный толерогенный компаунд
MX2023011157A (es) 2021-03-24 2024-01-25 Glo Pharma Inc Peptidos y metodos para reducir la pigmentacion de la piel.
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